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Volumn 77, Issue 3, 2009, Pages 695-709

Molecular mobility and physical stability of amorphous irbesartan

Author keywords

Amorphous form; DSC; Enthalpy relaxation; Irbesartan; Molecular mobility; Stability

Indexed keywords

IRBESARTAN;

EID: 70349272483     PISSN: 00368709     EISSN: 22180532     Source Type: Journal    
DOI: 10.3797/scipharm.0806-09     Document Type: Article
Times cited : (13)

References (22)
  • 1
    • 0031749397 scopus 로고    scopus 로고
    • A pragmatic tool of a simple calorimetric method for determining the fragility of some amorphous pharmaceutical materials
    • doi:10.1023/A:1011931305755
    • Hancock BC, Dalton CR, Pikal MJ, Shamblin SL. A pragmatic tool of a simple calorimetric method for determining the fragility of some amorphous pharmaceutical materials. Pharm Res. 1998: 15: 762-767. doi:10.1023/A: 1011931305755
    • (1998) Pharm Res , vol.15 , pp. 762-767
    • Hancock, B.C.1    Dalton, C.R.2    Pikal, M.J.3    Shamblin, S.L.4
  • 2
    • 0035997888 scopus 로고    scopus 로고
    • Disordered drug delivery: Destiny, dynamics and the Deborah number
    • doi:10.1211/0022357021778989
    • Hancock BC. Disordered drug delivery: destiny, dynamics and the Deborah number. J Pharm Pharmacol. 2002; 54: 737-746. doi:10.1211/0022357021778989
    • (2002) J Pharm Pharmacol , vol.54 , pp. 737-746
    • Hancock, B.C.1
  • 3
    • 33646689478 scopus 로고    scopus 로고
    • Structural relaxation of acetaminophen glass
    • doi:10.1007/s11095-006-9898-0
    • Gunawan L, Johari GP, Shankar RM. Structural relaxation of acetaminophen glass. Pharm Res. 2006; 23: 967-979. doi:10.1007/s11095-006-9898-0
    • (2006) Pharm Res , vol.23 , pp. 967-979
    • Gunawan, L.1    Johari, G.P.2    Shankar, R.M.3
  • 4
    • 0034019632 scopus 로고    scopus 로고
    • Interpretation of relaxation time constants for amorphous pharmaceutical systems
    • DOI 10.1002/(SICI)1520-6017(200003)89:3<417::AID-JPS12>3.0.CO;2-V
    • Shamblin SL, Hancock BC, Dupuis Y, Pikal MJ. Interpretation of relaxation time constants for amorphous pharmaceutical systems. J Pharm Sci. 2000; 89: 417-427. doi:10.1002/(SICI)1520-6017(200003)89:3〈417::AID-JPS12〉3.0. CO;2-V (Pubitemid 30152441)
    • (2000) Journal of Pharmaceutical Sciences , vol.89 , Issue.3 , pp. 417-427
    • Shamblin, S.L.1    Hancock, B.C.2    Dupuis, Y.3    Pikal, M.J.4
  • 5
    • 0031056536 scopus 로고    scopus 로고
    • Effects of sorbed water on the crystallization of indomethacin from the amorphous state
    • DOI 10.1021/js9602711
    • Andronis V, Yoshioka M, Zografi G. Effect of absorbed water on crystallization of of indomethacin from the amorphous state. J Pharm Sci. 1997; 86: 346-351. doi:10.1021/js9602711 (Pubitemid 27113770)
    • (1997) Journal of Pharmaceutical Sciences , vol.86 , Issue.3 , pp. 346-357
    • Andronis, V.1    Yoshioka, M.2    Zografi, G.3
  • 6
    • 0034061182 scopus 로고    scopus 로고
    • 1H NMR relaxation times
    • doi:10.1002/(SICI)1520-6017(200003)89:3〈408::AID-JPS11〉3.0. CO;2-#
    • 1H NMR relaxation times. J Pharm Sci. 2000; 89: 408-416. doi:10.1002/(SICI)1520-6017(200003)89:3〈408::AID- JPS11〉3.0.CO;2-#
    • (2000) J Pharm Sci , vol.89 , pp. 408-416
    • Aso, Y.1    Yoshioka, S.2    Kojima, S.3
  • 7
    • 0024404092 scopus 로고
    • Glassy state of pharmaceuticals. III. Thermal properties and stability of glassy pharmaceuticals and their binary glassy systems
    • Fukuoka E, Matika M, Yamamura S. Glassy state of pharmaceuticals. III. Thermal properties and stability of glassy pharmaceuticals and their binary glassy systems. Chem Pharm Bull. 1989; 37: 1047-1050.
    • (1989) Chem Pharm Bull , vol.37 , pp. 1047-1050
    • Fukuoka, E.1    Matika, M.2    Yamamura, S.3
  • 8
    • 0028268210 scopus 로고
    • The relationship between the glass transition temperature and the water content of amorphous pharmaceutical solids
    • DOI 10.1023/A:1018941810744
