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Volumn 49, Issue 1, 2010, Pages 120-124

Optimization of preparation of matrix pellets containing ethylcellulose

Author keywords

Breaking hardness; Dissolution; Ethylcellulose; Extrusion spheronization; Factorial design; Wetting

Indexed keywords

ACTIVE AGENTS; ATENOLOL; BREAKING HARDNESS; ETHYLCELLULOSE; EXTRUSION/SPHERONIZATION; FACTORIAL DESIGN; MATRIX; MATRIX STRUCTURE; MICROCRYSTALLINE CELLULOSE; MORPHOLOGICAL STUDY; OPERATIONAL PARAMETERS; RELATIVE IMPORTANCE; SPHERONIZATION; WATER ETHANOL MIXTURES; WETTING LIQUIDS;

EID: 75249091863     PISSN: 02552701     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.cep.2009.12.002     Document Type: Article
Times cited : (20)

References (42)
  • 2
    • 33745506391 scopus 로고    scopus 로고
    • Review of pulsatile drug delivery
    • Bussemer T., and Bodmeier R. Review of pulsatile drug delivery. Am. Pharm. Rev. 4 (2001) 24
    • (2001) Am. Pharm. Rev. , vol.4 , pp. 24
    • Bussemer, T.1    Bodmeier, R.2
  • 3
    • 0032865227 scopus 로고    scopus 로고
    • Chronopharmacokinetics: implications for drug treatment
    • Lemmer B. Chronopharmacokinetics: implications for drug treatment. J. Pharm. Pharmacol. 51 (1999) 887-890
    • (1999) J. Pharm. Pharmacol. , vol.51 , pp. 887-890
    • Lemmer, B.1
  • 5
    • 0001960774 scopus 로고
    • Biopharmaceutical aspects of multiparticulate
    • Ghebre-Selassie I. (Ed), Marcel Dekker, New York
    • Krämer J., and Blume H. Biopharmaceutical aspects of multiparticulate. In: Ghebre-Selassie I. (Ed). Multiparticulate Oral Drug Delivery (1994), Marcel Dekker, New York 307-332
    • (1994) Multiparticulate Oral Drug Delivery , pp. 307-332
    • Krämer, J.1    Blume, H.2
  • 6
    • 84892537488 scopus 로고
    • Controlled-release multi-units and single unit doses. A literature review
    • Bechgaard H., and Hagermann N.G. Controlled-release multi-units and single unit doses. A literature review. Drug. Dev. Ind. Pharm. 4 (1978) 53-67
    • (1978) Drug. Dev. Ind. Pharm. , vol.4 , pp. 53-67
    • Bechgaard, H.1    Hagermann, N.G.2
  • 7
    • 0022610593 scopus 로고
    • Effect of particle morphology in selecting pharmaceutical excipients
    • Bergeron M., Laurin P., and Tawashi R. Effect of particle morphology in selecting pharmaceutical excipients. Drug Dev. Ind. Pharm. 12 (1986) 915-926
    • (1986) Drug Dev. Ind. Pharm. , vol.12 , pp. 915-926
    • Bergeron, M.1    Laurin, P.2    Tawashi, R.3
  • 8
    • 0019213199 scopus 로고
    • The shape of rock particles, a critical review
    • Barret P.J. The shape of rock particles, a critical review. Sedimentology 27 (1980) 291-303
    • (1980) Sedimentology , vol.27 , pp. 291-303
    • Barret, P.J.1
  • 9
    • 0346352292 scopus 로고    scopus 로고
    • Extrusion and Extruders
    • Swarbrick J., and Boylan J.C. (Eds), Marcel Dekker Inc., New York and Basel
    • Newton J.M. Extrusion and Extruders. In: Swarbrick J., and Boylan J.C. (Eds). Encyclopedia of Pharmaceutical Technology (2002), Marcel Dekker Inc., New York and Basel 1220-1236
    • (2002) Encyclopedia of Pharmaceutical Technology , pp. 1220-1236
    • Newton, J.M.1
  • 10
    • 0028954910 scopus 로고
    • Physicomechanical characterization of the extrusion-spheronization process. 2. Rheological determinants for successful extrusion and spheronization
    • Shah R.D., Kabadi M., Pope D.G., and Augsburger L.L. Physicomechanical characterization of the extrusion-spheronization process. 2. Rheological determinants for successful extrusion and spheronization. Pharm. Res. 12 (1995) 496-507
    • (1995) Pharm. Res. , vol.12 , pp. 496-507
    • Shah, R.D.1    Kabadi, M.2    Pope, D.G.3    Augsburger, L.L.4
  • 11
    • 0035807459 scopus 로고    scopus 로고
    • Effect of drying rate on porosity and tableting behaviour of cellulose pellets
