SCOPUS 정보 검색 플랫폼

Volumn , Issue 3, 2009, Pages 437-440

Simple synthesis of 3-acetamido-β-resorcylic acids as potential FabF and FabH inhibitors without using protecting groups

(4) Maraš, Nenad a Anderluh, Petra Štefanič b Urleb, Uroš b Kočevar, Marijan a

a UNIVERSITY OF LJUBLJANA (Slovenia)

b Lek dd (Slovenia)

Author keywords

Acylations; Antibiotics; Carboxylic acids; Drugs; Phenols

Indexed keywords

EID: 62349123503 PISSN: 09365214 EISSN: 14372096 Source Type: Journal
DOI: 10.1055/s-0028-1087544 Document Type: Article

Times cited : (9)

References (29)

1
- 33744994317
- Wang, J.; Soisson, S. M.; Young, K.; Shoop, W.; Kodali, S.; Galgoci, A.; Painter, R.; Parthasarathy, G.; Tang, Y. S.; Cummings, R.; Ha, S.; Dorso, K.; Motyl, M.; Jayasuriya, H.; Ondeyka, J.; Herath, K.; Zhang, C.; Hernandez, L.; Allocco, J.; Basilio, ; Tormo, J. R.; Genilloud, O.; Vicente, F.; Pelaez, F.; Colwell, L.; Lee, S. H.; Michael, B.; Felcetto, T.; Gill, C.; Silver, L. L.; Hermes, J. D.; Bartizal, K.; Barrett, J.; Schmatz, D.; Becker, J. W.; Cully, D.; Singh, S. B. Nature (London) 2006, 441, 358.
- (a) Wang, J.; Soisson, S. M.; Young, K.; Shoop, W.; Kodali, S.; Galgoci, A.; Painter, R.; Parthasarathy, G.; Tang, Y. S.; Cummings, R.; Ha, S.; Dorso, K.; Motyl, M.; Jayasuriya, H.; Ondeyka, J.; Herath, K.; Zhang, C.; Hernandez, L.; Allocco, J.; Basilio, ; Tormo, J. R.; Genilloud, O.; Vicente, F.; Pelaez, F.; Colwell, L.; Lee, S. H.; Michael, B.; Felcetto, T.; Gill, C.; Silver, L. L.; Hermes, J. D.; Bartizal, K.; Barrett, J.; Schmatz, D.; Becker, J. W.; Cully, D.; Singh, S. B. Nature (London) 2006, 441, 358.

2
- 33748482185
- (b) Singh, S. B.; Jayasuriya, H.; Ondeyka, J. G.; Herath, K. B.; Zhang, C.; Zink, D. L.; Tsou, N. N.; Ball, R. G.; Basilio, A.; Genilloud, O.; Diez, M. T.; Vicente, F.; Pelaez, F.; Young, K.; Wang, J. J. Am. Chem. Soc. 2006, 128, 11916.
- (2006) J. Am. Chem. Soc , vol.128 , pp. 11916
- Singh, S.B.¹ Jayasuriya, H.² Ondeyka, J.G.³ Herath, K.B.⁴ Zhang, C.⁵ Zink, D.L.⁶ Tsou, N.N.⁷ Ball, R.G.⁸ Basilio, A.⁹ Genilloud, O.¹⁰ Diez, M.T.¹¹ Vicente, F.¹² Pelaez, F.¹³ Young, K.¹⁴ Wang, J.¹⁵

3
- 62349137282
- Int. Patent, WO2005009391, 196607
- (c) Basilio, A.; Genilloud, O.; Hernandez, P.; Singh, S. B.; Tormo, J. R.; Wang, J. Int. Patent, WO2005009391, 2005; Chem. Abstr. 2005, 142, 196607.
- (2005) Chem. Abstr , vol.142
- Basilio, A.¹ Genilloud, O.² Hernandez, P.³ Singh, S.B.⁴ Tormo, J.R.⁵ Wang, J.⁶

4
- 33750629319
- (a) Nicolaou, K. C.; Li, A.; Edmonds, D. J. Angew. Chem. Int. Ed. 2006, 45, 7086.
- (2006) Angew. Chem. Int. Ed , vol.45 , pp. 7086
- Nicolaou, K.C.¹ Li, A.² Edmonds, D.J.³

5
- 34248329634
- (b) Zou, Y.; Chen, C.-H.; Taylor, C. D.; Foxman, B. M.; Snider, B. B. Org. Lett. 2007, 9, 1825.
- (2007) Org. Lett , vol.9 , pp. 1825
- Zou, Y.¹ Chen, C.-H.² Taylor, C.D.³ Foxman, B.M.⁴ Snider, B.B.⁵

