Two polymorphs of safinamide, a selective and reversible inhibitor of monoamine oxidase B

Acta Crystallographica Section C: Crystal Structure Communications

Volumn 66, Issue 6, 2010, Pages

  Ravikumar, Krishnan ^a   Sridhar, Balasubramanian ^a  

^a INDIAN INSTITUTE OF CHEMICAL TECHNOLOGY   (India)

Author keywords

[No Author keywords available]

Indexed keywords

ADJACENT LAYERS; HYDROGEN BONDINGS; MONOAMINE OXIDASE B;

AMINATION; HYDROGEN; POLYMORPHISM;

HYDROGEN BONDS;

ALANINE; BENZYLAMINE DERIVATIVE; DRUG DERIVATIVE; MONOAMINE OXIDASE INHIBITOR; SAFINAMIDE;

ARTICLE; CHEMISTRY; CRYSTALLIZATION; HYDROGEN BOND; X RAY CRYSTALLOGRAPHY;

ALANINE; BENZYLAMINES; CRYSTALLIZATION; CRYSTALLOGRAPHY, X-RAY; HYDROGEN BONDING; MONOAMINE OXIDASE INHIBITORS;

EID: 77953217765     PISSN: 01082701     EISSN: 01082701     Source Type: Journal    
DOI: 10.1107/S0108270110019384     Document Type: Article

References (15)

1. Berman, H. M., Westbrook, J., Feng, Z., Gilliland, G., Bhat, T. N., Weissig, H., Shindyalow, I. N. & Bourne, P. E. (2000). Nucleic Acids Res. 28, 235-242.
2. Bernstein, J., Davis, R. E., Shimoni, L. & Chang, N. L. (1995). Angew. Chem. Int. Ed. Engl. 34, 1555-1573.
3. Binda, C., Wang, J., Pisani, L., Caccia, C., Carotti, A., Salvati, P., Edmondson, D. E. & Mattevi, A. (2007). J. Med. Chem. 50, 5848-5852.
4. Brandenburg, K. & Putz, H. (2005). DIAMOND. Release 3.0c. Crystal Impact GbR, Bonn, Germany.
5. Bruker (2001). SAINT (Version 6.28a) and SMART (Version 5.625). Bruker AXS Inc., Madison, Wisconsin, USA.
6. Caccia, C., Maj, R., Calabresi, M., Maestroni, S., Faravelli, L., Curatolo, L., Salvati, P. & Fariello, R. G. (2006). Neurology, 67, S18-S23.
7. Etter, M. C. (1990). Acc. Chem. Res. 23, 120-126.
8. Etter, M. C., MacDonald, J. C. & Bernstein, J. (1990). Acta Cryst. B46, 256-262.
9. Grant, D. J. W. (1999). Theory and Origin of Polymorphism. Polymorphism in Pharmaceutical Solids, edited by H. G. Brittain, pp. 1-34. New York: Marcel Dekker Inc.
10. Macrae, C. F., Bruno, I. J., Chisholm, J. A., Edgington, P. R., McCabe, P., Pidcock, E., Rodriguez-Monge, L., Taylor, R., van de Streek, J. & Wood, P. A. (2008). J. Appl. Cryst. 41, 466-470.
11. Pevarello, P., Bonsignori, A., Dostert, P., Heidempergher, F., Pinciroli, V., Colombo, M., McArthur, R. A., Salvati, P., Post, C., Fariello, R. G. & Varasi, M. (1998). J. Med. Chem. 41, 579-590.
12. Ravikumar, K. & Sridhar, B. (2007). Acta Cryst. E63, o1404-o1406.
13. Ravikumar, K. & Sridhar, B. (2009). Acta Cryst. C65, o502-o505.
14. Ravikumar, K., Sridhar, B., Krishnan, H. & Singh, A. N. (2008). Acta Cryst. C64, o653-o656.
15. Sheldrick, G. M. (2008). Acta Cryst. A64, 112-122.