    • Berggren J., and Alderborn G. Effect of drying rate on porosity and tableting behaviour of cellulose pellets. Int. J. Pharm. 227 (2001) 81-96
    • (2001) Int. J. Pharm. , vol.227 , pp. 81-96
    • Berggren, J.1    Alderborn, G.2
  • 12
    • 0003039780 scopus 로고    scopus 로고
    • Effect of different drying techniques on the physico-mechanical properties of beads containing microcrystalline cellulose produced by extrusion and spheronization
    • Habib Y.S., and Shangraw R.F. Effect of different drying techniques on the physico-mechanical properties of beads containing microcrystalline cellulose produced by extrusion and spheronization. Pharm. Res. 14 (1997) S14
    • (1997) Pharm. Res. , vol.14
    • Habib, Y.S.1    Shangraw, R.F.2
  • 13
    • 0028043172 scopus 로고
    • Shrinking and swelling properties of pellets containing MCC and low substituted hydroxy propyl cellulose. Part I. Shrinking properties
    • Kleinebudde P. Shrinking and swelling properties of pellets containing MCC and low substituted hydroxy propyl cellulose. Part I. Shrinking properties. Int. J. Pharm. 109 (1994) 209-219
    • (1994) Int. J. Pharm. , vol.109 , pp. 209-219
    • Kleinebudde, P.1
  • 14
    • 0028043747 scopus 로고
    • Effects of the drying method on mechanical and release properties of pellets prepared by extrusion-spheronization
    • Dyer A.M., Khan K.A., and Aulton M.E. Effects of the drying method on mechanical and release properties of pellets prepared by extrusion-spheronization. Drug Dev. Ind. Pharm. 20 (1994) 3045-3068
    • (1994) Drug Dev. Ind. Pharm. , vol.20 , pp. 3045-3068
    • Dyer, A.M.1    Khan, K.A.2    Aulton, M.E.3
  • 15
    • 0027403225 scopus 로고
    • Study of the influence of spheronisation and drying conditions on the physico-chemical properties of neutral spheroids containing Avicel PH101 and lactose
    • Bataille B., Ligarski K., Jacob M., Thomas C., and Duru C. Study of the influence of spheronisation and drying conditions on the physico-chemical properties of neutral spheroids containing Avicel PH101 and lactose. Drug Dev. Ind. Pharm. 19 (1993) 653-671
    • (1993) Drug Dev. Ind. Pharm. , vol.19 , pp. 653-671
    • Bataille, B.1    Ligarski, K.2    Jacob, M.3    Thomas, C.4    Duru, C.5
  • 16
    • 0028924865 scopus 로고
    • Factorial design in the feasibility of producing Microcel MC 101 pellets by extrusion/spheronisation
    • Sonaglio D., Bataille B., Ortigosa C., and Jacob M. Factorial design in the feasibility of producing Microcel MC 101 pellets by extrusion/spheronisation. Int. J. Pharm. 115 (1995) 53-60
    • (1995) Int. J. Pharm. , vol.115 , pp. 53-60
    • Sonaglio, D.1    Bataille, B.2    Ortigosa, C.3    Jacob, M.4
  • 17
    • 34547687424 scopus 로고    scopus 로고
    • Correlation between the permeability of metoprolol tartrate through plasticized isolated ethylcellulose/hydroxypropylmethylcellulose films and drug release from reservoir pellets
    • Ye Z.-W., Rombout P., Remon J.P., Vervaet C., and van den Mooter G. Correlation between the permeability of metoprolol tartrate through plasticized isolated ethylcellulose/hydroxypropylmethylcellulose films and drug release from reservoir pellets. Eur. J. Pharm. Biopharm. 67 (2007) 485-490
    • (2007) Eur. J. Pharm. Biopharm. , vol.67 , pp. 485-490
    • Ye, Z.-W.1    Rombout, P.2    Remon, J.P.3    Vervaet, C.4    van den Mooter, G.5
  • 18
    • 0001060092 scopus 로고    scopus 로고
    • Cellulose derivatives and natural products utilized in pharmaceutics
    • Swarbrick J., and Boylan J.C. (Eds), Marcel Dekker, New York and Basel
    • Wallace J.W. Cellulose derivatives and natural products utilized in pharmaceutics. In: Swarbrick J., and Boylan J.C. (Eds). Encyclopedia of Pharmaceutical Technology vol. 2 (2002), Marcel Dekker, New York and Basel
