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Volumn 8, Issue 9, 2010, Pages 2164-2173

Synthesis and biological evaluation of a triazole-based library of pyrido[2,3-d]pyrimidines as FGFR3 tyrosine kinase inhibitors

(10) Le Corre, Laurent a Girard, Anne Lise a Aubertin, Johannes b Radvanyi, Franois b Benoist Lasselin, Catherine a Jonquoy, Aurélie a Mugniery, Emilie a Legeai Mallet, Laurence a Busca, Patricia a Le Merrer, Yves a

a UNIVERSITÉ PARIS DESCARTES (France)

b INSTITUT CURIE (France)

Author keywords

[No Author keywords available]

Indexed keywords

ATP BINDING; AUTOPHOSPHORYLATION; BIOLOGICAL EVALUATION; CLICK CHEMISTRY; IN-VITRO; KINASE ACTIVITY; TYROSINE KINASE; TYROSINE KINASE INHIBITOR;

AMINO ACIDS; NITROGEN COMPOUNDS; PHOSPHORYLATION; SYNTHESIS (CHEMICAL);

PHOSPHATASES;

PROTEIN KINASE INHIBITOR; PROTEIN TYROSINE KINASE; PYRIDINE DERIVATIVE; PYRIMIDINE DERIVATIVE; RECOMBINANT PROTEIN; TRIAZOLE DERIVATIVE;

ARTICLE; BINDING SITE; CELL LINE; CHEMICAL STRUCTURE; CHEMISTRY; DRUG ANTAGONISM; DRUG DESIGN; HUMAN; MOLECULAR LIBRARY; STEREOISOMERISM; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

BINDING SITES; CELL LINE; DRUG DESIGN; HUMANS; MOLECULAR STRUCTURE; PROTEIN KINASE INHIBITORS; PROTEIN-TYROSINE KINASES; PYRIDINES; PYRIMIDINES; RECOMBINANT PROTEINS; SMALL MOLECULE LIBRARIES; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP; TRIAZOLES;

EID: 77951132083 PISSN: 14770520 EISSN: None Source Type: Journal
DOI: 10.1039/b923882d Document Type: Article

Times cited : (62)

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