메뉴 건너뛰기




Volumn 100, Issue 11, 2009, Pages 2188-2192

Evaluation of radioiodinated vesamicol analogs for sigma receptor imaging in tumor and radionuclide receptor therapy

Author keywords

[No Author keywords available]

Indexed keywords

1 (3,4 DIMETHOXYPHENETHYL) 4 (3 PHENYLPROPYL)PIPERAZINE; 2 [4 (4 IODOPHENYL)PIPERIDINO] CYCLOHEXANOL; HALOPERIDOL; RADIOACTIVE IODINE; SIGMA OPIATE RECEPTOR; UNCLASSIFIED DRUG; VESAMICOL DERIVATIVE;

EID: 71049136859     PISSN: 13479032     EISSN: 13497006     Source Type: Journal    
DOI: 10.1111/j.1349-7006.2009.01279.x     Document Type: Article
Times cited : (34)

References (28)
  • 2
    • 0029797712 scopus 로고    scopus 로고
    • Purification, molecular cloning, and expression of the mammalian sigma1-binding site
    • Hanner M, Moebius FF, Flandorfer A. Purification, molecular cloning, and expression of the mammalian sigma1-binding site. Proc Natl Acad Sci USA 1996, 93:8072-7.
    • (1996) Proc Natl Acad Sci USA , vol.93 , pp. 8072-8077
    • Hanner, M.1    Moebius, F.F.2    Flandorfer, A.3    et al4
  • 4
    • 0027853934 scopus 로고
    • Delineating biochemical and functional properties of sigma receptors: emerging concepts
    • Su TP. Delineating biochemical and functional properties of sigma receptors: emerging concepts. Crit Rev Neurobiol 1993, 7:187-203.
    • (1993) Crit Rev Neurobiol , vol.7 , pp. 187-203
    • Su, T.P.1
  • 5
    • 0028795145 scopus 로고
    • Sigma-1 and sigma-2 receptors are expressed in a wide variety of human and rodent tumor cell lines
    • Vilner BJ, John CS, Bowen WD. Sigma-1 and sigma-2 receptors are expressed in a wide variety of human and rodent tumor cell lines. Cancer Res 1995, 55:408-13.
    • (1995) Cancer Res , vol.55 , pp. 408-413
    • Vilner, B.J.1    John, C.S.2    Bowen, W.D.3
  • 6
    • 0026332936 scopus 로고
    • Overexpression of sigma receptors in nonneural human tumors
    • Bem WT, Thomas GE, Mamone JY. Overexpression of sigma receptors in nonneural human tumors. Cancer Res 1991, 51:6558-62.
    • (1991) Cancer Res , vol.51 , pp. 6558-6562
    • Bem, W.T.1    Thomas, G.E.2    Mamone, J.Y.3    et al4
  • 8
    • 0034010937 scopus 로고    scopus 로고
    • Sigma-2 receptors as a biomarker of proliferation in solid tumours
    • Wheeler KT, Wang LM, Wallen CA. Sigma-2 receptors as a biomarker of proliferation in solid tumours. Br J Cancer 2000, 82:1223-32.
    • (2000) Br J Cancer , vol.82 , pp. 1223-1232
    • Wheeler, K.T.1    Wang, L.M.2    Wallen, C.A.3    et al4
  • 9
    • 44349135064 scopus 로고    scopus 로고
    • Evaluation of radioiodinated 1-[2-(3,4-Dimethoxyphenyl) ethyl]-4-(2-iodophenylpropyl) piperazine as a tumor diagnostic agent with functional sigma receptor imaging by single photon emission computed tomography
    • Hirata M, Mori T, Umeda T, Abe T, Yamamoto T, Ohmomo Y. Evaluation of radioiodinated 1-[2-(3,4-Dimethoxyphenyl) ethyl]-4-(2-iodophenylpropyl) piperazine as a tumor diagnostic agent with functional sigma receptor imaging by single photon emission computed tomography. Biol Pharm Bull 2008, 31:879-83.
    • (2008) Biol Pharm Bull , vol.31 , pp. 879-883
    • Hirata, M.1    Mori, T.2    Umeda, T.3    Abe, T.4    Yamamoto, T.5    Ohmomo, Y.6
  • 10
    • 34547748903 scopus 로고    scopus 로고
    • Rapid reduction of sigma1-receptor binding and 18F-FDG uptake in rat gliomas after in vivo treatment with doxorubicin
    • van Waarde A, Shiba K, de Jong JR, Ishiwata K, Dierckx RA, Elsinga PH. Rapid reduction of sigma1-receptor binding and 18F-FDG uptake in rat gliomas after in vivo treatment with doxorubicin. J Nucl Med 2007, 48:1320-6.
    • (2007) J Nucl Med , vol.48 , pp. 1320-1326
    • van Waarde, A.1    Shiba, K.2    de Jong, J.R.3    Ishiwata, K.4    Dierckx, R.A.5    Elsinga, P.H.6
  • 11
    • 0037119033 scopus 로고    scopus 로고
    • Characterization of radioiodinated (-)-ortho-iodovesamicol binding in rat brain preparations
