메뉴 건너뛰기




Volumn 13, Issue 6, 2009, Pages 1307-1314

A practical solid form screen approach to identify a pharmaceutical glutaric acid cocrystal for development

Author keywords

[No Author keywords available]

Indexed keywords


EID: 72449150123     PISSN: 10836160     EISSN: 1520586X     Source Type: Journal    
DOI: 10.1021/op900137j     Document Type: Article
Times cited : (39)

References (36)
  • 2
    • 34250870110 scopus 로고    scopus 로고
    • An overview of pharmaceutical cocrystals as intellectual property
    • Trask Andrew, V. An overview of pharmaceutical cocrystals as intellectual property. Mol. Pharm. 2007, 4 (3), 301-309
    • (2007) Mol. Pharm. , vol.4 , Issue.3 , pp. 301-309
    • Trask Andrew, V.1
  • 4
    • 5044235632 scopus 로고    scopus 로고
    • Crystal engineering of the composition of pharmaceutical phases. Do pharmaceutical co-crystals represent a new path to improved medicines?
    • Almarsson, O.; Zaworotko, M. J. Crystal engineering of the composition of pharmaceutical phases. Do pharmaceutical co-crystals represent a new path to improved medicines? Chem. Commun. (Cambridge) 2004, 17, 1889-1896.
    • (2004) Chem. Commun. (Cambridge) , vol.17 , pp. 1889-1896
    • Almarsson, O.1    Zaworotko, M.J.2
  • 5
    • 19944371772 scopus 로고    scopus 로고
    • Pharmaceutical cocrystallization: Engineering a remedy for caffeine hydration
    • Trask, A. V.; Motherwell, W. D. S.; Jones, W. Pharmaceutical Cocrystallization: Engineering a Remedy for Caffeine Hydration. Cryst. Growth Des. 2005, 5 (3), 1013-1021.
    • (2005) Cryst. Growth Des. , vol.5 , Issue.3 , pp. 1013-1021
    • Trask, A.V.1    Motherwell, W.D.S.2    Jones, W.3
  • 6
    • 33746425242 scopus 로고    scopus 로고
    • Physical stability enhancement of theophylline via cocrystallization
    • Trask, A. V.; Motherwell, W. D. S.; Jones, W. Physical stability enhancement of theophylline via cocrystallization. Int. J. Pharm. 2006, 320 (1-2), 114-123.
    • (2006) Int. J. Pharm. , vol.320 , Issue.1-2 , pp. 114-123
    • Trask, A.V.1    Motherwell, W.D.S.2    Jones, W.3
  • 9
    • 66249101601 scopus 로고    scopus 로고
    • Solubility advantage of pharmaceutical cocrystals
    • Good, D. J.; Rodriguez-Hornedo, N. Solubility Advantage of Pharmaceutical Cocrystals. Cryst. Growth Des. 2009, 9 (5), 2252-2264.
    • (2009) Cryst. Growth Des. , vol.9 , Issue.5 , pp. 2252-2264
    • Good, D.J.1    Rodriguez-Hornedo, N.2
  • 11
    • 44349162927 scopus 로고    scopus 로고
    • A rapid thermal method for cocrystal screening
    • Lu, E.; Rodriguez-Hornedo, N.; Suryanarayanan, R. A rapid thermal method for cocrystal screening. CrystEngComm 2008, 10 (6), 665-668.
    • (2008) CrystEngComm , vol.10 , Issue.6 , pp. 665-668
    • Lu, E.1    Rodriguez-Hornedo, N.2    Suryanarayanan, R.3
  • 12
    • 33645178186 scopus 로고    scopus 로고
    • Crystal engineering of organic cocrystals by the solid-state grinding approach
    • Organic Solid State Reactions
    • Trask, A. V.; Jones, W. Crystal engineering of organic cocrystals by the solid-state grinding approach. (Organic Solid State Reactions) Top. Curr. Chem. 2005, 254, 41-70.
