메뉴 건너뛰기




Volumn 18, Issue 7, 2009, Pages 523-537

Prediction of antiproliferative activity of some flavone derivatives: QSAR study

Author keywords

Anticancer; Antiproliferative activity; Flavone; Isoflavone; Quantitative structure activity relationship

Indexed keywords

ANTINEOPLASTIC AGENT; FLAVONE 3 YL DERIVATIVE; FLAVONE 6 YL DERIVATIVE; FLAVONE 7 YL DERIVATIVE; FLAVONE DERIVATIVE; ISOFLAVONE 7 YL DERIVATIVE; ISOFLAVONE DERIVATIVE; OXIME DERIVATIVE; UNCLASSIFIED DRUG;

EID: 70349257449     PISSN: 10542523     EISSN: None     Source Type: Journal    
DOI: 10.1007/s00044-008-9146-8     Document Type: Article
Times cited : (5)

References (21)
  • 1
    • 0346887168 scopus 로고    scopus 로고
    • Antiproliferative activity of various flavonoids and related compounds: Additive effect of interferon-α2b
    • DOI 10.1016/j.bmcl.2003.10.029
    • VC Blank C Poli M Marder LP Roguin 2004 Antiproliferative activity of various flavonoids and related compounds: additive effect of interferon-alpha2b Bioorg Med Chem Lett 14 133 136 10.1016/j.bmcl.2003.10.029 14684314 10.1016/j.bmcl.2003.10.029 (Pubitemid 38010208)
    • (2004) Bioorganic and Medicinal Chemistry Letters , vol.14 , Issue.1 , pp. 133-136
    • Blank, V.C.1    Poli, C.2    Marder, M.3    Roguin, L.P.4
  • 2
    • 0037403574 scopus 로고    scopus 로고
    • Phenoxodiol, a novel isoflavone derivative, inhibits dimethylbenz[a] anthracene (DMBA)-induced mammary carcinogenesis in female Sprague-Dawley rats
    • DOI 10.1016/S0959-8049(03)00124-2
    • AI Constantinou R Mehta A Husband 2003 Phenoxodiol, a novel isoflavone derivative, inhibits dimethylbenz[a]anthracene (DMBA)-induced mammary carcinogenesis in female Sprague-Dawley rats Eur J Cancer 39 1012 1018 10.1016/S0959-8049(03)00124-2 12706372 10.1016/S0959-8049(03)00124-2 (Pubitemid 36428635)
    • (2003) European Journal of Cancer , vol.39 , Issue.7 , pp. 1012-1018
    • Constantinou, A.I.1    Mehta, R.2    Husband, A.3
  • 3
    • 33244472101 scopus 로고    scopus 로고
    • Silymarin and silibinin cause G1 and G2-M cell cycle arrest via distinct circuitries in human prostate cancer PC3 cells: A comparison of flavanone silibinin with flavanolignan mixture silymarin
    • DOI 10.1038/sj.onc.1209146, PII 1209146
    • G Deep RP Singh C Agrawal DJ Kroll R Agarwal 2006 Silymarin and silibinin cause G1 and G2-M cell cycle arrest via distinct circuitries in human prostate cancer PC3 cells: a comparison of flavanone silibinin with flavanolignan mixture silymarin Oncogene 25 1053 1069 10.1038/sj.onc.1209146 16205633 10.1038/sj.onc.1209146 (Pubitemid 43277013)
    • (2006) Oncogene , vol.25 , Issue.7 , pp. 1053-1069
    • Deep, G.1    Singh, R.P.2    Agarwal, C.3    Kroll, D.J.4    Agarwal, R.5
  • 4
    • 33947302242 scopus 로고    scopus 로고
    • The development of chalcones as promising anticancer agents
    • S Ducki 2007 The development of chalcones as promising anticancer agents Drugs 1 42 46
    • (2007) Drugs , vol.1 , pp. 42-46
    • Ducki, S.1
  • 5
    • 23844443498 scopus 로고    scopus 로고
