SAR studies on new bis-aryls 5-HT7 ligands: Synthesis and molecular modeling

Bioorganic and Medicinal Chemistry

Volumn 18, Issue 5, 2010, Pages 1958-1967

  Badarau, Eduard ^a,b   Bugno, Ryszard ^c   Suzenet, Franck ^a   Bojarski, Andrzej J ^c   Finaru, Adriana Luminita ^b   Guillaumet, Gérald ^a  

^a UNIVERSITÉ D'ORLÉANS   (France)

^b VASILE ALECSANDRI UNIVERSITY OF BACAU   (Romania)

^c INSTITUTE OF PHARMACOLOGY   (Poland)

Author keywords

Bis aryls; Molecular modeling; SAR

Indexed keywords

ALIPHATIC AMINE; BENZENE DERIVATIVE; POLYCYCLIC AROMATIC HYDROCARBON DERIVATIVE; PYRIDINE DERIVATIVE; SEROTONIN RECEPTOR; SULFADIAZINE; TRIAZINE;

ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; MOLECULAR DOCKING; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

EID: 77549084127     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2010.01.035     Document Type: Article

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