Effects of the H3 receptor inverse agonist thioperamide on cocaine-induced locomotion in mice: Role of the histaminergic system and potential pharmacokinetic interactions

Psychopharmacology

Volumn 202, Issue 4, 2009, Pages 673-687

  Brabant, Christian ^a,d   Alleva, Livia ^a   Grisar, Thierry ^a   Quertemont, Etienne ^a   Lakaye, Bernard ^a   Ohtsu, Hiroshi ^b   Lin, Jian Sheng ^c   Jatlow, Peter ^d   Picciotto, Marina R ^d   Tirelli, Ezio ^a  

^a UNIVERSITY OF LIÈGE   (Belgium)

^b TOHOKU UNIVERSITY   (Japan)

^c UNIVERSITÉ LYON 1   (France)

^d YALE UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

A 331440; Cocaine; H3 receptor; Histamine; Immepip; Knockout mouse; Locomotion; Thioperamide

Indexed keywords

A 331440; COCAINE; HISTAMINE; HISTAMINE H3 RECEPTOR; HISTAMINE H3 RECEPTOR AGONIST; IMMEPIP; THIOPERAMIDE; UNCLASSIFIED DRUG; 4 (1H IMIDAZOL 4 YLMETHYL)PIPERIDINE; 4' (3 (3(R) (DIMETHYLAMINO) PYRROLIDIN 1 YL) PROPOXY) BIPHENYL 4 CARBONITRILE; 4'-(3-(3(R)-(DIMETHYLAMINO)-PYRROLIDIN-1-YL)-PROPOXY)-BIPHENYL-4-CARBONITRILE; 4-(1H-IMIDAZOL-4-YLMETHYL)PIPERIDINE; BIPHENYL DERIVATIVE; HISTAMINE AGONIST; IMIDAZOLE DERIVATIVE; NITRILE; PIPERIDINE DERIVATIVE; PYRROLIDINE DERIVATIVE;

ANIMAL EXPERIMENT; ARTICLE; CONTROLLED STUDY; DRUG DOSE COMPARISON; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; HISTAMINE RELEASE; HYPERACTIVITY; INVERSE AGONISM; KNOCKOUT MOUSE; LOCOMOTION; MALE; MOUSE; NONHUMAN; PRIORITY JOURNAL; ULTRAVIOLET SPECTROSCOPY; ANIMAL; AREA UNDER THE CURVE; C57BL MOUSE; DOSE RESPONSE; DRUG ANTAGONISM; DRUG EFFECT; DRUG INTERACTION; GENETICS; MOTOR ACTIVITY; MOUSE MUTANT; PHYSIOLOGY;

ANIMALS; AREA UNDER CURVE; BIPHENYL COMPOUNDS; COCAINE; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG INTERACTIONS; HISTAMINE; HISTAMINE AGONISTS; HISTAMINE RELEASE; IMIDAZOLES; MALE; MICE; MICE, INBRED C57BL; MICE, KNOCKOUT; MOTOR ACTIVITY; NITRILES; PIPERIDINES; PYRROLIDINES; RECEPTORS, HISTAMINE H3;

EID: 59849107865     PISSN: 00333158     EISSN: 14322072     Source Type: Journal    
DOI: 10.1007/s00213-008-1345-y     Document Type: Article

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