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Volumn 3, Issue 1, 2009, Pages 42-49

A high throughput assay to identify small molecule modulators of prostatic acid phosphatase

Author keywords

[No Author keywords available]

Indexed keywords

ACID PHOSPHATASE PROSTATE ISOENZYME; ANTINOCICEPTIVE AGENT; BAS 00669251; BAS 02830262; BAS 03013122; BAS 07119722; BAS 08862870; BAS 08863852; BAS 08865249; DIFLUORO 4 METHYLUMBELLIFERYL PHOSPHATE; DIMETHYL SULFOXIDE; ENZYME INHIBITOR; FLUORESCENT DYE; TARTARIC ACID; UNCLASSIFIED DRUG;

EID: 77953388445     PISSN: None     EISSN: 18753973     Source Type: Journal    
DOI: 10.2174/1875397300903010042     Document Type: Article
Times cited : (6)

References (15)
  • 1
    • 64149093214 scopus 로고    scopus 로고
    • Recombinant mouse PAP has pH-dependent ectonucleotidase activity and acts through A(1)-adenosine receptors to mediate antinociception
    • Sowa NA, Vadakkan KI, Zylka MJ. Recombinant mouse PAP has pH-dependent ectonucleotidase activity and acts through A(1)-adenosine receptors to mediate antinociception. PLoS ONE 2009; 4: e42-8.
    • (2009) PLoS ONE , vol.4
    • Sowa, N.A.1    Vadakkan, K.I.2    Zylka, M.J.3
  • 2
    • 53049093740 scopus 로고    scopus 로고
    • Prostatic acid phosphatase is an ectonucleotidase and suppresses pain by generating adenosine
    • Zylka MJ, Sowa NA, Taylor-Blake B, et al. Prostatic acid phosphatase is an ectonucleotidase and suppresses pain by generating adenosine. Neuron 2008; 60: 111-122
    • (2008) Neuron , vol.60 , pp. 111-122
    • Zylka, M.J.1    Sowa, N.A.2    Taylor-Blake, B.3
  • 4
    • 0030272641 scopus 로고    scopus 로고
    • Phosphatase inhibitors - III. Benzylaminophosphonic acids as potent inhibitors of human prostatic acid phosphatase
    • Beers SA, Schwender CF, Loughney DA, Malloy E, Demarest K, Jordan J. Phosphatase inhibitors - III. Benzylaminophosphonic acids as potent inhibitors of human prostatic acid phosphatase. Bioorg Med Chem 1996; 4: 1693-1701
    • (1996) Bioorg Med Chem , vol.4 , pp. 1693-1701
    • Beers, S.A.1    Schwender, C.F.2    Loughney, D.A.3    Malloy, E.4    Demarest, K.5    Jordan, J.6
  • 6
    • 0036942826 scopus 로고    scopus 로고
    • The obligatory action of protein tyrosine phosphatases in ACTH-stimulated steroidogenesis is exerted at the level of StAR protein
    • DOI 10.1081/ERC-120016816
    • Poderoso C, Maciel FC, Gorostizaga A, Bey P, Paz C, Podesta EJ. The obligatory action of protein tyrosine phosphatases in ACTH-stimulated steroidogenesis is exerted at the level of StAR protein. Endocr Res 2002; 28: 413-417 (Pubitemid 36042494)
    • (2002) Endocrine Research , vol.28 , Issue.4 , pp. 413-417
    • Poderoso, C.1    Cornejo Maciel, F.2    Gorostizaga, A.3    Bey, P.4    Paz, C.5    Podesta, E.J.6
  • 7
    • 0038350685 scopus 로고    scopus 로고
    • Tyrosine phosphorylation is involved in Ca(2+)entry in human gingival fibroblasts
    • Ogata Y, Nakao S, Shimizu E, et al. Tyrosine phosphorylation is involved in Ca(2+)entry in human gingival fibroblasts. Cell Biol Int 2003; 27: 689-693
    • (2003) Cell Biol Int , vol.27 , pp. 689-693
    • Ogata, Y.1    Nakao, S.2    Shimizu, E.3
  • 9
    • 0034651985 scopus 로고    scopus 로고
    • Crystal structure of human prostatic acid phosphatase
    • DOI 10.1002/(SICI)1097-0045(20000215)42:3<211::AID-PROS7>3.0.CO;2-U