    • (2002) Encyclopedia of Pharmaceutical Technology , vol.2
    • Wallace, J.W.1
  • 19
    • 0027466515 scopus 로고
    • Evaluation of drug layering and coating: effect of process mode and binder level
    • Iyer R.M., Augsburger L.L., and Parikh D.M. Evaluation of drug layering and coating: effect of process mode and binder level. Drug Dev. Ind. Pharm. 19 (1993) 981-998
    • (1993) Drug Dev. Ind. Pharm. , vol.19 , pp. 981-998
    • Iyer, R.M.1    Augsburger, L.L.2    Parikh, D.M.3
  • 20
    • 21244440195 scopus 로고    scopus 로고
    • A subchronic toxicity study in rats and genotoxicity tests with an aqueous ethylcellulose dispersion
    • DeMerlis C.C., Schoneker D.R., and Borzelleca J.F. A subchronic toxicity study in rats and genotoxicity tests with an aqueous ethylcellulose dispersion. Food Chem. Toxicol. 43 (2005) 1355-1364
    • (2005) Food Chem. Toxicol. , vol.43 , pp. 1355-1364
    • DeMerlis, C.C.1    Schoneker, D.R.2    Borzelleca, J.F.3
  • 21
    • 59249104734 scopus 로고    scopus 로고
    • Coating of potassium chloride with ethylcellulose aqueous dispersion-effects of processing parameters on film formation and film properties
    • Naelapää K., Veski P., Kristensen H.G., and Bertelsen P. Coating of potassium chloride with ethylcellulose aqueous dispersion-effects of processing parameters on film formation and film properties. Eur. J. Pharm. Sci. 32 (2007) S20
    • (2007) Eur. J. Pharm. Sci. , vol.32
    • Naelapää, K.1    Veski, P.2    Kristensen, H.G.3    Bertelsen, P.4
  • 26
    • 25344453878 scopus 로고
    • The biological and clinical effects of atenolol (Tenormin) a cardioselective-antagonist
    • Goldberg M.E. (Ed), American Pharmaceutical Association Press, Washington DC
    • Fitzgerald J.D. The biological and clinical effects of atenolol (Tenormin) a cardioselective-antagonist. In: Goldberg M.E. (Ed). Pharmacological and Biochemical Properties of Drug Substances vol. II (1979), American Pharmaceutical Association Press, Washington DC
    • (1979) Pharmacological and Biochemical Properties of Drug Substances , vol.II
    • Fitzgerald, J.D.1
  • 27
    • 0008773526 scopus 로고
    • Review of clinical pharmacology of atenolol
    • Thompson F.D. Review of clinical pharmacology of atenolol. Proc. R. Soc. Med. 70 Suppl. 5 (1977) 5-8
    • (1977) Proc. R. Soc. Med. , vol.70 , Issue.SUPPL. 5 , pp. 5-8
    • Thompson, F.D.1
  • 28
    • 0036010423 scopus 로고    scopus 로고
    • Atenolol: pharmacokinetic/dynamic aspects of comparative developmental toxicity
    • Tabacova S.A., and Kimmel C.A. Atenolol: pharmacokinetic/dynamic aspects of comparative developmental toxicity. Reprod. Toxicol. 16 (2002) 1-7
    • (2002) Reprod. Toxicol. , vol.16 , pp. 1-7
    • Tabacova, S.A.1    Kimmel, C.A.2
  • 29
    • 0342313576 scopus 로고    scopus 로고
    • Extrusion-spheronization of pH-sensitive polymeric matrix pellets for possible colonic drug delivery
    • Karin K., Jyrki H., Johanna V., Martti M., Osmo A., and Jouko Y. Extrusion-spheronization of pH-sensitive polymeric matrix pellets for possible colonic drug delivery. Int. J. Pharm. 199 (2000) 187-194
    • (2000) Int. J. Pharm. , vol.199 , pp. 187-194
    • Karin, K.1    Jyrki, H.2    Johanna, V.3    Martti, M.4    Osmo, A.5    Jouko, Y.6
  • 30
    • 0033955439 scopus 로고    scopus 로고
    • Effect of formulation and process variables on porosity parameters and release rates from a multi unit erosion matrix of a poorly soluble drug
    • Ketan A.M., Kislalioglu M.S., Phuapradit W., Malick A.W., and Shah N.H. Effect of formulation and process variables on porosity parameters and release rates from a multi unit erosion matrix of a poorly soluble drug. J. Control. Release 63 (2000) 201-211
    • (2000) J. Control. Release , vol.63 , pp. 201-211
