Identification of new agonists of urotensin-II from a cyclic peptide library

Bioorganic and Medicinal Chemistry

Volumn 17, Issue 18, 2009, Pages 6742-6747

  Odagami, Takenao ^a   Tsuda, Yuko ^b   Kogami, Yuji ^a   Kouji, Hiroyuki ^a   Okada, Yoshio ^b  

^a PRISM Bio Lab Corporation 4259 3   (Japan)

^b KOBE GAKUIN UNIVERSITY   (Japan)

Author keywords

Agonist for urotensin II receptor; Cyclic hexapeptide library; GPR 14; Lactam bridge

Indexed keywords

CYCLOPEPTIDE; PEPTIDE LIBRARY; UNCLASSIFIED DRUG; UROTENSIN II; UROTENSIN II RECEPTOR STIMULATING AGENT;

AGONIST; AMINO ACID SEQUENCE; ARTICLE; CALCIUM MOBILIZATION; CONCENTRATION RESPONSE; DRUG DESIGN; DRUG RECEPTOR BINDING; MONTE CARLO METHOD; PROTEIN CONFORMATION; PROTEIN SECONDARY STRUCTURE;

AMINO ACID SEQUENCE; CELL LINE; HUMANS; MODELS, MOLECULAR; MOLECULAR CONFORMATION; PEPTIDE LIBRARY; PEPTIDES, CYCLIC; RECEPTORS, G-PROTEIN-COUPLED; UROTENSINS;

EID: 69249131356     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2009.07.058     Document Type: Article

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