6
- 34250812701
- (c) Nicolaou, K. C.; Tang, Y.; Wang, J. Chem. Commun. 2007, 1922.
- (2007) Chem. Commun , pp. 1922
- Nicolaou, K.C.¹ Tang, Y.² Wang, J.³

7
- 34250702223
- (d) Nicolaou, K. C.; Edmonds, D. J.; Li, A.; Scott Tria, G. Angew. Chem. Int. Ed. 2007, 46, 3942.
- (2007) Angew. Chem. Int. Ed , vol.46 , pp. 3942
- Nicolaou, K.C.¹ Edmonds, D.J.² Li, A.³ Scott Tria, G.⁴

8
- 55949084611
- (e) Matsuo, J.; Takeuchi, K.; Ishibashi, H. Org. Lett. 2008, 10, 4049.
- (2008) Org. Lett , vol.10 , pp. 4049
- Matsuo, J.¹ Takeuchi, K.² Ishibashi, H.³

9
- 36348961991
- (f) Lalic, G.; Corey, E. J. Org. Lett. 2007, 9, 4921.
- (2007) Org. Lett , vol.9 , pp. 4921
- Lalic, G.¹ Corey, E.J.²

10
- 35649019236
- (g) Tiefenbacher, K.; Mulzer, J. Angew. Chem. Int. Ed. 2007, 46, 8074.
- (2007) Angew. Chem. Int. Ed , vol.46 , pp. 8074
- Tiefenbacher, K.¹ Mulzer, J.²

11
- 35048904473
- (h) Ghosh, A. K.; Xi, K. Org. Lett. 2007, 9, 4013.
- (2007) Org. Lett , vol.9 , pp. 4013
- Ghosh, A.K.¹ Xi, K.²

12
- 34547811676
- (i) Li, P.; Payette, J. N.; Yamamoto, H. J. Am. Chem. Soc. 2007, 129, 9534.
- (2007) J. Am. Chem. Soc , vol.129 , pp. 9534
- Li, P.¹ Payette, J.N.² Yamamoto, H.³

13
- 41949129210
- Tiefenbacher, K.; Mulzer, J. Angew. Chem. Int. Ed. 2008, 47, 2548.
- (2008) Angew. Chem. Int. Ed , vol.47 , pp. 2548
- Tiefenbacher, K.¹ Mulzer, J.²

14
- 34347219762
- (a) Jayasuriya, H.; Herath, K. B.; Zhang, C.; Zink, D. L.; Basilio, A.; Genilloud, O.; Diez, M. T.; Vicente, F.; Gonzalez, I.; Salazar, O.; Pelaez, F.; Cummings, R.; Ha, S.; Wang, J.; Singh, S. B. Angew. Chem. Int. Ed. 2007, 46, 4684.
- (2007) Angew. Chem. Int. Ed , vol.46 , pp. 4684
- Jayasuriya, H.¹ Herath, K.B.² Zhang, C.³ Zink, D.L.⁴ Basilio, A.⁵ Genilloud, O.⁶ Diez, M.T.⁷ Vicente, F.⁸ Gonzalez, I.⁹ Salazar, O.¹⁰ Pelaez, F.¹¹ Cummings, R.¹² Ha, S.¹³ Wang, J.¹⁴ Singh, S.B.¹⁵

15
- 62349091400
- Int. Patent, WO2005115400, 5523
- (b) Basilio, A.; Genilloud, O.; Jayasuriya, H.; Gonzalez, I.; Singh, S. B.; Salazar, O.; Wang, J. Int. Patent, WO2005115400, 2005; Chem. Abstr. 2005, 144, 5523.
- (2005) Chem. Abstr , vol.144
- Basilio, A.¹ Genilloud, O.² Jayasuriya, H.³ Gonzalez, I.⁴ Singh, S.B.⁵ Salazar, O.⁶ Wang, J.⁷

16
- 34347267633
- (a) Nicolaou, K. C.; Lister, T.; Denton, R. M.; Montero, A.; Edmonds, D. J. Angew. Chem. Int. Ed. 2007, 46, 4712.
- (2007) Angew. Chem. Int. Ed , vol.46 , pp. 4712
- Nicolaou, K.C.¹ Lister, T.² Denton, R.M.³ Montero, A.⁴ Edmonds, D.J.⁵

17
- 36849044252
- (b) Nicolaou, K. C.; Tang, Y.; Wang, J.; Stepan, A. F.; Li, A.; Montero, A. J. Am. Chem. Soc. 2007, 129, 14850.
- (2007) J. Am. Chem. Soc , vol.129 , pp. 14850
- Nicolaou, K.C.¹ Tang, Y.² Wang, J.³ Stepan, A.F.⁴ Li, A.⁵ Montero, A.⁶