    • Potential role of flavonoids in the prevention of intestinal neoplasia: A review of their mode of action and their clinical perspectives
    • 10.1385/IJGC:35:3:187 16110120 10.1385/IJGC:35:3:187
    • HP Hoensch W Kirch 2005 Potential role of flavonoids in the prevention of intestinal neoplasia: a review of their mode of action and their clinical perspectives Int J Gastrointest Cancer 35 187 195 10.1385/IJGC:35:3:187 16110120 10.1385/IJGC:35:3:187
    • (2005) Int J Gastrointest Cancer , vol.35 , pp. 187-195
    • Hoensch, H.P.1    Kirch, W.2
  • 6
    • 33748311541 scopus 로고    scopus 로고
    • QSAR analysis of Indomethacin derivatives as selective COX-2 inhibitors
    • HK Jain RK Agrawal 2004 QSAR analysis of Indomethacin derivatives as selective COX-2 inhibitors Int Elec J Mol Des 5 224 236
    • (2004) Int Elec J Mol Des , vol.5 , pp. 224-236
    • Jain, H.K.1    Agrawal, R.K.2
  • 7
    • 33748329448 scopus 로고    scopus 로고
    • Inhibitory mode of 2-acetoxyphenyl alkyl sulfides against COX-1 and COX-2: QSAR analyses
    • DOI 10.1016/j.bmcl.2006.08.002, PII S0960894X06008900
    • HK Jain VK Mourya RK Agrawal 2006 Inhibitory mode of 2-acetoxyphenyl alkyl sulfides against COX-1 and COX-2: QSAR analyses Bioorg Med Chem Lett 16 5280 5284 10.1016/j.bmcl.2006.08.002 16908140 10.1016/j.bmcl.2006.08.002 (Pubitemid 44332227)
    • (2006) Bioorganic and Medicinal Chemistry Letters , vol.16 , Issue.20 , pp. 5280-5284
    • Jain, H.K.1    Mourya, V.K.2    Agrawal, R.K.3
  • 9
    • 0036669812 scopus 로고    scopus 로고
    • Cancer preventive effects of flavonoids - A review
    • DOI 10.1016/S0753-3322(02)00186-5, PII S0753332202001865
    • L Le Marchand 2002 Cancer preventive effects of flavonoids-a review Biomed Pharmacother 56 296 301 10.1016/S0753-3322(02)00186-5 12224601 10.1016/S0753-3322(02)00186-5 (Pubitemid 35245313)
    • (2002) Biomedicine and Pharmacotherapy , vol.56 , Issue.6 , pp. 296-301
    • Le Marchand, L.1
  • 10
    • 33750720916 scopus 로고    scopus 로고
    • Apigenin suppresses cancer cell growth through ERβ
    • DOI 10.1593/neo.06538
    • P Mak YK Leung WY Tang C Harwood SM Ho 2006 Apigenin suppresses cancer cell growth through ERbeta Neoplasia 8 896 904 10.1593/neo.06538 17132221 10.1593/neo.06538 (Pubitemid 44706239)
    • (2006) Neoplasia , vol.8 , Issue.11 , pp. 896-904
    • Mak, P.1    Leung, Y.-K.2    Tang, W.-Y.3    Harwood, C.4    Ho, S.-M.5
  • 11
    • 35548940757 scopus 로고    scopus 로고
    • Identification of new flavone-8-acetic acid metabolites using mouse microsomes and comparison with human microsomes
    • DOI 10.1124/dmd.107.017012
    • MH Pham N Auzeil A Regezzetti D Dauzonne A Dugay MC Menet D Scherman GG Chabot 2007 Identification of new flavone-8-acetic acid metabolites using mouse microsomes and comparison with human microsomes Drug Metab Dispos 35 2023 2034 10.1124/dmd.107.017012 17664249 10.1124/dmd.107.017012 (Pubitemid 350005191)
    • (2007) Drug Metabolism and Disposition , vol.35 , Issue.11 , pp. 2023-2034
