Fluorescent ligands for the histamine H 2 receptor: Synthesis and preliminary characterization

Bioorganic and Medicinal Chemistry

Volumn 12, Issue 24, 2004, Pages 6495-6503

  Malan, Sarel F ^a,b   Marle, Andre Van ^b   Menge, Wiro M ^b   Zuliana, Valentina ^b   Hoffman, Marcel ^b   Timmerman, Henk ^b   Leurs, Rob ^b  

^a NORTH WEST UNIVERSITY   (South Africa)

^b VU UNIVERSITY AMSTERDAM   (Netherlands)

Author keywords

Fluorescent histamine H 2 ligands

Indexed keywords

2 (5 METHYL 4 IMIDAZOLYL)METHYLTHIOETHYLAMINE; FLUORESCENT DYE; HISTAMINE H2 RECEPTOR; HISTAMINE H2 RECEPTOR ANTAGONIST; IODINE 125; IODOAMINOPOTENTIDINE; N CYANO N' [OMEGA [3 (1 PIPERIDINYLMETHYL)PHENOXY]ALKYL]GUANIDINE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; CHEMICAL ANALYSIS; CONTROLLED STUDY; FLUORESCENCE; NONHUMAN; RECEPTOR BINDING; SYNTHESIS;

FLUORESCENT DYES; GUANIDINES; HUMANS; IODINE RADIOISOTOPES; LIGANDS; PIPERIDINES; PROTEIN BINDING; RADIOLIGAND ASSAY; RECEPTORS, HISTAMINE H2;

EID: 8844238270     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2004.09.018     Document Type: Article

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