Synthesis and antiviral activity of new pyrazole and thiazole derivatives

European Journal of Medicinal Chemistry

Volumn 44, Issue 9, 2009, Pages 3746-3753

  El Sabbagh, Osama I ^a   Baraka, Mohamed M ^a   Ibrahim, Samy M ^a   Pannecouque, Christophe ^b   Andrei, Graciela ^b   Snoeck, Robert ^b   Balzarini, Jan ^b   Rashad, Adel A ^a  

^a Zagazig University   (Egypt)

^b REGA INSTITUTE FOR MEDICAL RESEARCH   (Belgium)

Author keywords

Antiviral activity; Poxviruses; Pyrazole; Synthesis; Thiazole

Indexed keywords

1 ACETYL 5 [4 (BENZYLOXY)PHENYL] 3 (4 CHLOROPHENYL) 4,5 DIHYDRO (1H) PYRAZOLE; 5 (2 BROMOVINYL) 2' DEOXYURIDINE; ANTIVIRUS AGENT; CIDOFOVIR; DS 5000; GANCICLOVIR; NEVIRAPINE; PYRAZOLE DERIVATIVE; RIBAVIRIN; THIAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; ANTIVIRAL ACTIVITY; ARTICLE; CONCENTRATION RESPONSE; CONTROLLED STUDY; CYCLIZATION; DRUG CYTOTOXICITY; DRUG SYNTHESIS; HUMAN; HUMAN CELL; NONHUMAN; POXVIRUS; REACTION ANALYSIS; STRUCTURE ACTIVITY RELATION; VACCINIA VIRUS;

ANIMALS; ANTIVIRAL AGENTS; CERCOPITHECUS AETHIOPS; HELA CELLS; HUMANS; MICROBIAL SENSITIVITY TESTS; PYRAZOLES; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLES; VERO CELLS; VIRUSES;

EID: 67650383465     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2009.03.038     Document Type: Article

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