    • Minh, H.P.1    Auzeil, N.2    Regazzetti, A.3    Dauzonne, D.4    Dugay, A.5    Menet, M.-C.6    Scherman, D.7    Chabot, G.G.8
  • 12
    • 33947607163 scopus 로고    scopus 로고
    • Predicting anti-HIV activity of PETT derivatives: CoMFA approach
    • DOI 10.1016/j.bmcl.2007.01.103, PII S0960894X07001515
    • V Ravichandran RK Agrawal 2007 Predicting anti-HIV activity of PETT derivatives: CoMFA approach Bioorg Med Chem Lett 17 2197 10.1016/j.bmcl.2007.01. 103 17307357 10.1016/j.bmcl.2007.01.103 (Pubitemid 46484318)
    • (2007) Bioorganic and Medicinal Chemistry Letters , vol.17 , Issue.8 , pp. 2197-2202
    • Ravichandran, V.1    Agrawal, R.K.2
  • 13
    • 34548456464 scopus 로고    scopus 로고
    • QSAR study of novel 1,1,3 trioxo [1,2,4]-thiadiazine (TTDs) analogues as potent anti-HIV agents
    • V Ravichandran VK Mourya RK Agrawal 2007 QSAR study of novel 1,1,3 trioxo [1,2,4]-thiadiazine (TTDs) analogues as potent anti-HIV agents Arkivoc XIV 204 212
    • (2007) Arkivoc , vol.14 , pp. 204-212
    • Ravichandran, V.1    Mourya, V.K.2    Agrawal, R.K.3
  • 14
    • 0038807711 scopus 로고    scopus 로고
    • Flavonoids: Promising anticancer agents
    • DOI 10.1002/med.10033
    • W Ren Z Qiao H Wang L Zhu L Zhang 2003 Flavonoids: promising anticancer agents Med Res Rev 23 519 534 10.1002/med.10033 12710022 10.1002/med.10033 (Pubitemid 36706514)
    • (2003) Medicinal Research Reviews , vol.23 , Issue.4 , pp. 519-534
    • Ren, W.1    Qiao, Z.2    Wang, H.3    Zhu, L.4    Zhang, L.5
  • 15
    • 34948822189 scopus 로고    scopus 로고
    • QSAR analysis of caffeoyl naphthalene sulfonamide derivatives as HIV-1 integrase inhibitors
    • DOI 10.1007/s00044-006-0020-2
    • KK Sahu V Ravichandran VK Mourya RK Agrawal 2007 QSAR analysis of caffeoyl naphthalene sulfonamide derivatives as HIV-1 integrase inhibitors Med Chem Res 15 418 430 10.1007/s00044-006-0020-2 10.1007/s00044-006-0020-2 (Pubitemid 47522218)
    • (2007) Medicinal Chemistry Research , vol.15 , Issue.7-8 , pp. 418-430
    • Sahu, K.K.1    Ravichandran, V.2    Mourya, V.K.3    Agrawal, R.K.4
  • 16
    • 3242766866 scopus 로고    scopus 로고
    • 2+-mediated, calpain/caspase-12-dependent apoptosis in breast cancer cells
    • 10.1016/j.bbrc.2004.06.173 15358198 10.1016/j.bbrc.2004.06.173
    • 2+-mediated, calpain/caspase-12-dependent apoptosis in breast cancer cells Biochem Biophys Res Commun 321 462 467 10.1016/j.bbrc.2004.06.173 15358198 10.1016/j.bbrc.2004. 06.173
    • (2004) Biochem Biophys Res Commun , vol.321 , pp. 462-467
    • Sergeev, I.N.1
  • 17
    • 33845199356 scopus 로고    scopus 로고
    • 2+-mediated apoptosis in breast cancer cells
    • DOI 10.1016/j.lfs.2006.09.006, PII S0024320506007132
    • IN Sergeev S Li J Colby CT Ho S Dushenkov 2006 Polymethoxylated flavones induce Ca(2+)-mediated apoptosis in breast cancer cells Life Sci 80 245 253 10.1016/j.lfs.2006.09.006 17046027 10.1016/j.lfs.2006.09.006 (Pubitemid 44853992)
    • (2006) Life Sciences , vol.80 , Issue.3 , pp. 245-253
    • Sergeev, I.N.1    Li, S.2    Colby, J.3    Ho, C.-T.4    Dushenkov, S.5