    • (2005) Top. Curr. Chem. , vol.254 , pp. 41-70
    • Trask, A.V.1    Jones, W.2
  • 13
    • 0036408746 scopus 로고    scopus 로고
    • Mechanochemistry and co-crystal formation: Effect of solvent on reaction kinetics
    • Shan, N.; Toda, F.; Jones, W. Mechanochemistry and co-crystal formation: effect of solvent on reaction kinetics. Chem. Commun. (Cambridge) 2002, 20, 2372-2373.
    • (2002) Chem. Commun. (Cambridge) , vol.20 , pp. 2372-2373
    • Shan, N.1    Toda, F.2    Jones, W.3
  • 14
    • 61749100493 scopus 로고    scopus 로고
    • Synthesis and structural characterization of cocrystals and pharmaceutical cocrystals: Mechanochemistry vs. slow evaporation from solution
    • Weyna, D. R.; Shattock, T.; Vishweshwar, P.; Zaworotko, M. J. Synthesis and Structural Characterization of Cocrystals and Pharmaceutical Cocrystals: Mechanochemistry vs. Slow Evaporation from Solution. Cryst. Growth Des. 2009, 9 (2), 1106-1123.
    • (2009) Cryst. Growth Des. , vol.9 , Issue.2 , pp. 1106-1123
    • Weyna, D.R.1    Shattock, T.2    Vishweshwar, P.3    Zaworotko, M.J.4
  • 15
    • 40549089922 scopus 로고    scopus 로고
    • Indomethacin-saccharin cocrystal: Design, synthesis and preliminary pharmaceutical characterization
    • Basavoju, S.; Bostrom, D.; Velaga Sitaram, P. Indomethacin-saccharin cocrystal: design, synthesis and preliminary pharmaceutical characterization. Pharm. Res. 2008, 25 (3), 530-541
    • (2008) Pharm. Res. , vol.25 , Issue.3 , pp. 530-541
    • Basavoju, S.1    Bostrom, D.2    Velaga Sitaram, P.3
  • 16
    • 53849093843 scopus 로고    scopus 로고
    • Cocrystal screening of stanolone and mestanolone using slurry crystallization
    • Takata, N.; Shiraki, K.; Takano, R.; Hayashi, Y.; Terada, K. Cocrystal Screening of Stanolone and Mestanolone Using Slurry Crystallization. Cryst. Growth Des. 2008, 8 (8), 3032-3037.
    • (2008) Cryst. Growth Des. , vol.8 , Issue.8 , pp. 3032-3037
    • Takata, N.1    Shiraki, K.2    Takano, R.3    Hayashi, Y.4    Terada, K.5
  • 17
    • 34249106473 scopus 로고    scopus 로고
    • Efficient co-crystal screening using solution-mediated phase transformation
    • Zhang, G. G. Z.; Henry, R. F.; Borchardt, T. B.; Lou, X. Efficient co-crystal screening using solution-mediated phase transformation. J. Pharm. Sci. 2007, 96 (5), 990-995.
    • (2007) J. Pharm. Sci. , vol.96 , Issue.5 , pp. 990-995
    • Zhang, G.G.Z.1    Henry, R.F.2    Borchardt, T.B.3    Lou, X.4
  • 18
    • 65249139350 scopus 로고    scopus 로고
    • Cocrystallization: A solution chemistry perspective and the case of benzophenone and diphenylamine
    • Chadwick, K.; Davey, R. J.; Dent, G.; Pritchard, R. G.; Hunter, C. A.; Musumeci, D. Cocrystallization: A Solution Chemistry Perspective and the Case of Benzophenone and Diphenylamine. Cryst. Growth Des. 2009, 9 (4), 1990-1999.
    • (2009) Cryst. Growth Des. , vol.9 , Issue.4 , pp. 1990-1999
    • Chadwick, K.1    Davey, R.J.2    Dent, G.3    Pritchard, R.G.4    Hunter, C.A.5    Musumeci, D.6