    • Shiba K, Yano T, Sato W, Mori H, Tonami N. Characterization of radioiodinated (-)-ortho-iodovesamicol binding in rat brain preparations. Life Sci 2002, 71:1591-8.
    • (2002) Life Sci , vol.71 , pp. 1591-1598
    • Shiba, K.1    Yano, T.2    Sato, W.3    Mori, H.4    Tonami, N.5
  • 12
    • 12844269941 scopus 로고    scopus 로고
    • In vitro characterization of radioiodinated (+)-2-[4-(4-iodophenyl) piperidino]cyclohexanol [(+)-pIV] as a sigma-1 receptor ligand
    • Shiba K, Ogawa K, Mori H. In vitro characterization of radioiodinated (+)-2-[4-(4-iodophenyl) piperidino]cyclohexanol [(+)-pIV] as a sigma-1 receptor ligand. Bioorg Med Chem 2005, 13:1095-9.
    • (2005) Bioorg Med Chem , vol.13 , pp. 1095-1099
    • Shiba, K.1    Ogawa, K.2    Mori, H.3
  • 13
    • 0033567923 scopus 로고    scopus 로고
    • Targeting sigma receptor-binding benzamides as in vivo diagnostic and therapeutic agents for human prostate tumors
    • John CS, Vilner BJ, Geyer BC, Moody T, Bowen WD. Targeting sigma receptor-binding benzamides as in vivo diagnostic and therapeutic agents for human prostate tumors. Cancer Res 1999, 59:4578-83.
    • (1999) Cancer Res , vol.59 , pp. 4578-4583
    • John, C.S.1    Vilner, B.J.2    Geyer, B.C.3    Moody, T.4    Bowen, W.D.5
  • 14
    • 0028955134 scopus 로고
    • Synthesis of radioiodinated analogs of 2-(4-phenylpiperidino) cyclohexanol (vesamicol) as vesamicol-like agent
    • Shiba K, Mori H, Matsuda H. Synthesis of radioiodinated analogs of 2-(4-phenylpiperidino) cyclohexanol (vesamicol) as vesamicol-like agent. Nucl Med Biol 1995, 22:205-10.
    • (1995) Nucl Med Biol , vol.22 , pp. 205-210
    • Shiba, K.1    Mori, H.2    Matsuda, H.3    et al4
  • 15
    • 0024328329 scopus 로고
    • Synthesis, in vitro acetylcholine-storage-blocking activities, and biological properties of derivatives and analogues of trans-2-(4-phenylpiperidino) cyclohexanol (vesamicol)
    • Rogers GA, Parsons SM, Anderson DC. Synthesis, in vitro acetylcholine-storage-blocking activities, and biological properties of derivatives and analogues of trans-2-(4-phenylpiperidino) cyclohexanol (vesamicol). J Med Chem 1989, 32:1217-30.
    • (1989) J Med Chem , vol.32 , pp. 1217-1230
    • Rogers, G.A.1    Parsons, S.M.2    Anderson, D.C.3    et al4
  • 16
    • 37349102472 scopus 로고    scopus 로고
    • A change of in vivo characteristics depending on specific activity of radioiodinated (+)-2-[4-(4-iodophenyl) piperidino]cyclohexanol [(+)-pIV] as a ligand for sigma receptor imaging
    • Akhter N, Shiba K, Ogawa K. A change of in vivo characteristics depending on specific activity of radioiodinated (+)-2-[4-(4-iodophenyl) piperidino]cyclohexanol [(+)-pIV] as a ligand for sigma receptor imaging. Nucl Med Biol 2008, 35:29-34.
    • (2008) Nucl Med Biol , vol.35 , pp. 29-34
    • Akhter, N.1    Shiba, K.2    Ogawa, K.3    et al4
  • 17
    • 33644785824 scopus 로고    scopus 로고
    • Synthesis and binding affinities of methylvesamicol analogs for the acetylcholine transporter and sigma receptor
    • Shiba K, Ogawa K, Ishiwata K, Yajima K, Mori H. Synthesis and binding affinities of methylvesamicol analogs for the acetylcholine transporter and sigma receptor. Bioorg Med Chem 2006, 14:2620-6.
    • (2006) Bioorg Med Chem , vol.14 , pp. 2620-2626
    • Shiba, K.1    Ogawa, K.2    Ishiwata, K.3    Yajima, K.4    Mori, H.5
  • 18
    • 0035255404 scopus 로고    scopus 로고
    • An admonition when measuring the lipophilicity of radiotracers using counting techniques
    • Wilson AA, Jin L, Garcia A, DaSilva JN, Houle S. An admonition when measuring the lipophilicity of radiotracers using counting techniques. Appl Radiat Isot 2001, 54:203-8.
    • (2001) Appl Radiat Isot , vol.54 , pp. 203-208
    • Wilson, A.A.1    Jin, L.2    Garcia, A.3    DaSilva, J.N.4    Houle, S.5
  • 19
    • 33646547897 scopus 로고    scopus 로고
    • Rhenium-186-monoaminemonoamidedithiol-conjugated bisphosphonate derivatives for bone pain palliation