  • 18
    • 46649101520 scopus 로고    scopus 로고
    • Prediction of caspase-3 inhibitory activity of 1,3-dioxo-4-methyl-2,3- dihydro-1h-pyrrolo[3,4-c] quinolines: QSAR study
    • DOI 10.1080/14756360701652476, PII 793954150
    • S Sharma V Ravichandran PK Jain VK Mourya RK Agrawal 2008 Prediction of caspase-3 inhibitory activity of 1,3-dioxo-4-methyl-2,3-dihydro-1 h-pyrrolo[3,4-c] quinolines: QSAR study J Enzyme Inhib Med Chem 23 424 431 10.1080/14756360701652476 18569350 10.1080/14756360701652476 (Pubitemid 351935066)
    • (2008) Journal of Enzyme Inhibition and Medicinal Chemistry , vol.23 , Issue.3 , pp. 424-431
    • Sharma, S.1    Ravichandran, V.2    Jain, P.3    Mourya, V.K.4    Agrawal, R.K.5
  • 19
    • 20444431504 scopus 로고    scopus 로고
    • The antitumor and antiangiogenic activity of vascular endothelial growth factor receptor inhibition is potentiated by ErbB1 blockade
    • DOI 10.1158/1078-0432.CCR-04-1954
    • P Sini L Wyder C Schnell T O'Reilly A Littlewood R Brandt NE Hynes J Wood 2005 The antitumor and antiangiogenic activity of vascular endothelial growth factor receptor inhibition is potentiated by ErbB1 blockade Clin Cancer Res 11 4521 4532 10.1158/1078-0432.CCR-04-1954 15958638 10.1158/1078-0432.CCR-04-1954 (Pubitemid 40825643)
    • (2005) Clinical Cancer Research , vol.11 , Issue.12 , pp. 4521-4532
    • Sini, P.1    Wyder, L.2    Schnell, C.3    O'Reilly, T.4    Littlewood, A.5    Brandt, R.6    Hynes, N.E.7    Wood, J.8
  • 20
    • 33750693398 scopus 로고    scopus 로고
    • Accumulation and metabolism of the anticancer flavonoid 5,7-dimethoxyflavone compared to its unmethylated analog chrysin in the Atlantic killifish
    • DOI 10.1016/j.cbi.2006.08.023, PII S0009279706002328
    • PA Tsuji RN Winn T Walle 2006 Accumulation and metabolism of the anticancer flavonoid 5,7-dimethoxyflavone compared to its unmethylated analog chrysin in the Atlantic killifish Chem Biol Interact 164 85 92 10.1016/j.cbi.2006.08.023 16999945 10.1016/j.cbi.2006.08.023 (Pubitemid 44709714)
    • (2006) Chemico-Biological Interactions , vol.164 , Issue.1-2 , pp. 85-92
    • Tsuji, P.A.1    Winn, R.N.2    Walle, T.3
  • 21
    • 25844486965 scopus 로고    scopus 로고
    • Synthesis, antiproliferative, and antiplatelet activities of oxime- and methyloxime-containing flavone and isoflavone derivatives
    • DOI 10.1016/j.bmc.2005.06.004, PII S0968089605005092
    • T Wang IL Chen PJ Lu CH Wong CH Liao KC Tsiao KM Chang YL Chen CC Tzeng 2005 Synthesis, and cytotoxic and antiplatelet activities of oxime- and methyloxime-containing flavone, isoflavone, and xanthone derivatives Bioorg Med Chem 13 6045 6053 10.1016/j.bmc.2005.06.004 15990314 10.1016/j.bmc.2005.06.004 (Pubitemid 41399915)
    • (2005) Bioorganic and Medicinal Chemistry , vol.13 , Issue.21 , pp. 6045-6053
    • Wang, T.-C.1    Chen, I.-L.2    Lu, P.-J.3    Wong, C.-H.4    Liao, C.-H.5    Tsiao, K.-C.6    Chang, K.-M.7    Chen, Y.-L.8    Tzeng, C.-C.9


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.