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Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 53, Issue 2, 2010, Pages 63-67

Radiosynthesis of N-[4-(4-fluorobenzyl) piperidin-1-yl]-N'-(2-[ 11C]oxo-1,3-dihydrobenzimidazol-5-yl)oxamide, a NR2B-selective NMDA receptor antagonist

(8) Labas, Romain a,b Sobrio, Franck a,b Bramoullé, Yann c Hérard, Anne Sophie c Guillermier, Martine c Hantraye, Philippe c Dollé, Frédéric c Barre, Louisa a,b,d

a DIF (France)

b UNIVERSITÉ DE CAEN (France)

c SERVICE HOSPITALIER FRÉDÉRIC JOLIOT (France)

d Centre Cyceron (France)

Author keywords

Carbon 11; NMDA; NR2B; PET; Radiolabelling

Indexed keywords

CARBON;

CARBON-11; IN-VIVO IMAGING; LABELINGS; NMDA; NMDA RECEPTOR; NR2B; OXAMIDES; RADIOLABELLING; RADIOSYNTHESIS; RECEPTOR ANTAGONISTS;

POSITRON EMISSION TOMOGRAPHY;

2 ACETAMIDO N (2 OXO 2,3 DIHYDROBENZIMIDAZOL 5 YL)ACETIC ACID; 4 (4 FLUOROBENZYL)PIPERIDINE; 4 BENZYL ALPHA (4 HYDROXYPHENYL) BETA METHYL 1 PIPERIDINEPROPANOL H 3; ACETONITRILE; BENZIMIDAZOLONE C 11; ETHYL 2 ACETAMIDO N (2 OXO 2,3 DIHYDROBENZIMIDAZOL 5 YL)ACETATE; ETHYL 2 ACETAMIDO N (4 AMINO 3 NITROPHENYL)ACETATE; METHANE C 11; N (3,4 DIAMINOPHENYL) N [4 (4 FLUOROBENZYL)PIPERIDIN 1 YL] OXAMIDE; N METHYL DEXTRO ASPARTIC ACID RECEPTOR 2B; N METHYL DEXTRO ASPARTIC ACID RECEPTOR BLOCKING AGENT; N [4 (4 FLUOROBENZYL)PIPERIDIN 1 YL] N (2 OXO 1,3 DIHYDROBENZIMIDAZOL 5 YL)OXAMIDE; N [4 (4 FLUOROBENZYL)PIPERIDIN 1 YL] N (4 AMINO 3 NITROPHENYL)OXAMIDE; N [4 (4 FLUOROBENZYL)PIPERIDIN 1 YL] N' (2 OXO 1,3 DIHYDROBENZIMIDAZOL 5 YL)OXAMIDE C 11; OXAMIC ACID; PHENYLENEDIAMINE; PHOSGENE; PHOSGENE C 11; RADIOLIGAND; RADIOPHARMACEUTICAL AGENT; UNCLASSIFIED DRUG;

AFFINITY LABELING; ARTICLE; BINDING ASSAY; DRUG FORMULATION; DRUG HALF LIFE; DRUG PURIFICATION; DRUG RECEPTOR BINDING; DRUG SCREENING; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; IC 50; IN VIVO STUDY; ISOTOPE LABELING; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; RADIOACTIVITY; RADIOCHEMISTRY; RADIOISOTOPE DECAY; THIN LAYER CHROMATOGRAPHY;

EID: 77249125378 PISSN: 03624803 EISSN: 10991344 Source Type: Journal
DOI: 10.1002/jlcr.1702 Document Type: Article

Times cited : (15)

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