Betulin and ursolic acid synthetic derivatives as inhibitors of Papilloma virus

Bioorganic and Medicinal Chemistry Letters

Volumn 20, Issue 14, 2010, Pages 4088-4090

  Kazakova, Oxana B ^a   Giniyatullina, Gul'nara V ^a   Yamansarov, Emil Yu ^a   Tolstikov, Genrikh A ^a  

^a INSTITUTE OF ORGANIC CHEMISTRY   (Russian Federation)

Author keywords

Antiviral activity; Betulin; Triterpenoids; Ursolic acid

Indexed keywords

28 O METHOXYCYNNAMOYLBETULIN; 3BETA,28 DI O NICOTINOYLBETULIN; 3BETA,28 DIHYDROXY 29 NORLUP 20(30) YNE; BETULIN; IMIDE; TRITERPENOID; UNCLASSIFIED DRUG; URSOLIC ACID;

ANTIVIRAL ACTIVITY; ARTICLE; CYTOTOXICITY; DRUG SCREENING; DRUG SELECTIVITY; DRUG SYNTHESIS; HUMAN PAPILLOMAVIRUS TYPE 11; IC 50; IN VITRO STUDY; INFLUENZA VIRUS A H1N1; NONHUMAN; REPLICON; STRUCTURE ACTIVITY RELATION;

ANTIVIRAL AGENTS; MICROBIAL SENSITIVITY TESTS; PAPILLOMAVIRIDAE; TRITERPENES;

HEPATITIS C VIRUS; HUMAN PAPILLOMAVIRUS TYPE 11; PAPILLOMAVIRIDAE;

EID: 77953870088     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2010.05.083     Document Type: Article

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21. 4: C, 77.26; N{cyrillic}, 8.64; N, 4.29. Found: C, 77.03; H, 8.41; N, 4.05.
22. 4: C, 79.69; N{cyrillic}, 9.70. Found: C, 79.28; H, 9.84.
23. 4: C, 76.97; N{cyrillic}, 9.15; N, 2.49. Found: C, 77.08; H, 9.03; N, 2.29.
24. 2: C, 81.63; H, 10.87. Found: C, 81.44; H, 10.62.
25. 2: S{cyrillic}, 78.21; N{cyrillic}, 10.94; N, 5.07. Found: S{cyrillic}, 78.02; N{cyrillic}, 10.76; N, 4.83.
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