    • Yoshioka M, Hancock B, Zografi G. Crystallization of indomethacin from the amorphous stet below and above its glass transition temperature. J Pharm Sci. 1994; 83: 1700-1705. doi:10.1002/jps.2600831211 (Pubitemid 24144434)
    • (1994) Pharmaceutical Research , vol.11 , Issue.4 , pp. 471-477
    • Hancock, B.C.1    Zografi, G.2
  • 9
    • 0027174285 scopus 로고
    • Molecular mobility in mixtures of absorbed water and solid poly(vinylpyrrolidone)
    • DOI 10.1023/A:1018988506336
    • Oksanen C, Zografi G. Molecular mobility in mixtures of absorbed water and solid poly(vinylpyrolidone). Pharm Res. 1993; 10: 791-799. doi:10.1023/A:1018988506336 (Pubitemid 23167558)
    • (1993) Pharmaceutical Research , vol.10 , Issue.6 , pp. 791-799
    • Oksanen, C.A.1    Zografi, G.2
  • 10
    • 0025102704 scopus 로고
    • The molecular basis of moisture effects on the physical and chemical stability of drugs in the solid state
    • DOI 10.1016/0378-5173(90)90221-O
    • Ahlneck C, Zografi G. The molecular basis of moisture effects on the physical and chemical stability of drugs in the solid state. Int J Pharm. 1990; 62: 87-95. doi:10.1016/0378-5173(90)90221-O (Pubitemid 20261777)
    • (1990) International Journal of Pharmaceutics , vol.62 , Issue.2-3 , pp. 87-95
    • Ahlneck, C.1    Zografi, G.2
  • 11
    • 34548672900 scopus 로고    scopus 로고
    • A comparative assessment of solubility advantage from glassy and crystalline forms of a water-insoluble drug
    • DOI 10.1016/j.ejps.2007.05.111, PII S0928098707002515
    • Chawla G, Bansal AK. A comparative assessment of solubility advantage from glassy and crystalline forms of a water-insoluble drug. Eur J Pharm Sci. 2007; 32: 45-57. doi:10.1016/j.ejps.2007.05.111 (Pubitemid 47411498)
    • (2007) European Journal of Pharmaceutical Sciences , vol.32 , Issue.1 , pp. 45-57
    • Chawla, G.1    Bansal, A.K.2
  • 12
    • 0034886795 scopus 로고    scopus 로고
    • Physicochemical considerations in the preparation of amorphous ritonavir-poly(ethylene glycol) 8000 solid dispersions
    • doi:10.1002/jps.1054
    • Law B, Krill SL, Schmitt EA, Fort JJ, Qiu Y, Wang W, Porter WR. Physicochemical considerations in the preparation of amorphous ritonavir-poly(ethylene glycol) 8000 solid dispersions. J Pharm Sci. 2001; 90: 1015-1025. doi:10.1002/jps.1054
    • (2001) J Pharm Sci , vol.90 , pp. 1015-1025
    • Law, B.1    Krill, S.L.2    Schmitt, E.A.3    Fort, J.J.4    Qiu, Y.5    Wang, W.6    Porter, W.R.7
  • 13
    • 0035991640 scopus 로고    scopus 로고
    • Physical stability of amorphous pharmaceuticals: Importance of configurational thermodynamic quantities and molecular mobility
    • DOI 10.1002/jps.10169
    • Zhou D, Zhang GGZ, Law D, Grant DJW, Schmitt EA. Physical stability of amorphous pharmaceuticals: Importance of configurational thermodynamic quantities and molecular mobility. J Pharm Sci. 2002; 91: 1863-1872. doi:10.1002/jps.10169 (Pubitemid 34810531)
    • (2002) Journal of Pharmaceutical Sciences , vol.91 , Issue.8 , pp. 1863-1872
    • Zhou, D.1    Zhang, G.G.Z.2    Law, D.3    Grant, D.J.W.4    Schmitt, E.A.5
  • 14
    • 0030217476 scopus 로고    scopus 로고
    • Supercooled liquids and glasses
    • doi:10.1021/jp953538d
    • Ediger MD, Angell CA, Nagel SR. Supercooled liquids and glasses. J Phys Chem. 1996; 100: 13200-13212. doi:10.1021/jp953538d
    • (1996) J Phys Chem , vol.100 , pp. 13200-13212
    • Ediger, M.D.1    Angell, C.A.2    Nagel, S.R.3
  • 15
    • 33749435820 scopus 로고    scopus 로고
    • A calorimetric method to estimate molecular mobility of amorphous solids at relatively low temperatures
    • DOI 10.1007/s11095-006-9071-9
    • Mao C, Chamarthy SP, Byrn SR, Pinal R. A calorimetric method to estimate molecular mobility of amorphous solids at relatively low temperatures. Pharm Res. 2006; 23: 2269-2276. doi:10.1007/s11095-006-9071-9 (Pubitemid 44511508)
    • (2006) Pharmaceutical Research , vol.23 , Issue.10 , pp. 2269-2276
