First mariner Mos1 transposase inhibitors

Mini-Reviews in Medicinal Chemistry

Volumn 9, Issue 4, 2009, Pages 431-439

  Bouchet, N ^a,b   Bischerour, J ^a,b   Germon, S ^a   Guillard, J ^a,b   Dubernet, M ^a,b   Viaud Massuard, M C ^a,b   Delelis, O ^d   Ryabinin, V ^e   Bigot, Y ^a,b,c   Auge Gouillou C ^a,b  

^a CNRS UMR6239   (France)

^b UNIVERSITÉ DE TOURS   (France)

^c UNIVERSITY HOSPITAL OF TOURS   (France)

^d Ecole Normale Superieure de Cachan   (France)

^e INSTITUTE OF CHEMICAL BIOLOGY AND FUNDAMENTAL MEDICINE   (Russian Federation)

Author keywords

Heterocyclic chemistry; HIV 1 integrase inhibitor; Maleimides; Mariner inhibitor; Transposon inhibitor

Indexed keywords

BENZOIC ACID DERIVATIVE; CARBOXYLIC ACID DERIVATIVE; CINNAMIC ACID DERIVATIVE; COUMARIN DERIVATIVE; DNA; INTEGRASE; INTEGRASE INHIBITOR; MALEIMIDE DERIVATIVE; NUCLEOTIDYLTRANSFERASE INHIBITOR; PYRROLE DERIVATIVE; THIAZOLIDINE DERIVATIVE; TRANSPOSASE; TRANSPOSASE INHIBITOR; UNCLASSIFIED DRUG; DNA BINDING PROTEIN; MARINER TRANSPOSASES; P31 INTEGRASE PROTEIN, HUMAN IMMUNODEFICIENCY VIRUS 1;

ARTICLE; DNA STRAND; DNA TRANSPOSITION; DRUG MECHANISM; DRUG RESEARCH; DRUG STRUCTURE; ENZYME INHIBITION; GEL MOBILITY SHIFT ASSAY; HUMAN IMMUNODEFICIENCY VIRUS 1; IN VITRO STUDY; INHIBITION KINETICS; PROKARYOTE; TRANSPORT KINETICS; CHEMISTRY; CROSS REACTION; DRUG ANTAGONISM; DRUG DEVELOPMENT; DRUG EFFECT; REVIEW;

CROSS REACTIONS; DNA-BINDING PROTEINS; DRUG DISCOVERY; HIV INTEGRASE; MALEIMIDES; TRANSPOSASES;

EID: 67549145642     PISSN: 13895575     EISSN: None     Source Type: Journal    
DOI: 10.2174/138955709787847912     Document Type: Article

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