Dihydroehanoanthracene derivatives reverse in vitro quinoline resistance in Plasmodium falciparum malaria

Medicinal Chemistry

Volumn 4, Issue 5, 2008, Pages 426-437

  Henry, Maud ^a,b   Alibert, Sandrine ^c   Baragatti, Mcili ^a,b   Mosnier, Joel ^a,b   Baret, Eric ^a,b   Amalvict, Rémy ^a,b   Legrand, Eric ^d   Fusai, Thierry ^a,b   Barbe, Jacques ^c   Rogier, Christophe ^a,b   Pagès, Jean Marie ^c   Pradines, Bruno ^a,b  

^a SERVICE DE SANTÉ DES ARMÉES   (France)

^b AIX MARSEILLE UNIVERSITÉ   (France)

^c Aix Marseille University   (France)

^d INSTITUT PASTEUR DE LA GUYANE   (French Guiana)

Author keywords

Antimalarial drug; Chemosesitizer; Malaria; Quinoline resistance; Reversal agent

Indexed keywords

ANTIMALARIAL AGENT; BG 1001; BG 918; BG 920; BG 958; CHLOROQUINE; CHLORPROMAZINE; CYPROHEPTADINE; DEETHYLAMODIAQUINE; KETOTIFEN; MEFLOQUINE; NICARDIPINE; QUININE; RESERPINE; UNCLASSIFIED DRUG; VERAPAMIL; ANTHRACENE DERIVATIVE; QUINOLINE DERIVATIVE;

ARTICLE; CONTROLLED STUDY; DRUG ANTAGONISM; DRUG POTENCY; DRUG POTENTIATION; DRUG RESISTANCE; DRUG SENSITIVITY; IC 50; IN VITRO STUDY; NONHUMAN; PLASMODIUM FALCIPARUM; PRIORITY JOURNAL; QUINOLINE RESISTANCE REVERSAL; ANIMAL; DRUG EFFECT; GROWTH, DEVELOPMENT AND AGING; HUMAN; MALARIA FALCIPARUM; PARASITOLOGY; STRUCTURE ACTIVITY RELATION;

ANIMALS; ANTHRACENES; ANTIMALARIALS; DRUG RESISTANCE; HUMANS; INHIBITORY CONCENTRATION 50; MALARIA, FALCIPARUM; PARASITIC SENSITIVITY TESTS; PLASMODIUM FALCIPARUM; QUINOLINES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 56649099571     PISSN: 15734064     EISSN: None     Source Type: Journal    
DOI: 10.2174/157340608785700234     Document Type: Article

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