Amiodarone and its putative metabolites fail to activate wild type hTAAR1

Bioorganic and Medicinal Chemistry Letters

Volumn 19, Issue 20, 2009, Pages 5913-5914

  Lewin, Anita H ^a   Navarro, Hernán A ^a   Gilmour, Brian P ^a  

^a RTI INTERNATIONAL   (United States)

Author keywords

Amiodarone; G protein coupled receptors; hTAAR1; Human trace amine associated receptor 1

Indexed keywords

AMIODARONE; CYCLIC AMP; DRUG METABOLITE; G PROTEIN COUPLED RECEPTOR; PHENETHYLAMINE; PROTEIN TAAR1; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CONTROLLED STUDY; DRUG IDENTIFICATION; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME ACTIVATION; HUMAN; HUMAN CELL; NONHUMAN; PROTEIN EXPRESSION;

AMIODARONE; ANIMALS; CHO CELLS; CRICETINAE; CRICETULUS; HUMANS; RATS; RECEPTORS, G-PROTEIN-COUPLED; TRANSFECTION;

RODENTIA;

EID: 70349264146     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2009.08.058     Document Type: Article

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