    • Jakob CG, Lewinski K, Kuciel R, Ostrowski W, Lebioda L. Crystal structure of human prostatic acid phosphatase. Prostate 2000; 42: 211-218 (Pubitemid 30080420)
    • (2000) Prostate , vol.42 , Issue.3 , pp. 211-218
    • Jakob, C.G.1    Lewinski, K.2    Kuciel, R.3    Ostrowski, W.4    Lebioda, L.5
  • 10
    • 0037457813 scopus 로고    scopus 로고
    • Crystal structures of human prostatic acid phosphatase in complex with a phosphate ion and alpha-benzylaminobenzylphosphonic acid update the mechanistic picture and offer new insights into inhibitor design
    • DOI 10.1021/bi0265067
    • Ortlund E, LaCount MW, Lebioda L. Crystal structures of human prostatic acid phosphatase in complex with a phosphate ion and alpha- benzylaminobenzylphosphonic acid update the mechanistic picture and offer new insights into inhibitor design. Biochem 2003; 42: 383-389 (Pubitemid 36105756)
    • (2003) Biochemistry , vol.42 , Issue.2 , pp. 383-389
    • Ortlund, E.1    Lacount, M.W.2    Lebioda, L.3
  • 11
    • 0027201613 scopus 로고
    • Three-dimensional structure of rat acid phosphatase
    • Schneider G, Lindqvist Y, Vihko P. Three-dimensional structure of rat acid phosphatase. EMBO J 1993; 12: 2609-2615 (Pubitemid 23218309)
    • (1993) EMBO Journal , vol.12 , Issue.7 , pp. 2609-2615
    • Schneider, G.1    Lindqvist, Y.2    Vihko, P.3
  • 12
    • 0033566587 scopus 로고    scopus 로고
    • Fluorogenic substrates based on fluorinated umbelliferones for continuous assays of phosphatases and β-galactosidases
    • Gee KR, Sun WC, Bhalgat MK, et al. Fluorogenic substrates based on fluorinated umbelliferones for continuous assays of phosphatases and β-galactosidases. Anal Biochem 1999; 273: 41-48
    • (1999) Anal Biochem , vol.273 , pp. 41-48
    • Gee, K.R.1    Sun, W.C.2    Bhalgat, M.K.3
  • 13
    • 0033003760 scopus 로고    scopus 로고
    • A simple statistical parameter for use in evaluation and validation of high throughput screening assays
    • DOI 10.1177/108705719900400206
    • Zhang J, Thomas D, Chung Y, Oldenburg KR. A simple statistical parameter for use in evaluation and validation of high throughput screening assays. J Biomol Screen 1999; 4: 67-74. (Pubitemid 29278954)
    • (1999) Journal of Biomolecular Screening , vol.4 , Issue.2 , pp. 67-73
    • Zhang, J.-H.1    Chung, T.D.Y.2    Oldenburg, K.R.3
  • 14
    • 0032515075 scopus 로고    scopus 로고
    • Structural origins of L(+)-tartrate inhibition of human prostatic acid phosphatase
    • DOI 10.1074/jbc.273.46.30406
    • LaCount MW, Handy G, Lebioda L. Structural origins of L(+)-tartrate inhibition of human prostatic acid phosphatase. J Biol Chem 1998; 273: 30406-30409 (Pubitemid 28545512)
    • (1998) Journal of Biological Chemistry , vol.273 , Issue.46 , pp. 30406-30409
    • Lacount, M.W.1    Handy, G.2    Lebioda, L.3
  • 15
    • 0035336797 scopus 로고    scopus 로고
    • Simultaneous direct determination of amiloride and triamterene in urine using isopotential fluorometry
    • Pulgarin JAM, Molina AA, Lopez PF. Simultaneous direct determination of amiloride and triamterene in urine using isopotential fluorometry. Anal Biochem 2001; 292: 59-68.
    • (2001) Anal Biochem , vol.292 , pp. 59-68
    • Pulgarin, J.A.M.1    Molina, A.A.2    Lopez, P.F.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.