Optimization of salting-out taste-masking system for micro-beads containing drugs with high solubility

Chemical and Pharmaceutical Bulletin

Volumn 56, Issue 11, 2008, Pages 1579-1584

  Yoshida, Takayuki ^a   Tasaki, Hiroaki ^a   Maeda, Atsushi ^a   Katsuma, Masataka ^a   Sako, Kazuhiro ^a   Uchida, Takahiro ^b  

^a ASTELLAS PHARMA INC   (Japan)

^b MUKOGAWA WOMEN'S UNIVERSITY   (Japan)

Author keywords

Lag time; Particle size; Release; Salting out taste masking system; Solubility

Indexed keywords

EUDRAGIT; HEXADECANOL; HYDROXYPROPYLMETHYLCELLULOSE; IMIPRAMINE; PARACETAMOL; POLYMER; POVIDONE; SODIUM CARBONATE; SOLVENT; SUCROSE; TALC;

ARTICLE; DRUG BIOAVAILABILITY; DRUG COATING; DRUG FORMULATION; DRUG RELEASE; DRUG SOLUBILITY; PARTICLE SIZE; TABLET;

ACETAMINOPHEN; CARBONATES; CHEMISTRY, PHARMACEUTICAL; DRUG DELIVERY SYSTEMS; IMIPRAMINE; METHYLCELLULOSE; MICROSPHERES; PARTICLE SIZE; PHARMACEUTICAL PREPARATIONS; POVIDONE; SOLUBILITY; SPECTROPHOTOMETRY, ULTRAVIOLET; TABLETS; TASTE;

EID: 55749084003     PISSN: 00092363     EISSN: 13475223     Source Type: Journal    
DOI: 10.1248/cpb.56.1579     Document Type: Article

References (33)

1. Fu Y., Yang S., Jeong S. H., Kimura S., Park K., Crit. Rev. Ther. Drug Carrier Syst., 21, 433-475 (2004).
2. Seager H., J. Pharm. Pharmacol., 50, 375-382 (1998).
3. Mizumoto T., Masuda Y., Yamamoto T., Yonemochi E., Terada K., Int. J. Pharm., 306, 83-90 (2005).
4. Verma R. K., Garg S., Pharm. Tech. On-line, 25, 1-14 (2001).
5. Khankari R. K., Hontz J., Chastain S. J., Katzner L., U. S. Patent 6024981, 15 February 2000.
6. Shimizu T., Nakano Y., Morimoto S., Tabata T., Hamaguchi N., Igari Y., Chem. Pharm. Bull., 51, 942-947 (2003).
7. Morita T., Yakugaku Zasshi, 123, 665-671 (2003).
8. Helm J. F., Dodds W. J., Riedel D. R., Teeter B. C., Hogan W. J., Arndorfer R. C., Gastroenterology, 85, 607-612 (1983).
9. Oguchi K., Saitoh E., Mizuno M., Baba M., Okui M., Suzuki M., Jpn. J. Reh. Med., 37, 375-382 (2000).
10. Pather S. I., Khankari R. K., Moe D. V., "Modified-Release Drug Delivery Technology," ed. by Rathbone M. J., Hadgraft J., Roberts M. S., Marcel Dekker Inc., New York, 2003, pp. 203-216.
11. van Schaick E. A., Lechat P., Remmerie B. M., Ko G., Lasseter K. C., Mannaert E., Clin. Ther., 25, 1687-1699 (2003).
12. Baldi F., Malfertheiner P., Digestion, 67, 1-5 (2003).
13. Yoshida T., Tasaki H., Maeda A., Katsuma M., Sako K., Uchida T., J. Controlled Release, 131, 47-53 (2008).
14. Shimizu T., Sugaya M., Nakano Y., Izutsu D., Mizukami Y., Okochi K., Tabata T., Hamaguchi N., Igari Y., Chem. Pharm. Bull., 51, 1121-1127 (2003).
15. Ishikawa T., Mukai B., Shiraishi S., Utoguchi N., Fujii M., Matsumoto M., Watanabe Y., Chem. Pharm. Bull., 49, 134-139 (2001).
16. Nagai T., Prakongpan S., Chem. Pharm. Bull., 32, 340-343 (1984).
17. Rogers V., Dor Philippe J. M., Fix J. A., Kojima H., Sako K., WO03/041,656, 22 May 2003.
18. Rege P. R., Fegely K. A., Scattergood L. K., Rajabi-Siahboomi A. R., "Proceedings of the Controlled Release Society Annual Meeting," Controlled Release Society, Minneapolis, 2005, p. 509.
19. Borgquist P., Nevsten P., Nilsson B., Wallenberg L. R., Axelsson A., J. Controlled Release, 97, 453-465 (2004).
20. Ragnarsson G., Johansson M. O., Drug Dev. Ind. Pharm., 14, 2285-2297 (1988).
21. Ragnarsson G., Sandberg A., Johansson M. O., Lindstedt B., Sjögren J., Int. J. Pharm., 79, 223-232 (1992).
22. Lindstedt B., Ragnarsson G., Hjärtstam J., Int. J. Pharm., 56, 261-268 (1989).
23. Heng P. W., Hao J., Chan L. W., Chew S. H., Drug Dev. Ind. Pharm., 30, 213-20 (2004).
24. Schultz P., Kleinebudde P., J. Controlled Release, 47, 181-189 (1997).
25. Zhang Y., Zhang Z., Wu F., J. Controlled Release, 89, 47-55 (2003).
26. Taupin C., Dvolaitzky M., Sauterey C., Biochemistry, 14, 4771-4775 (1975).
27. Verma R. K., Mishra B., Garg S., Drug Dev. Ind. Pharm., 26, 695-708 (2000).
28. Li S., Doyle P., Metz S., Royce A. E., Serajuddin A. T. M., J. Pharm. Sci., 94, 2224-2231 (2005).
29. Chena L.-H., Choia Y.-S., Kwonc J., Wangb R.-S., Leec T., Ryud S. H., Park J. W., Tetrahedron, 60, 7293-7299 (2004).
30. Nakano T., Yuasa H., Int. J. Pharm., 215, 3-12 (2001).
31. Nakano T., Yuasa H., Kanaya Y., Pharm. Res., 16, 1616-1620 (1999).
32. Azorlosa J. L., Martinelli A. J., "Water-Soluble Resins," ed. by Davidson R. L., Sitting M., Reinhold Book Corporation, New York, 1962, pp. 131-153.
33. Ritger P. L., Peppas N. A., J. Controlled Release, 5, 23-36 (1987).