Aminocarnitine ureidic derivatives as inhibitors of carnitine palmitoyltransferase I

ChemMedChem

Volumn 5, Issue 5, 2010, Pages 666-669

  Tassoni, Emanuela ^a   Conti, Roberto ^a   Gallo, Grazia ^a   Vincenti, Silvia ^a   Dell'Uomo, Natalina ^a   Mastrofrancesco, Lucilla ^a   Ricciolini, Rita ^a   Cabri, Walter ^a   Carminati, Paolo ^a   Giannessi, Fabio ^a  

^a Sigma Tau SpA   (Italy)

Author keywords

Carnitine palmitoyltransferases; Carnitines; Inhibitors; Teglicar; Type II diabetes

Indexed keywords

ANTIDIABETIC AGENT; CARBOXYLIC ACID; CARNITINE ACETYLTRANSFERASE; CARNITINE PALMITOYLTRANSFERASE I; CARNITINE PALMITOYLTRANSFERASE INHIBITOR; EMERIAMINE; GLUCOSE; PHOSPHONIUM DERIVATIVE; ST 1326; TEGLICAR; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; CURTIUS REARRANGEMENT; DRUG ACTIVITY; DRUG EFFICACY; DRUG SELECTIVITY; DRUG SYNTHESIS; ENZYME INHIBITION; HUMAN; IN VITRO STUDY; IN VIVO STUDY; INSULIN RESISTANCE; INSULIN SENSITIVITY; MOUSE; NON INSULIN DEPENDENT DIABETES MELLITUS; NONHUMAN; PRIORITY JOURNAL; RAT;

ANIMALS; BETAINE; BINDING SITES; CARNITINE; CARNITINE O-PALMITOYLTRANSFERASE; COMPUTER SIMULATION; DIABETES MELLITUS, TYPE 2; ENZYME INHIBITORS; HYPOGLYCEMIC AGENTS; MICE; RATS;

EID: 77951691340     PISSN: 18607179     EISSN: 18607187     Source Type: Journal    
DOI: 10.1002/cmdc.200900535     Document Type: Article

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