Fluphenazine release from biodegradable microparticles: Characterization and modelling of release

Journal of Microencapsulation

Volumn 26, Issue 5, 2009, Pages 403-410

  Dunne, Margaret M ^a   Ramtoola, Zebunnissa ^b   Corrigan, Owen I ^a  

^a TRINITY COLLEGE DUBLIN   (Ireland)

^b ROYAL COLLEGE OF SURGEONS IN IRELAND   (Ireland)

Author keywords

Burst effect; Fluphenazine; Modelling release; PLGA

Indexed keywords

FLUPHENAZINE; MICROSPHERE; POLYGLACTIN; POLYMER;

ARTICLE; BIODEGRADATION; CATALYSIS; CONTROLLED DRUG RELEASE; DRUG DIFFUSION; DRUG RELEASE; ENCAPSULATION;

BIOCOMPATIBLE MATERIALS; BIODEGRADATION, ENVIRONMENTAL; DELAYED-ACTION PREPARATIONS; DIFFUSION; FLUPHENAZINE; LACTIC ACID; MICROSPHERES; MODELS, CHEMICAL; POLYGLYCOLIC ACID; TIME FACTORS;

EID: 66049162375     PISSN: 02652048     EISSN: 14645246     Source Type: Journal    
DOI: 10.1080/02652040802396575     Document Type: Article

References (28)

1. Batycky RP, Hanes J, Langer R, Edwards DA. 1997. A theoretical model of erosion and macromolecular drug release from biodegrading microspheres. J Pharm Sci 86:1464-1477. (Pubitemid 28018331)
2. Beck LR, Cowsar DR, Lewis DH, Cosgrove RJ, Riddle CT, Lowry SL, et al. 1979. A new long-acting injectable microcapsule system for the administration of progesterone. Fertility Sterility 31:545-551.
3. Benita S, Benoit JP, Puisieux F, Thies C. 1984. Characterisation of drug loaded poly(D,L-lactide) microspheres. J Pharm Sci 73:1721-1724.
4. Carstensen JT. 2000. Solid state stability. In: Carstensen JT, Rhodes CT, editors. Drug stability principles and practices. Drugs and the pharmaceutical sciences. 3rd ed. Vol.107, Basel, NY: Marcel Dekker Inc. pp 145-189.
5. Cha Y, Pitt CG. 1988. A one-week subdermal delivery system for L-methadone based on biodegradable microcapsules. J Contr Rel 7:69-78.
6. Conti B, Pavanetto F, Genta I. 1992. Use of polylactic acid for the preparation of microparticulate drug delivery systems. J Microencapsulation 9:153-166.
7. Corrigan OI, Heelan BA. 2001. Characterization of drug release from diltiazem-loaded polylactide microspheres prepared using sodium caseinate and whey protein as emulsifying agents. J Microencapsulation 18:335-345.
8. Dunne M, Corrigan OI, Ramtoola Z. 2000. Influence of particle size and dissolution conditions on the degradation properties of polylactide-coglycolide particles. Biomaterials 21:1659-1668.
9. Faisant N, Siepmann J, Benoit JP. 2002. PLGA-based microparticles: Elucidation of mechanisms and a new, simple mathematical model quantifying drug release. Eur J Pharm Sci 15:355-366. (Pubitemid 34436923)
10. Fitzgerald JF, Corrigan OI. 1993. Mechanisms governing drug release from poly-hydroxy aliphatic esters. Diltiazem base release from poly (lactide-co-glycolide) delivery systems. In: El-Nokaly MA, Piatt DM, Charpentier BA, editors. Polymeric delivery systems, properties and applications, ACS Symposium series 520. Washington, DC: American Chemical Society. pp 311-326.
11. Fitzgerald JF, Corrigan OI. 1996. Investigation of the mechanisms governing the release of levamisole from poly-lactide-co-glycolide delivery systems. J Contr Rel 42:125-132.
12. Gallagher KM, Corrigan OI. 2000. Mechanistic aspects of the release of levamisole hydrochloride from biodegradable polymers. J Contr Rel 69:261-272.
13. Guiziou B, Armstrong DJ, Elliot PNC, Ford JL, Rostron C. 1996. Investigation of in-vitro release characteristics of NSAID-loaded polylactic acid microspheres. J Microencapsulation 13:701-708.
14. Jalil R, Nixon RJ. 1990. Effect of temperature of dissolution on the release kinetics of phenobarbitone from poly (D,L-lactic acid) microcapsules: Calculation of activation energy. Drug Dev Ind Pharm 16:2257-2266.
15. Leelarasamee N, Howard SA, Malanga CJ, Luzzi LA, Hogan TF, Kandzari SJ, et al. 1986. Kinetics of drug release from polylactic acid-- hydrocortisone microcapsules. J Microencapsulation 3:171-179.
16. Maulding H, Tice DR, Cowsar DR, Fong JW, Pearson JE, Nazareno JP. 1986. Biodegradation of microcapsules: Acceleration of polymer excipient hydrolytic rate by incorporation of a basic medicament. J Contr Rel 3:103-117.
17. Mollo AR, Corrigan OI. 2002. An investigation of the mechanism of release of the amphoteric drug amoxycillin from poly(DL-lactide-co-glycolide) matrices. Pharm Dev Technol 7:333-343.
18. Mollo AR, Corrigan OI. 2003. Effect of poly hydroxy aliphatic ester polymer type on amoxycillin release from cylindrical compacts. Int J Pharm 268(1-2):71-79.
19. Pradhan RS, Vasavada RC. 1994. Formulation and in vitro release study on poly (D,L-lactide) microspheres containing hydrophilic compounds: Glycine homopeptides. J Contr Rel 30:143-154.
20. Prout EG, Tompkins FC. 1944. The thermal decomposition of potassium permanganate. Trans Faraday Soc 40:488-498.
21. Ramtoola Z, Corrigan OI, Barrett C. 1992. Release kinetics of fluphenazine from biodegradable microspheres. J Microencapsulation 9:415-423.
22. Sanders LM, Kent JS, Mc Rae GI, Vickery BH, Tice TR, Lewis DH. 1984. Controlled release of a luteinizing hormone-releasing hormone analogue from poly(D,L-lactide-co-glycolide) microspheres. J Pharm Sci 73:1294-1297.
23. Shah SS, Cha Y, Pitt CG. 1992. Poly(glycolic acid-co-D,L-lactic acid): Diffusion or degradation controlled drug delivery. J Contr Rel 18: 261-270.
24. Siepmann J, Faisant N, Akiki J, Richard J, Benoit JP. 2004. Effect of the size of biodegradable microparticles on drug release: Experiment and theory. J Contr Rel 96:123-134.
25. Siepmann J, Göpferich A. 2001. Mathematical modelling of bioerodible, polymeric drug delivery systems. Adv Drug Del Rev 48: 229-247.
26. Spenlehauer G, Vert M, Benoit JP, Chabot F, Veillard M. 1988. Biodegradable cisplatin microspheres prepared by the solvent evaporation method: Morphology and release characteristics. J Contr Rel 7:217-229.
27. Vert M, Li S, Garreau H. 1991. More about the degradation of LA/GA-derived matrices in aqueous media. J Contr Rel 16:15-26.
28. Wakiyama N, Juni K, Nakano M. 1981. Preparation and evaluation in vitro of polylactic acid microspheres containing local anaesthetics. Chem Pharm Bull 29:3363-3368.