Structure of the catalytic domain of avian sarcoma virus integrase with a bound HIV-1 integrase-targeted inhibitor

Proceedings of the National Academy of Sciences of the United States of America

Volumn 95, Issue 9, 1998, Pages 4831-4836

  Lubkowski, Jacek ^a   Yang, Fan ^a   Alexandratos, Jerry ^a   Wlodawer, Alexander ^a   Zhao, He ^b   Burke Jr , Terrence R ^b   Neamati, Nouri ^b   Pommier, Yves ^b   Merkel, George ^c   Skalka, Anna Marie ^c  

^a NATIONAL CANCER INSTITUTE   (United States)

^b NATIONAL CANCER INSTITUTE   (United States)

^c FOX CHASE CANCER CENTER   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

DIVALENT CATION; INTEGRASE; INTEGRASE INHIBITOR; MANGANESE;

AMINO ACID SEQUENCE; ARTICLE; AVIAN SARCOMA VIRUS; CRYSTAL STRUCTURE; ENZYME ACTIVE SITE; ENZYME ACTIVITY; ENZYME CONFORMATION; ENZYME INHIBITOR INTERACTION; ENZYME STRUCTURE; HUMAN IMMUNODEFICIENCY VIRUS 1; NONHUMAN; PRIORITY JOURNAL; PROTEIN DOMAIN; X RAY CRYSTALLOGRAPHY;

AVIAN SARCOMA VIRUSES; BINDING SITES; CRYSTALLOGRAPHY, X-RAY; HIV INTEGRASE INHIBITORS; HYDROGEN-ION CONCENTRATION; INTEGRASES; MANGANESE; MODELS, MOLECULAR; MOLECULAR SEQUENCE DATA; NAPHTHALENESULFONATES; PROTEIN STRUCTURE, TERTIARY;

AVES; AVIAN SARCOMA VIRUS; HUMAN IMMUNODEFICIENCY VIRUS; HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 0342569810     PISSN: 00278424     EISSN: None     Source Type: Journal    
DOI: 10.1073/pnas.95.9.4831     Document Type: Article

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