  • 19
    • 61749087193 scopus 로고    scopus 로고
    • Role of cocrystal and solution chemistry on the formation and stability of cocrystals with different stoichiometry
    • Jayasankar, A.; Reddy, L. S.; Bethune, S. J.; Rodriguez-Hornedo, N. Role of Cocrystal and Solution Chemistry on the Formation and Stability of Cocrystals with Different Stoichiometry. Cryst. Growth Des. 2009, 9 (2), 889-897.
    • (2009) Cryst. Growth Des. , vol.9 , Issue.2 , pp. 889-897
    • Jayasankar, A.1    Reddy, L.S.2    Bethune, S.J.3    Rodriguez-Hornedo, N.4
  • 21
    • 34250814473 scopus 로고    scopus 로고
    • Celecoxib:nicotinamide dissociation: Using excipients to capture the cocrystal's potential
    • Remenar, J. F.; Peterson, M. L.; Stephens, P. W.; Zhang, Z.; Zimenkov, Y.; Hickey, M. B. Celecoxib:nicotinamide dissociation: using excipients to capture the cocrystal's potential. Mol. Pharm. 2007, 4 (3), 386-400.
    • (2007) Mol. Pharm. , vol.4 , Issue.3 , pp. 386-400
    • Remenar, J.F.1    Peterson, M.L.2    Stephens, P.W.3    Zhang, Z.4    Zimenkov, Y.5    Hickey, M.B.6
  • 22
    • 0028954527 scopus 로고
    • Design and synthesis of hydrogenbonded aggregates. Theory and computation applied to three systems based on the cyanuric acid-melamine lattice
    • Simanek, E. E.; Mammen, M.; Gordon, D. M.; Chin, D.; Mathias, J. P.; Seto, C. T.; Whitesides, G. M. Design and synthesis of hydrogenbonded aggregates. Theory and computation applied to three systems based on the cyanuric acid-melamine lattice. Tetrahedron 1995, 51 (2), 607-619
    • (1995) Tetrahedron , vol.51 , Issue.2 , pp. 607-619
    • Simanek, E.E.1    Mammen, M.2    Gordon, D.M.3    Chin, D.4    Mathias, J.P.5    Seto, C.T.6    Whitesides, G.M.7
  • 23
    • 0000584813 scopus 로고
    • Self-assembly based on the cyanuric acid-melamine lattice
    • Seto, C. T.; Whitesides, G. M. Self-assembly based on the cyanuric acid-melamine lattice. J. Am. Chem. Soc. 1990, 112 (17), 6409-6411
    • (1990) J. Am. Chem. Soc. , vol.112 , Issue.17 , pp. 6409-6411
    • Seto, C.T.1    Whitesides, G.M.2
  • 24
    • 0000607654 scopus 로고    scopus 로고
    • Building organic assemblies with 2-pyridone and dicarboxylic acids: Relating molecular conformation and synthon stability to crystal structure
    • Aakeroy, C. B.; Beatty, A. M.; Zou, M. Building organic assemblies with 2-pyridone and dicarboxylic acids: relating molecular conformation and synthon stability to crystal structure. Cryst. Eng. 1999, 1 (3/ 4), 225-241.
    • (1999) Cryst. Eng. , vol.1 , Issue.3-4 , pp. 225-241
    • Aakeroy, C.B.1    Beatty, A.M.2    Zou, M.3
  • 25
    • 34250891895 scopus 로고    scopus 로고
    • Hierarchy of supramolecular synthons: Persistent hydroxyl⋯pyridine hydrogen bonds in cocrystals that contain a cyano acceptor
    • Bis, J. A.; Vishweshwar, P.; Weyna, D.; Zaworotko, M. J. Hierarchy of Supramolecular Synthons: Persistent Hydroxyl⋯Pyridine Hydrogen Bonds in Cocrystals That Contain a Cyano Acceptor. Mol. Pharm. 2007, 4 (3), 401-416.
    • (2007) Mol. Pharm. , vol.4 , Issue.3 , pp. 401-416