    • Ketan, A.M.1    Kislalioglu, M.S.2    Phuapradit, W.3    Malick, A.W.4    Shah, N.H.5
  • 31
    • 0035184990 scopus 로고    scopus 로고
    • The influence of model drugs on the preparation of pellets by extrusion/spheronization: II spheronization parameters
    • Tomer G., Podczeck F., and Newton J.M. The influence of model drugs on the preparation of pellets by extrusion/spheronization: II spheronization parameters. Int. J. Pharm. 231 (2002) 107-119
    • (2002) Int. J. Pharm. , vol.231 , pp. 107-119
    • Tomer, G.1    Podczeck, F.2    Newton, J.M.3
  • 32
    • 79955412254 scopus 로고
    • Nürnberg E., and Surmann P. (Eds), Springer Verlag, Bd. 2 Methoden, Berlin, New York
    • In: Nürnberg E., and Surmann P. (Eds). Hagers Handbuch der pharmazeutischen Praxis. fifth edition (1991), Springer Verlag, Bd. 2 Methoden, Berlin, New York 60
    • (1991) Hagers Handbuch der pharmazeutischen Praxis. fifth edition , pp. 60
  • 34
    • 0041883581 scopus 로고    scopus 로고
    • Solidification with water as a treatment method for air pollution control residues
    • Todorovic J., Ecke H., and Lagerkvis A. Solidification with water as a treatment method for air pollution control residues. Waste Manage. 23 (2003) 621-629
    • (2003) Waste Manage. , vol.23 , pp. 621-629
    • Todorovic, J.1    Ecke, H.2    Lagerkvis, A.3
  • 35
    • 0037429310 scopus 로고    scopus 로고
    • Ethylene and 1-butene copolymerization catalyzed by a Ziegler-Natta/metallocene hybrid catalyst through a 23 factorial experimental design
    • Forte M.M.C., Cunha F.O.V., Santos J.H.Z., and Zacca J.J. Ethylene and 1-butene copolymerization catalyzed by a Ziegler-Natta/metallocene hybrid catalyst through a 23 factorial experimental design. Polymer 44 (2003) 1377-1384
    • (2003) Polymer , vol.44 , pp. 1377-1384
    • Forte, M.M.C.1    Cunha, F.O.V.2    Santos, J.H.Z.3    Zacca, J.J.4
  • 36
    • 44249095369 scopus 로고    scopus 로고
    • The effect of wetting of a powder mixture on the preparation of hydrophilic matrix granules with a high-shear granulator
    • Bajdik J., Baki G., Kelemen A., and Pintye-Hódi K. The effect of wetting of a powder mixture on the preparation of hydrophilic matrix granules with a high-shear granulator. Chem Eng. Res. Des. 86 (2008) 1-7
    • (2008) Chem Eng. Res. Des. , vol.86 , pp. 1-7
    • Bajdik, J.1    Baki, G.2    Kelemen, A.3    Pintye-Hódi, K.4
  • 37
    • 0037570797 scopus 로고    scopus 로고
    • Development of modified release diltiazem HCl tablets using composite index to identify optimal formulation
    • Gohel M.C., Patel M.M., and Amin A.F. Development of modified release diltiazem HCl tablets using composite index to identify optimal formulation. Drug Dev. Ind. Pharm. 29 (2003) 565-574
    • (2003) Drug Dev. Ind. Pharm. , vol.29 , pp. 565-574
    • Gohel, M.C.1    Patel, M.M.2    Amin, A.F.3
  • 38
    • 0036804726 scopus 로고    scopus 로고
    • Factors affecting incorporation of drug into solid solution with HPMC during solvent change co-precipitation
    • Sertsou G., Butler J., Scott A., Hempenstall J., and Rades T. Factors affecting incorporation of drug into solid solution with HPMC during solvent change co-precipitation. Int. J. Pharm. 245 (2002) 99-108
    • (2002) Int. J. Pharm. , vol.245 , pp. 99-108
    • Sertsou, G.1    Butler, J.2    Scott, A.3    Hempenstall, J.4    Rades, T.5
  • 40
    • 23744494201 scopus 로고    scopus 로고
    • Process analytical technology: the route to process understanding and control
    • Davies B., and Ellis S. Process analytical technology: the route to process understanding and control. Pharma. Technol. Eur. 17 (2005) 17-23
    • (2005) Pharma. Technol. Eur. , vol.17 , pp. 17-23
    • Davies, B.1    Ellis, S.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.