    • Ogawa K, Mukai T, Arano Y. Rhenium-186-monoaminemonoamidedithiol-conjugated bisphosphonate derivatives for bone pain palliation. Nucl Med Biol 2006, 33:513-20.
    • (2006) Nucl Med Biol , vol.33 , pp. 513-520
    • Ogawa, K.1    Mukai, T.2    Arano, Y.3    et al4
  • 20
    • 33749343263 scopus 로고    scopus 로고
    • The expression and functional characterization of sigma 1 receptors in breast cancer cell lines
    • Aydar E, Onganer P, Perrett R, Djamgoz MB, Palmer CP. The expression and functional characterization of sigma 1 receptors in breast cancer cell lines. Cancer Lett 2006, 242:245-57.
    • (2006) Cancer Lett , vol.242 , pp. 245-257
    • Aydar, E.1    Onganer, P.2    Perrett, R.3    Djamgoz, M.B.4    Palmer, C.P.5
  • 21
    • 20744437475 scopus 로고    scopus 로고
    • Carbon-11 labeled sigma 2 receptor ligands for imaging breast cancer
    • Tu Z, Dence CS, Ponde DE. Carbon-11 labeled sigma 2 receptor ligands for imaging breast cancer. Nucl Med Biol 2005, 32:423-30.
    • (2005) Nucl Med Biol , vol.32 , pp. 423-430
    • Tu, Z.1    Dence, C.S.2    Ponde, D.E.3    et al4
  • 22
    • 33749852123 scopus 로고    scopus 로고
    • Sigma receptor ligands: possible application as therapeutic drugs and as radiopharmaceuticals
    • Hashimoto K, Ishiwata K. Sigma receptor ligands: possible application as therapeutic drugs and as radiopharmaceuticals. Curr Pharm Des 2006, 12:3857-76.
    • (2006) Curr Pharm Des , vol.12 , pp. 3857-3876
    • Hashimoto, K.1    Ishiwata, K.2
  • 23
    • 0028180570 scopus 로고
    • Rat liver and kidney contain high densities of sigma 1 and sigma 2 receptors: characterization by ligand binding and photoaffinity labeling
    • Hellewell SB, Bruce A, Feinstein G, Orringer J, Williams W, Bowen WD. Rat liver and kidney contain high densities of sigma 1 and sigma 2 receptors: characterization by ligand binding and photoaffinity labeling. Eur J Pharmacol 1994, 268:9-18.
    • (1994) Eur J Pharmacol , vol.268 , pp. 9-18
    • Hellewell, S.B.1    Bruce, A.2    Feinstein, G.3    Orringer, J.4    Williams, W.5    Bowen, W.D.6
  • 24
    • 0035005333 scopus 로고    scopus 로고
    • [18F]N-4′-fluorobenzyl-4-(3-bromophenyl) acetamide for imaging the sigma receptor status of tumors: comparison with [18F]FDG, and [125I]IUDR
    • Mach RH, Huang Y, Buchheimer N. [18F]N-4′-fluorobenzyl-4-(3-bromophenyl) acetamide for imaging the sigma receptor status of tumors: comparison with [18F]FDG, and [125I]IUDR. Nucl Med Biol 2001, 28:451-8.
    • (2001) Nucl Med Biol , vol.28 , pp. 451-458
    • Mach, R.H.1    Huang, Y.2    Buchheimer, N.3    et al4
  • 26
    • 0029862067 scopus 로고    scopus 로고
    • Structure distribution relationship of iodine-123-iodobenzamides as tracers for the detection of melanotic melanoma
    • Brandau W, Niehoff T, Pulawski P. Structure distribution relationship of iodine-123-iodobenzamides as tracers for the detection of melanotic melanoma. J Nucl Med 1996, 37:1865-71.
    • (1996) J Nucl Med , vol.37 , pp. 1865-1871
    • Brandau, W.1    Niehoff, T.2    Pulawski, P.3    et al4
  • 27
    • 31744445492 scopus 로고    scopus 로고
    • Evaluation of [11C]SA5845 and [11C]SA4503 for imaging of sigma receptors in tumors by animal PET
    • Kawamura K, Kubota K, Kobayashi T. Evaluation of [11C]SA5845 and [11C]SA4503 for imaging of sigma receptors in tumors by animal PET. Ann Nucl Med 2005, 19:701-9.
    • (2005) Ann Nucl Med , vol.19 , pp. 701-709
    • Kawamura, K.1    Kubota, K.2    Kobayashi, T.3    et al4
  • 28
    • 0030610886 scopus 로고    scopus 로고
    • In vivo evaluation of [18F]1-(3-fluoropropyl)-4-(4-cyanophenoxymethyl) piperidine: a selective sigma-1 receptor radioligand for PET
    • Waterhouse RN, Collier TL. In vivo evaluation of [18F]1-(3-fluoropropyl)-4-(4-cyanophenoxymethyl) piperidine: a selective sigma-1 receptor radioligand for PET. Nucl Med Biol 1997, 24:127-34.
    • (1997) Nucl Med Biol , vol.24 , pp. 127-134
    • Waterhouse, R.N.1    Collier, T.L.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.