-
1
-
-
38849161554
-
Chiral tertiary diamines in asymmetric synthesis
-
Kizirian, J.-C. Chiral tertiary diamines in asymmetric synthesis. Chem. Rev. 2008, 108, 140-205.
-
(2008)
Chem. Rev.
, vol.108
, pp. 140-205
-
-
Kizirian, J.-C.1
-
2
-
-
20744455249
-
4 receptor agonists
-
4 receptor agonists. Bioorg. Med. Chem. 2005, 13, 4667-4678;
-
(2005)
Bioorg. Med. Chem.
, vol.13
, pp. 4667-4678
-
-
Wang, X.1
Bhatia, P.A.2
Daanen, J.F.3
Latsaw, S.P.4
Rohde, J.5
Kolasa, T.6
Hakeem, A.A.7
Matulenko, M.A.8
Nakane, M.9
Uchic, M.E.10
Miller, L.N.11
Chang, R.12
Moreland, R.B.13
Brioni, J.D.14
Stewart, A.O.15
-
3
-
-
43849094200
-
First stereoselective synthesis and assignment of the absolute configuration of the nebracetam eutomer and derivatives
-
(b) Lima, E. C.; Domingos, J. L. O.; Dias, A. G.; Costa, P. R. R. First stereoselective synthesis and assignment of the absolute configuration of the nebracetam eutomer and derivatives. Tetrahedron: Asymmetry 2008, 19, 1161-1165;
-
(2008)
Tetrahedron: Asymmetry
, vol.19
, pp. 1161-1165
-
-
Lima, E.C.1
Domingos, J.L.O.2
Dias, A.G.3
Costa, P.R.R.4
-
4
-
-
53649098571
-
The formal synthesis of isofebrifugine using stereoselective intramolecular Michael addition
-
(c) Sudhakar, N.; Srinivasulu, G.; Rao, G. S.; Rao, B. V. The formal synthesis of isofebrifugine using stereoselective intramolecular Michael addition. Tetrahedron: Asymmetry 2008, 19, 2153-2158;
-
(2008)
Tetrahedron: Asymmetry
, vol.19
, pp. 2153-2158
-
-
Sudhakar, N.1
Srinivasulu, G.2
Rao, G.S.3
Rao, B.V.4
-
5
-
-
44649117342
-
Asymmetric synthesis of the optically active piperidine alkaloid (\+)-b-conhydrine
-
(d) Lebrun, S.; Couture, A.; Deniau, E.; Grandclaudon, P. Asymmetric synthesis of the optically active piperidine alkaloid (\+)-b-conhydrine. Tetrahedron: Asymmetry 2008, 19, 1245-1249;
-
(2008)
Tetrahedron: Asymmetry
, vol.19
, pp. 1245-1249
-
-
Lebrun, S.1
Couture, A.2
Deniau, E.3
Grandclaudon, P.4
-
6
-
-
35848940252
-
Stereoselective synthesis of a novel 2-aza-7-oxabicy-clo[3.3.0]octane as neurokinin-1 receptor antagonist
-
(e) Shishido, Y.; Ito, F.; Morita, H.; Ikunaka, M. Stereoselective synthesis of a novel 2-aza-7-oxabicy-clo[3.3.0]octane as neurokinin-1 receptor antagonist. Bioorg. Med. Chem. Lett. 2007, 17, 6887-6890.
-
(2007)
Bioorg. Med. Chem. Lett.
, vol.17
, pp. 6887-6890
-
-
Shishido, Y.1
Ito, F.2
Morita, H.3
Ikunaka, M.4
-
7
-
-
1942456786
-
Biological relevance and synthesis of C-substituted morpholine derivatives
-
Bioactive compounds, containing morpholine moiety: (a) Wijtmans, R.; Vink, M. K. S.; Schoemaker, H. E.; van Delft, F. L.; Blaauw, R. H.; Rutjes, F. P. J. T. Biological relevance and synthesis of C-substituted morpholine derivatives. Synthesis 2004, 641-662;
-
(2004)
Synthesis
, pp. 641-662
-
-
Wijtmans, R.1
Vink, M.K.S.2
Schoemaker, H.E.3
Van Delft, F.L.4
Blaauw, R.H.5
Rutjes, F.P.J.T.6
-
8
-
-
41849121199
-
Design and synthesis of morpholine derivatives: SAR for dual serotonin and noradrenaline reuptake inhibition
-
(b) Fish, P. V.; Deur, C.; Gan, X.; Greene, K.; Hoople, D.; Mackenny, M.; Para, K. S.; Reeves, K.; Ryckmans, T.; Stiff, C.; Stobie, A.; Wakenhut, F.; Whitlock, G. A. Design and synthesis of morpholine derivatives: SAR for dual serotonin and noradrenaline reuptake inhibition. Bioorg. Med. Chem. Lett. 2008, 18, 2562-2566;
-
(2008)
Bioorg. Med. Chem. Lett.
