Using compression calorimetry to characterize powder compaction behavior of pharmaceutical materials

Journal of Pharmaceutical Sciences

Volumn 99, Issue 2, 2010, Pages 861-870

  Buckner, Ira S ^a   Friedman, Ross A ^a   Wurster, Dale Eric ^a  

^a UNIVERSITY OF IOWA   (United States)

Author keywords

Calorimetry; Compaction; Compression; Deformation mechanism; Mechanical properties; Tableting; Thermodynamics

Indexed keywords

CALCIUM PHOSPHATE DIBASIC; LACTOSE; MAGNESIUM STEARATE; MICROCRYSTALLINE CELLULOSE; PARACETAMOL;

ARTICLE; CALORIMETRY; DECOMPRESSION; POWDER; THERMODYNAMICS;

EID: 74049098567     PISSN: 00223549     EISSN: 15206017     Source Type: Journal    
DOI: 10.1002/jps.21881     Document Type: Article

References (35)

1. De Boer AH, Bolhuis GK, Lerk CF. 1978. Bonding characteristics by scanning electron microscopy of powders mixed with magnesium stearate. Powder Technol 20:75-82.
2. Roberts RJ, Rowe RC. 1985. The effect of punch velocity on the compaction of a variety of materials. J Pharm Pharmacol 37:377-384.
3. Hiestand EN. 1997. Mechanical properties of compacts and particles that control tableting success. J Pharm Sci 86:985-990.
4. Lieberman HA, Lachman L, editors. 1980. Pharmaceutical dosage forms. Tablets. 1st edition. New York, NY: Marcel Dekker.
5. Leuenberger H, Leu R. 1992. Formation of a tablet: A site and bond percolation phenomenon. J Pharm Sci 81:976-982.
6. Mullarney MP, Hancock BC. 2004. Improving the prediction of exceptionally poor tableting performance: An investigation into Hiestand's "special case." J Pharm Sci 93:2017-2021.
7. Aburub A, Buckner IS. 2007. Utilization of compaction energetics for understanding particle deformation mechanism. Pharm Dev Technol 12:405-414.
8. Ragnarsson G, Sjogren J. 1985. Force-displacement measurements in tableting. J Pharm Pharmacol 37:145-150.
9. Zhao J, Burt HM, Miller RA. 2006. The Gurnham Equation in characterizing the compressibility of pharmaceutical materials. Int J Pharm 317:109-113.
10. Coffin-Beach DP, Hollenbeck RG. 1983. Determination of the energy of tablet formation during compression of selected pharmaceutical powders. Int J Pharm 17:313-324.
11. DeCrosta MT, Schwartz JB, Wigent RJ, Marshall K. 2000. Thermodynamic analysis of compact formation; compaction, unloading, and ejection I. Design and development of a compaction calorimeter and mechanical and thermal energy determinations of powder compaction. Int J Pharm 198:113-134.
12. Wurster DE, Rowlings CE, Creekmore JR. 1995. Calorimetric analysis of powder compression: I. Design and development of a compression calorimeter. Int J Pharm 116:179-189.
13. Zavaliangos A, Galen S, Cunningham J, Winstead D. 2008. Temperature evolution during compaction of pharmaceutical powders. J Pharm Sci 97:3291-3304.
14. Creekmore JR. 1986. Measurement of the thermal energy change upon tablet compression. Ph.D. Thesis, University of Iowa, Iowa City, IA.
15. Rowlings CE. 1989. Compression calorimetry. Ph.D. Thesis, University of Iowa, Iowa City, IA.
16. Ternik RL. 1996. Design and development of a compression calorimeter and the determination of compression-decompression induced energy changes. Ph.D. Thesis, University of Iowa, Iowa City, IA.
17. Kothapalli VM. 2001. Elucidation of the dependence of the thermodynamic energy terms for compaction of carbohydrate polymers upon water vapor sorption and molecular weight. Ph.D. Thesis, University of Iowa, Iowa City, IA.
18. Gharaibeh SF. 2005. The use of the compression calorimeter for the estimation of thermodynamic parameters associated with the compaction of binary powder mixtures. Ph.D. Thesis, University of Iowa, Iowa City, IA.
19. Buckner IS. 2008. Compression calorimetry, powder compaction thermodynamics and deformation mechanisms. Ph.D. Thesis, University of Iowa, Iowa City, IA.
20. Alderborn G, Nystrom C, editors. 1996. Pharmaceutical powder compaction technology. 1st edition. New York: Marcel Dekker, Inc.
21. Ruegger CE, Celik M. 2000. The effect of compression and decompression speed on the mechanical strength of compacts. Pharm Dev Technol 5:485-494.
22. Schmidt PC, Herzog R. 1993. Calcium phosphates in pharmaceutical tableting. 2. Comparison of tableting properties. Pharm World Sci 15:116-122.
23. Zhang Y, Law Y, Chakrabarti S. 2003. Physical properties and compact analysis of commonly used direct compression binders. AAPS PharmSciTech 4:62.
24. Lin M-C, Duncan-Hewitt WC. 1994. Deformation kinetics of acetaminophen crystals. Int J Pharm 106:187-200.
25. Higuchi T, Nelson E, Busse LW. 1954. The physics of tablet compression 3. Design and construction of an instrumented tableting machine. J Am Pharm Assoc Sci 43:344-348.
26. Nelson E, Naqvi SM, Busse LW, Higuchi T. 1954. The physics of tablet compression 4. Relationship of ejection, and upper and lower punch forces during compressional process: Application of measurements to comparison of tablet lubricants. J Am Pharm Assoc Sci 43:596-602.
27. Carslaw HS, Jaeger JC. 1959. Conduction of heat in solids. 2nd edition. London: Oxford University Press. p. 9, 336
28. Crank J. 1975. The mathematics of diffusion. 2nd edition. London: Oxford University Press. p. 32.
29. Duberg M, Nystrom C. 1986. Studies on direct compression of tablets XVII. Porosity-pressure curves for the characterization of volume reduction mechanisms in powder compression. Powder Technol 46:67-75.
30. Heinicke G. 1984. Tribochemistry. 1st edition. Berlin: Akademie-Verlag. p. 55.
31. Godovsky YK. 1992. Thermophysical properties of polymers. 1st edition. New York: Springer-Verlag.
32. Salamatina OB, Hohne GWH, Rudnev SN, Oleinik EF. 1994. Work, heat and stored energy in compressive plastic deformation of glassy polymers. Thermochim Acta 247:1-18.
33. Hiestand EN. 1997. Principles, tenets and notions of tablet bonding and measurements of strength. Eur J Pharm Biopharm 44:229-242.
34. Ilkka J, Paronen P. 1993. Prediction of the compression behavior of powder mixtures by the Heckel Equation. Int J Pharm 94:181-187.
35. Bolhuis GK, Hölzer AW. 1996. Lubricant sensitivity. In: Alderborn G, Nystrom C, editors. Pharmaceutical powder compaction technology. 1st edition. New York: Marcel Dekker, Inc. p. 521.