18
- 34347343834
- (c) Singh, S. B.; Herath, K. B.; Wang, J.; Tsou, N.; Ball, R. G. Tetrahedron Lett. 2007, 48, 5429.
- (2007) Tetrahedron Lett , vol.48 , pp. 5429
- Singh, S.B.¹ Herath, K.B.² Wang, J.³ Tsou, N.⁴ Ball, R.G.⁵

19
- 55949136978
- (d) Yeung, Y.-Y.; Corey, E. J. Org. Lett. 2008, 10, 3877.
- (2008) Org. Lett , vol.10 , pp. 3877
- Yeung, Y.-Y.¹ Corey, E.J.²

20
- 33749030702
- Häbich, D.; von Nussbaum, F. ChemMedChem 2006, 1, 951.
- (2006) ChemMedChem , vol.1 , pp. 951
- Häbich, D.¹ von Nussbaum, F.²

21
- 34548672579
- Heretsch, P.; Giannis, A. Synthesis 2007, 2614.
- (2007) Synthesis , pp. 2614
- Heretsch, P.¹ Giannis, A.²

22
- 41049117431
- Nicolaou, K. C.; Tria, G. S.; Edmonds, D. J. Angew. Chem. Int. Ed. 2008, 47, 1780.
- (2008) Angew. Chem. Int. Ed , vol.47 , pp. 1780
- Nicolaou, K.C.¹ Tria, G.S.² Edmonds, D.J.³

23
- 46749145371
- Hayashida, J.; Rawal, V. H. Angew. Chem. Int. Ed. 2008, 47, 4373.
- (2008) Angew. Chem. Int. Ed , vol.47 , pp. 4373
- Hayashida, J.¹ Rawal, V.H.²

24
- 33947461091
- Lindsey, A. S.; Jeskey, H. Chem. Rev. 1957, 57, 583.
- (1957) Chem. Rev , vol.57 , pp. 583
- Lindsey, A.S.¹ Jeskey, H.²

25
- 0009288042
- Reimer, K.; Tiemann, F. Ber. Dtsch. Chem. Ges. 1876, 9, 1285.
- (1876) Ber. Dtsch. Chem. Ges , vol.9 , pp. 1285
- Reimer, K.¹ Tiemann, F.²

26
- 37049095531
- Sasson, Y.; Razintsky, M. J. Chem. Soc., Chem. Commun. 1985, 1134.
- (1985) J. Chem. Soc., Chem. Commun , pp. 1134
- Sasson, Y.¹ Razintsky, M.²

27
- 33750403113
- Wiley: New York
- Nierenstein, M.; Clibbens, D. A. Org. Synth., Coll. Vol. II; Wiley: New York, 1943, 557.
- (1943) Org. Synth., Coll , vol.2 , pp. 557
- Nierenstein, M.¹ Clibbens, D.A.²

28
- 0001610492
- Meek, W. H.; Fuchsman, C. H. J. Chem. Eng. Data 1969, 14, 388.
- (1969) J. Chem. Eng. Data , vol.14 , pp. 388
- Meek, W.H.¹ Fuchsman, C.H.²

29
- 62349121513
- General Procedure for the Preparation of N-Acyl-2,6- dihydroxyanilines 5a-e Using Acid Chlorides: To a solution of 2-aminoresorcinol (4; 7 mmol) in EtOAc (30 mL) stirred in an ice bath was added pyridine (0.76 mL, 10 mmol) followed a dropwise introduction of a solution of an acid chloride (6 mmol) in EtOAc (30 mL, After 1 h the reaction mixture was washed with H2O (30 mL, aq NaHCO3 (5, 30 mL, aq HCl (1 M, 30 mL, H2O (30 mL, then dried over Na 2SO4 and evaporated in vacuo yielding 5. General Procedure for the Preparation of N-Acyl-2,6-dihydroxyanilines 5f-j Using Acids and CDI: To a solution of a carboxylic acid (1.16 g, 6 mmol) in THF (10 mL) was added carbonyldiimidazole (1.00 g, 6 mmol, After stirring for 1 h at r.t, it was added to a solution of 2-aminoresorcinol (4, 7 mmol) in EtOAc 30 mL, The mixture was left stirring for 24 h at r.t, washed with diluted h
- 2), 6.43 (d, J = 8.8 Hz, 1 H, ArH), 7.56 (d, J = 8.8 Hz, 1 H, ArH), 8.91 (s, 1 H, NH), 10.23 (s, 1 H, OH)

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