    • Bis, J.A.1    Vishweshwar, P.2    Weyna, D.3    Zaworotko, M.J.4
  • 27
    • 0001752768 scopus 로고    scopus 로고
    • The cambridge structural database: A quarter of a million crystal structures and rising
    • Allen, F. H. The Cambridge Structural Database: a quarter of a million crystal structures and rising. Acta Crystallogr., Sect. B 2002, B58 (3, No. 1), 380-388.
    • (2002) Acta Crystallogr., Sect. B , vol.B58 , Issue.1-3 , pp. 380-388
    • Allen, F.H.1
  • 28
    • 65249148409 scopus 로고    scopus 로고
    • Cambridge structural database analysis of molecular complementarity in cocrystals
    • Fabian, L. Cambridge Structural Database Analysis of Molecular Complementarity in Cocrystals. Cryst. Growth Des. 2009, 9 (3), 1436-1443.
    • (2009) Cryst. Growth Des. , vol.9 , Issue.3 , pp. 1436-1443
    • Fabian, L.1
  • 30
    • 60849106279 scopus 로고    scopus 로고
    • The role of solvent in mechanochemical and sonochemical cocrystal formation: A solubility-based approach for predicting cocrystallisation outcome
    • Friscic, T.; Childs, S. L.; Rizvi, S. A. A.; Jones, W. The role of solvent in mechanochemical and sonochemical cocrystal formation: a solubility-based approach for predicting cocrystallisation outcome. CrystEngComm 2009, 11 (3), 418-426.
    • (2009) CrystEngComm , vol.11 , Issue.3 , pp. 418-426
    • Friscic, T.1    Childs, S.L.2    Rizvi, S.A.A.3    Jones, W.4
  • 32
    • 60849091081 scopus 로고    scopus 로고
    • Control and interconversion of cocrystal stoichiometry in grinding: Stepwise mechanism for the formation of a hydrogen-bonded cocrystal
    • Karki, S.; Friscic, T.; Jones, W. Control and interconversion of cocrystal stoichiometry in grinding: stepwise mechanism for the formation of a hydrogen-bonded cocrystal. CrystEngComm 2009, 11 (3), 470-481.
    • (2009) CrystEngComm , vol.11 , Issue.3 , pp. 470-481
    • Karki, S.1    Friscic, T.2    Jones, W.3
  • 33
    • 32644436069 scopus 로고    scopus 로고
    • Phase solubility diagrams of cocrystals are explained by solubility product and solution complexation
    • Nehm, S. J.; Rodriguez-Spong, B.; Rodriguez-Hornedo, N. Phase Solubility Diagrams of Cocrystals Are Explained by Solubility Product and Solution Complexation. Cryst. Growth Des. 2006, 6 (2), 592-600.
    • (2006) Cryst. Growth Des. , vol.6 , Issue.2 , pp. 592-600
    • Nehm, S.J.1    Rodriguez-Spong, B.2    Rodriguez-Hornedo, N.3
  • 34
    • 68949135612 scopus 로고    scopus 로고
    • Cocrystal formation in solution: In situ solute concentration monitoring of the two components and kinetic pathways
    • Gagniere, E.; Mangin, D.; Puel, F.; Bebon, C.; Klein, J.-P.; Monnier, O.; Garcia, E. Cocrystal Formation in Solution: In Situ Solute Concentration Monitoring of the Two Components and Kinetic Pathways. Cryst. Growth Des. 2009, 9 (8), 3376-3383.
    • (2009) Cryst. Growth Des. , vol.9 , Issue.8 , pp. 3376-3383
    • Gagniere, E.1    Mangin, D.2    Puel, F.3    Bebon, C.4    Klein, J.-P.5    Monnier, O.6    Garcia, E.7


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.