Trace amine-associated receptor 1 (TAAR1) is activated by amiodarone metabolites

Bioorganic and Medicinal Chemistry Letters

Volumn 18, Issue 22, 2008, Pages 5920-5922

  Snead, Aaron N ^a   Miyakawa, Motonori ^a   Tan, Edwin S ^a   Scanlan, Thomas S ^a,b  

^a UNIVERSITY OF CALIFORNIA   (United States)

^b OREGON HEALTH AND SCIENCE UNIVERSITY   (United States)

Author keywords

Amiodarone; G protein coupled receptors; TAAR1; Trace amine associated receptor 1

Indexed keywords

AMIODARONE; DRUG METABOLITE; G PROTEIN COUPLED RECEPTOR; IODOTHYRONAMINE; THYROID HORMONE; THYROID HORMONE DERIVATIVE; TRACE AMINE ASSOCIATED RECEPTOR 1; UNCLASSIFIED DRUG;

AGONIST; ARTICLE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; HUMAN CELL; STRUCTURE ACTIVITY RELATION;

AMIODARONE; ANIMALS; ANTI-ARRHYTHMIA AGENTS; ARRHYTHMIAS, CARDIAC; COMBINATORIAL CHEMISTRY TECHNIQUES; HUMANS; MICE; MOLECULAR STRUCTURE; RATS; RECEPTORS, G-PROTEIN-COUPLED;

EID: 55249125403     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2008.08.013     Document Type: Article

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