Synthesis and evaluation of novel neamine derivatives effectively targeting to RNA

Bioorganic and Medicinal Chemistry Letters

Volumn 19, Issue 8, 2009, Pages 2103-2106

  Xu, Yanli ^a   Jin, Hongwei ^a   Yang, Zhenjun ^a   Zhang, Liangren ^a   Wang, Qi ^a   Li, Manning ^a   Zhang, Lihe ^a  

^a PEKING UNIVERSITY HEALTH SCIENCE CENTER   (China)

Author keywords

16S RNA; Molecular modeling; Neamine derivative; TAR RNA

Indexed keywords

NEAMINE; NEAMINE DERIVATIVE; RNA; RNA 16S; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ARTICLE; BINDING AFFINITY; DRUG ACTIVITY; DRUG BINDING; DRUG SYNTHESIS; DRUG TARGETING; NONHUMAN; RNA BINDING;

ANTI-HIV AGENTS; BASE SEQUENCE; BINDING SITES; DRUG DELIVERY SYSTEMS; DRUG EVALUATION, PRECLINICAL; FRAMYCETIN; MICROBIAL SENSITIVITY TESTS; MODELS, MOLECULAR; MOLECULAR SEQUENCE DATA; RNA, VIRAL;

EID: 63149178647     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2009.03.021     Document Type: Article

References (34)

1. Sucheck S.J., and Wong C.H. Curr. Opin. Chem. Biol. 4 (2000) 678
2. Ecker D.J., and Griffey R.H. Drug Discovery Today 4 (1999) 420
3. Ramakrishna V., and Moore P.B. Curr. Opin. Struct. Biol. 11 (2001) 144
4. Fourmy D.I., Recht M., and Puglisi J.D. J. Mol. Biol. 277 (1998) 347
5. Mei H.Y., Cui M., Heldsinger A., Heldsinger A., Lemrow S.M., Loo J.A., Sannes-Lowery K.A., Sharmeen L., and Czarnik A.W. Biochemistry 37 (1998) 14204
6. Gait M.J., and Karn J. Trends Biochem. Sci. 18 (1993) 255
7. Mei H.Y., Galan A.A., Halim N.S., Mack D.P., Moreland D.W., Sanders K.B., Truong H.N., and Czarnikt A.W. Bioorg. Med. Chem. Lett. 5 (1995) 2755
8. Koeda T., Umemura K., and Yokoda M. In: Umezawa H., and Hooper I.R. (Eds). Aminoglycoside Antibiotics Vol. 62 (1982), Springer, Berlin, New York 293
9. Tanaka N. Arch. Pharm. Res. 6 (1983) 93
10. Greenberg W.A., Priestley E.S., Sears P.S., Alper P.B., Rosenbohm C., Hendrix M., Hung S.C., and Wong C.H. J. Am. Chem. Soc. 121 (1999) 6527
11. Silva G.S., and Carvalho I. Curr. Med. Chem. 14 (2007) 1101
12. Zhou J., Wang G.N., Zhang L.H., and Ye X.S. Med. Res. Rev. 27 (2007) 279
13. Calnan B.J., Tidor B., Biancalana S., Hudson D., and Frankel A.D. Science 252 (1991) 1167
14. Weeks K.M., Ampe C., Schultz S.C., Steitz T.A., and Crothers D.M. Science 249 (1990) 1281
15. Litovchick A., Evdokimov A.G., and Lapidot A. Biochemistry 39 (2000) 2838
16. Lapidot A., Vijayabaskar V., Litovchick A., Yu J.G., and James T.L. FEBS Lett. 577 (2004) 415
17. Kawamoto S.A., Sudhahar C.G., Hatfield C.L., Sun J., Behrman E.J., and Gopalan V. Nucleic Acids Res. 36 (2008) 697
18. Lapidot A., Peled A., Berchanski A., Pal B., Kollet O., Lapidot T., and Borkow G. Biochim. Biophys. Acta (BBA) 1780 (2008) 914
19. Borkow G., Lara H.H., and Lapidot A. Biochem. Biophys. Res. Commun. 312 (2003) 1047
20. Borkow G., Vijayabaskar V., Lara H.H., Kalinkovich A., and Lapidot A. Antiviral Res. 60 (2003) 181
21. Eubank T.D., Biswas R., Jovanovic M., Litovchick A., Lapidot A., and Gopalan V. FEBS Lett. 511 (2002) 107
22. Hamasaki K., and Ueno A. Bioorg. Med. Chem. Lett. 11 (2001) 591
23. Cabrera C., Gutierrez A., Barretina J., Blanco J., Litovchick A., Lapidot A., Clotet B., and Este J.A. Antiviral Res. 53 (2002) 1
24. Litovchick A., Evdokimov A.G., and Lapidot A. FEBS Lett. 445 (1999) 73
25. Lapidot A., Vijayabaskar V., Litovchick A., Yu J.H., and James T.L. FEBS Lett. 577 (2004) 415
26. Hegde R., Borkow G., Berchanski A., and Lapidot A. FEBS J. 274 (2007) 6523
27. Watanable K., Katou T., Lkezawa Y., Yajima S., Shionnoya H., Akagi T., and Hamasaki K. Nucleic Acids Symp. Ser. 51 (2007) 209
28. Yajima S., Shionoya H., Akagi T., and Hamasaki K. Bioorg. Med. Chem. 14 (2006) 2799
29. Wu B.G., Yang J., He Y., and Swayze E.E. Org. Lett. 4 (2002) 3455
30. Cai L., Li Q., Ren B., Yang Z.J., Zhang L.R., and Zhang L.H. Tetrahedron 63 (2007) 8135
31. Davis T.M., and Wilson W.D. Methods Enzymol. 340 (2001) 22
32. Hendrix M., Priestley Z.S., Joyce G.F., and Wong C.H. J. Am.Chem. Soc. 119 (1997) 3641
33. Morris G.M., Goodsell D.S., Halliday R.S., Hucy R., Hart W.E., Belew R.K., and Olson A.J. J. Comput. Chem. 19 (1998) 1639
34. Jorgensen J.H., Turnidge J.D., and Washington J.A. In: Murray P.R., Baron E.J.M., Pfaller A., Tenover F.C., and Yolken R.H. (Eds). Manual of Clinical Microbiology. 7th Ed. (1999), ASM, Washington, D.C. 1526