, vol.18
, pp. 2562-2566
-
-
Fish, P.V.1
Deur, C.2
Gan, X.3
Greene, K.4
Hoople, D.5
MacKenny, M.6
Para, K.S.7
Reeves, K.8
Ryckmans, T.9
Stiff, C.10
Stobie, A.11
Wakenhut, F.12
Whitlock, G.A.13
-
9
-
-
2342658950
-
Synthesis of morpholine nucleo-side triphosphates
-
(c) Abramova, T. V.; Bakharev, P. A.; Vasilyeva, S. V.; Silnikov, V. N. Synthesis of morpholine nucleo-side triphosphates. Tetrahedron Lett. 2004, 45, 4361-4364;
-
(2004)
Tetrahedron Lett.
, vol.45
, pp. 4361-4364
-
-
Abramova, T.V.1
Bakharev, P.A.2
Vasilyeva, S.V.3
Silnikov, V.N.4
-
10
-
-
22044439589
-
Enantioselective synthesis of (2R,3R)-and (2S,3S)-2-[(3-chlorophenyl)-(2- methoxyphe-noxy)methyl]morpholine
-
(d) Harding, W. W.; Hodge, M.; Wang, Z.; Woolverton, W. L.; Parrish, D.; Deschamps, J. R.; Prisinzano, T. E. Enantioselective synthesis of (2R,3R)-and (2S,3S)-2-[(3-chlorophenyl)-(2-methoxyphe-noxy)methyl]morpholine. Tetrahedron: Asymmetry 2005, 16, 2249-2256;
-
(2005)
Tetrahedron: Asymmetry
, vol.16
, pp. 2249-2256
-
-
Harding, W.W.1
Hodge, M.2
Wang, Z.3
Woolverton, W.L.4
Parrish, D.5
Deschamps, J.R.6
Prisinzano, T.E.7
-
11
-
-
52649144883
-
Stereoselective cyclopropanation of serine-and threonine-derived oxazines to access new morpholine-based scaffolds
-
(e) Sladojevich, F.; Trabocchi, A.; Guarna, A. Stereoselective cyclopropanation of serine-and threonine-derived oxazines to access new morpholine-based scaffolds. Org. Biomol. Chem. 2008, 6, 3328-3336.
-
(2008)
Org. Biomol. Chem.
, vol.6
, pp. 3328-3336
-
-
Sladojevich, F.1
Trabocchi, A.2
Guarna, A.3
-
12
-
-
52149113820
-
The advent and development of organocatalysis
-
MacMillan, D. W. C. The advent and development of organocatalysis. Nature 2008, 455, 304-308.
-
(2008)
Nature
, vol.455
, pp. 304-308
-
-
MacMillan, D.W.C.1
-
13
-
-
38349100690
-
Asymmetric enamine catalysis
-
Some recent reviews: (a) Mukherjee, S.; Yang, J. W.; Hoffmann, S.; List, B. Asymmetric enamine catalysis. Chem. Rev. 2007, 107, 5471-5569;
-
(2007)
Chem. Rev.
, vol.107
, pp. 5471-5569
-
-
Mukherjee, S.1
Yang, J.W.2
Hoffmann, S.3
List, B.4
-
14
-
-
38349178582
-
Iminium catalysis
-
(b) Erkkila, A.; Majander, I.; Pihko, P. M. Iminium catalysis. Chem. Rev. 2007, 107, 5416-5470;
-
(2007)
Chem. Rev.
, vol.107
, pp. 5416-5470
-
-
Erkkila, A.1
Majander, I.2
Pihko, P.M.3
-
15
-
-
34547463692
-
Chiral amines as organocatalysts for asymmetric conjugate addition to nitroolefins and vinyl sulfones via enamine activation
-
(c) Sulzer-Mosse, S.; Alexakis, A. Chiral amines as organocatalysts for asymmetric conjugate addition to nitroolefins and vinyl sulfones via enamine activation. Chem. Commun. 2007, 3123-3135.
-
(2007)
Chem. Commun.
, pp. 3123-3135
-
-
Sulzer-Mosse, S.1
Alexakis, A.2
-
16
-
-
33745169362
-
Anchimeric assistance in the case of vicinal dimesylate: Formation of enantiomeric or meso-bimorpholine
-
(a) Kanger, T.; Laars, M.; Kriis, K.; Kailas, T.; Müürisepp, A.-M.; Pehk, T.; Lopp, M. Anchimeric assistance in the case of vicinal dimesylate: Formation of enantiomeric or meso-bimorpholine. Synthesis 2006, 11, 1853-1857;
-
(2006)
Synthesis
, vol.11
, pp. 1853-1857
-
-
Kanger, T.1
Laars, M.2
Kriis, K.3
Kailas, T.4
Müürisepp, A.-M.5
Pehk, T.6
Lopp, M.7
-
18
-
-
41449101549
-
2-symmetric heterocyclic organocatalysts in asymmetric aldol reactions
-
2-symmetric heterocyclic organocatalysts in asymmetric aldol reactions. Tetrahedron: Asymmetry 2008, 19, 641-645;
-
(2008)
Tetrahedron: Asymmetry
, vol.19
, pp. 641-645
-
-
Laars, M.1
Kriis, K.2
Kailas, T.3
Müürisepp, A.-M.4
Pehk, T.5
Kanger, T.6
Lopp, M.7
-
19
-
-
34447311656
-
Bimorpholine-mediated enantiose-lective intramolecular and intermolecular aldol condensation
-
(b) Kanger, T.; Kriis, K.; Laars, M.; Kailas, T.; Muurisepp, A.-M.; Pehk, T.; Lopp, M. Bimorpholine-mediated enantiose-lective intramolecular and intermolecular aldol condensation. J. Org. Chem. 2007, 72, 5168-5173;
-
(2007)