    • Mao, C.1    Prasanth Chamarthy, S.2    Byrn, S.R.3    Pinal, R.4
  • 16
    • 0035861398 scopus 로고    scopus 로고
    • Molecular mobility of amorphous pharmaceuticals determined using differential scanning calorimetry
    • DOI 10.1016/S0040-6031(01)00663-3, PII S0040603101006633
    • Hancock B, Shamblin S. Molecular mobility of amorphous pharmaceuticals determined using differential scanning calorimetry. Thermochim Acta. 2001; 380: 95-107. doi:10.1016/S0040-6031(01)00663-3 (Pubitemid 33096427)
    • (2001) Thermochimica Acta , vol.380 , Issue.2 , pp. 95-107
    • Hancock, B.C.1    Shamblin, S.L.2
  • 17
    • 33751124528 scopus 로고
    • Nonexponential relaxations in strong and fragile glass formers
    • doi:10.1063/1.466117
    • Bohmer R, Ngai KL, Angell CA, Plazek DJ. Nonexponential relaxations in strong and fragile glass formers. J Chem Phys. 1993; 99: 4201-4209. doi:10.1063/1.466117
    • (1993) J Chem Phys , vol.99 , pp. 4201-4209
    • Bohmer, R.1    Ngai, K.L.2    Angell, C.A.3    Plazek, D.J.4
  • 18
    • 0001182230 scopus 로고    scopus 로고
    • Characterization of the time scales of molecular motion in pharmaceutically important glasses
    • Shamblin SL, Tang X, Chang L, Hancock BC, Pikal MJ. Characterization of the time scales of molecular motion in pharmaceutically important glasses. J Phys Chem B. 1999; 103: 4113-4121. doi:10.1021/jp983964+ (Pubitemid 129702538)
    • (1999) Journal of Physical Chemistry B , vol.103 , Issue.20 , pp. 4113-4121
    • Shamblin, S.L.1    Tang, X.2    Chang, L.3    Hancock, B.C.4    Pikal, M.J.5
  • 19
    • 0035897584 scopus 로고    scopus 로고
    • Amorphous pharmaceutical solids: Preparation, characterization and stabilization
    • DOI 10.1016/S0169-409X(01)00098-9, PII S0169409X01000989
    • Yu L. Amorphous pharmaceutical solids: preparation, characterization and stabilization. Adv Drug Del Rev. 2001; 48: 27-42. doi:10.1016/S0169-409X(01) 00098-9 (Pubitemid 32454482)
    • (2001) Advanced Drug Delivery Reviews , vol.48 , Issue.1 , pp. 27-42
    • Yu, L.1
  • 20
    • 0030638567 scopus 로고    scopus 로고
    • Characteristics and Significance of the Amorphous State in Pharmaceutical Systems
    • Hancock BC, Zografi G. Characteristics and significance of the amorphous state in pharmaceutical systems. J Pharm Sci. 1997; 86: 1-12. doi:10.1021/js9601896 (Pubitemid 127489650)
    • (1997) Journal of Pharmaceutical Sciences , vol.86 , Issue.1
    • Hancock, B.C.1    Zografi, G.2
  • 21
    • 33344473894 scopus 로고    scopus 로고
    • Characterization of the molecular distribution of drugs in glassy solid dispersions at the nano-meter scale, using differential scanning calorimetry and gravimetric water vapour sorption techniques
    • DOI 10.1016/j.ijpharm.2005.12.007, PII S0378517305008203
    • Drooge D, Hinrichs W, Visser M, Frijlink H. Characterization of the molecular distribution of drugs in glassy solid dispersions at the nano-meter scale, using differential scanning calorimetry and gravimetric water vapour sorption techniques. Int J Pharm. 2006; 310: 220-229. doi:10.1016/j.ijpharm. 2005.12.007 (Pubitemid 43287987)
    • (2006) International Journal of Pharmaceutics , vol.310 , Issue.1-2 , pp. 220-229
    • Van Drooge, D.J.1    Hinrichs, W.L.J.2    Visser, M.R.3    Frijlink, H.W.4
  • 22
    • 0032745368 scopus 로고    scopus 로고
    • Characterisation of moisture uptake effects on the glass transitional behavior of an amorphous drug using modulated temperature DSC
    • doi:10.1016/S0378-5173(99)00270-7
    • Royall PG, Craig DCM, Doherty C. Characterisation of moisture uptake effects on the glass transitional behavior of an amorphous drug using modulated temperature DSC. Int J Pharm. 1999; 192: 39-46. doi:10.1016/S0378-5173(99)00270- 7
    • (1999) Int J Pharm , vol.192 , pp. 39-46
    • Royall, P.G.1    Craig, D.C.M.2    Doherty, C.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.