Presence of a putative steroidal allosteric site on glycoprotein hormone receptors

European Journal of Pharmacology

Volumn 623, Issue 1-3, 2009, Pages 155-159

  Rossi, Mario ^a   Dimida, Antonio ^a   Ferrarini, Eleonora ^a   Silvano, Elena ^b   De Marco, Giuseppina ^a   Agretti, Patrizia ^a   Aloisi, Gabriella ^b   Simoncini, Tommaso ^a   Di Bari, Lorenzo ^a   Tonacchera, Massimo ^a   Giorgi, Franco ^a   Maggio, Roberto ^b  

^a UNIVERSITY OF PISA   (Italy)

^b UNIVERSITY OF L'AQUILA   (Italy)

Author keywords

Adenylyl cyclase; Allosteric compound; Luteinizing hormone receptor; Steroid; Steroid receptor; Thyroid stimulating hormone receptor

Indexed keywords

CHLORPHENOTANE; CHORIONIC GONADOTROPIN; CYCLIC AMP; DIETHYLSTILBESTROL; ESTRADIOL; ESTROGEN RECEPTOR; ESTROGEN RECEPTOR ALPHA; ESTROGEN RECEPTOR BETA; LUTEINIZING HORMONE RECEPTOR; QUERCETIN; THYROTROPIN RECEPTOR;

ANIMAL CELL; ARTICLE; BINDING SITE; CELL STIMULATION; CELL STRAIN COS7; CHO CELL; CONCENTRATION RESPONSE; CONTROLLED STUDY; GENETIC TRANSFECTION; NONHUMAN; PRIORITY JOURNAL; PROTEIN ANALYSIS; PROTEIN ASSEMBLY; RAT;

ADENYLATE CYCLASE; ALLOSTERIC SITE; ANIMALS; CELL LINE; CERCOPITHECUS AETHIOPS; CHO CELLS; CHORIONIC GONADOTROPIN; COS CELLS; CRICETINAE; CRICETULUS; CYCLIC AMP; DDT; DIETHYLSTILBESTROL; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG EVALUATION, PRECLINICAL; ESTRADIOL; ESTROGENS; ISOENZYMES; PROTEIN BINDING; QUERCETIN; RATS; RATS, INBRED F344; RECEPTORS, CYTOPLASMIC AND NUCLEAR; RECEPTORS, ESTROGEN; RECEPTORS, LH; RECEPTORS, THYROTROPIN; STEROIDS; STRUCTURE-ACTIVITY RELATIONSHIP; THYROTROPIN;

EID: 70350303317     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejphar.2009.09.029     Document Type: Article

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