J. Org. Chem.
, vol.72
, pp. 5168-5173
-
-
Kanger, T.1
Kriis, K.2
Laars, M.3
Kailas, T.4
Muurisepp, A.-M.5
Pehk, T.6
Lopp, M.7
-
20
-
-
34250710661
-
Bimorpholines as alternative organocatalysts in asymmetric aldol reactions
-
(c) Kriis, K.; Laars, M.; Lippur, K.; Kanger, T. Bimorpholines as alternative organocatalysts in asymmetric aldol reactions. Chimia 2007, 61, 232-235;
-
(2007)
Chimia
, vol.61
, pp. 232-235
-
-
Kriis, K.1
Laars, M.2
Lippur, K.3
Kanger, T.4
-
21
-
-
33746321842
-
Enantioselective synthesis of Wieland-Miescher ketone through bimorpholine-catalyzed organocatalytic aldol condensation
-
(d) Kriis, K.; Kanger, T.; Laars, M.; Kailas, T.; Muurisepp, A.-M.; Pehk, T.; Lopp, M. Enantioselective synthesis of Wieland-Miescher ketone through bimorpholine-catalyzed organocatalytic aldol condensation. Synlett 2006, 1699-1702;
-
(2006)
Synlett
, pp. 1699-1702
-
-
Kriis, K.1
Kanger, T.2
Laars, M.3
Kailas, T.4
Muurisepp, A.-M.5
Pehk, T.6
Lopp, M.7
-
22
-
-
33745542958
-
0-bimorpholine derivatives as a new class of organocatalysts for asymmetric michael addition
-
0-bimorpholine derivatives as a new class of organocatalysts for asymmetric michael addition. Org. Lett. 2006, 8, 2559-2562.
-
(2006)
Org. Lett.
, Issue.8
, pp. 2559-2562
-
-
Mosse, S.1
Laars, M.2
Kriis, K.3
Kanger, T.4
Alexakis, A.5
-
23
-
-
33846849105
-
0-quaternary salts as chiral phase transfer catalysts
-
0-quaternary salts as chiral phase transfer catalysts. Tetrahedron: Asymmetry 2007, 18, 137-141.
-
(2007)
Tetrahedron: Asymmetry
, vol.18
, pp. 137-141
-
-
Lippur, K.1
Kanger, T.2
Kriis, K.3
Kailas, T.4
Müürisepp, A.-M.5
Pehk, T.6
Lopp, M.7
-
25
-
-
33845283356
-
Cyanide as an efficient and mild catalyst in the aminolysis of esters
-
(b) Hogberg, T.; Strom, P.; Ebner, M.; Ramsby, S. Cyanide as an efficient and mild catalyst in the aminolysis of esters. J. Org. Chem. 1987, 52, 2033-2036.
-
(1987)
J. Org. Chem.
, vol.52
, pp. 2033-2036
-
-
Hogberg, T.1
Strom, P.2
Ebner, M.3
Ramsby, S.4
-
26
-
-
1642486447
-
Efficient, stereoselective synthesis of trans-2,5-disubstituted morpholines
-
Lanman, B. A.; Myers, A. G. Efficient, stereoselective synthesis of trans-2,5-disubstituted morpholines. Org. Lett. 2004, 6, 1045-1047.
-
(2004)
Org. Lett.
, vol.6
, pp. 1045-1047
-
-
Lanman, B.A.1
Myers, A.G.2
-
27
-
-
0041508387
-
Metal oxide in aqueous organic solution promoted chemoselective N-sulfonylation of hydrophilic amino alcohols
-
Kang, H. H., Rho, H. S., Kim, D. H., Oh, S.-G. Metal oxide in aqueous organic solution promoted chemoselective N-sulfonylation of hydrophilic amino alcohols. Tetrahedron Lett. 2003, 44, 7225-7227.
-
(2003)
Tetrahedron Lett.
, vol.44
, pp. 7225-7227
-
-
Kang, H.H.1
Rho, H.S.2
Kim, D.H.3
Oh, S.-G.4
-
28
-
-
33846615885
-
Highly efficient synthesis of enantiomerically enriched 2-hydroxymethylaziridines by enzymatic desymmetrization
-
Choi, J. Y.; Borch, R. F. Highly efficient synthesis of enantiomerically enriched 2-hydroxymethylaziridines by enzymatic desymmetrization. Org. Lett. 2007, 9, 215-218.
-
(2007)
Org. Lett.
, vol.9
, pp. 215-218
-
-
Choi, J.Y.1
Borch, R.F.2
|