Pentazocine transport by square-wave AC iontophoresis with an adjusted duty cycle

Journal of Medical and Dental Sciences

Volumn 55, Issue 1, 2008, Pages 15-27

  Ogami, Saori ^a   Hayashi, Shizuka ^a   Shibaji, Takao ^a   Umino, Masahiro ^a  

^a TOKYO MEDICAL AND DENTAL UNIVERSITY   (Japan)

Author keywords

Duty cycle; Iontophoresis; Pentazocine; Square wave; Voltage

Indexed keywords

CELLOPHANE; LACTIC ACID; NARCOTIC ANALGESIC AGENT; PENTAZOCINE;

ARTICLE; ARTIFICIAL MEMBRANE; DRUG DELIVERY SYSTEM; ELECTRODE; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; IONTOPHORESIS; METHODOLOGY; REGRESSION ANALYSIS;

ANALGESICS, OPIOID; CELLOPHANE; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; DRUG DELIVERY SYSTEMS; ELECTRODES; IONTOPHORESIS; LACTIC ACID; LEAST-SQUARES ANALYSIS; MEMBRANES, ARTIFICIAL; PENTAZOCINE;

EID: 52449108692     PISSN: 13428810     EISSN: 13428810     Source Type: Journal    
DOI: None     Document Type: Article

References (37)

1. Vedrinne C, Vedrinne JM, Guiraud M,et al. Nitrogen-Sparing effect of epidural administration of local anesthetics in colon surgery, Anesth Analg 1989;69:354-359.
2. Sugai N. Recent developments in pharmacology and clinical use of pentazocine. Masui 1991;40:1037-1041.
3. Berkowitz BA, Asling JH, Shnider SM,et al. Relationship of pentazocine plasma levels to pharmacological activity in man. Clin Pharmacol Ther 1969;10:320-328.
4. Ehrnebo M, Boreus LO, Lonroth U. Bioavailability and first-pass metabolism of oral pentazocine in man. Clin Pharmacol Ther 1977;22:888-892.
5. Chien YW, Siddiqui O, Sun Y,et al. Transdermal iontophoretic delivery of therapeutic peptides/proteins. Ann N Y Acad Sci 1987;507:32-51
6. Kalia YN, Naik A, Garrison J,et al. lontophoretic drug delivery. Adv Drug Deliv Rev 2004;56:619-658.
7. Ashburn MA, Gauthier M, Love G,et al. lontophoretic administration of 2% lidocaine HCI and 1:100,000 epinephrine in humans. Clin J Pain 1997;13:22-26.
8. Rose JB, Galinkin JL, Jantzen EC,et al. A study of lidocaine iontophoresis for pediatric venipuncture. Anesth Analg 2002;94:867-871.
9. Sherwin J, Awad IT, Sadler PJ,et al. Analgesia during radial artery cannulation: comparison of the effects of lidocaine applied by local injection or iontophoresis. Anaesthesia 2003;58:471-479.
10. Reinauer S, Neusser A, Schauf G,et al. Iontophoresis with alternating current and direct current offset (AC/DC iontophoresis): a new approach for the treatment of hyperhidrosis. Br J Dermatol 1993;129:166-169.
11. Viscusi ER, Reynolds L, Tait S,et al. An iontophoretic fentanyl patient-activated analgesic delivery system for postoperative pain: a double-blind, placebo-controlled trial. Anesth Analg 2006;102:188-194.
12. Potts RO, Tamada JA, Tierney MJ. Glucose monitoring by reverse iontophoresis. Diabetes Metab Res Rev 2002;18:49-53.
13. Howard JP, Drake TR, Kellogg DL Jr. Effects of alternating current iontophoresis on drug delivery. Arch Phys Med Rehabil 1995;76:463-466.
14. Umino M, Oda N, Yasuhara Y. Experimental and theoretical studies of the effect of electrode polarization on capacitances of blood and potassium chloride solution. Med Biol Eng Comput 2002;40:533-541.
15. Sudeji K, Kawasaki M, Inada H,et al. Enhanced percutaneous absorption of formoterol fumarate via pulsed iontophoresis. I. Effect of constant current and constant voltage. Yakugaku Zasshi 1989a;109:766-770.
16. Sudeji K, Furusawa K, Inada H,et al. Enhanced percutaneous absorption of formoterol fumarate via pulsed iontophoresis. II. Effect of polarity, pulse frequency and duty. Yakugaku Zasshi 1989b;109:771-777.
17. Pikal MJ, Stah S. Study of the mechanisms of flux enhancement through hairless mouse skin by pulsed DC iontophoresis. Pharm Res 1991;78:365-369.
18. Li SK, Ghanem AH, Peck KD,et al. Pore induction in human epidermal membrane during low to moderate voltage iontophoresis: A study using AC iontophoresis. J Pharm Sci 1999;88:419-427.
19. Meyer PF, Oddsson LIE. Alternating-pulse iontophoresis for targeted cutaneous anesthesia. J Neurol Sci 2003;125:209-214.
20. Yan G., Higuchi Wl, Szabo A,et al. Correlation of transdermal iontophoresis phenylalanine and mannitol transport: test of the internal standard concept under DC iontophoresis and constant resistance AC iontophoresis conditions. J Control Release 2004a;98:127-138.
21. Yan G, Li SK, Peck KD,et al. Quantitative study of electrophoretic and electroosmotic enhancement during alternating current iontophoresis across synthetic membranes. J Pharm Sci 2004b;93:2895-2908.
22. Yan G, Peck KD, Zhu H,et al. Effects of electrophoresis and electroosmosis during alternating current iontophoresis across human epidermal membrane, J Pharm Sci 2005;94:547-558.
23. Naik A, Kalia YN, Guy RH. Transdermal drug delivery: overcoming the skin's barrier function. PSTT 3 2000;318-326.
24. Kinoshita T, Shibaji T, Umino M. Transdermal delivery of lidocaine in vitro by alternating current. J Med Dent Sci 2003;50:71-77.
25. Haga H, Shibaji T, Umino M. Lidocaine transport through living rat skin using alternating current. Med Biol Eng Comput 2005;43:622-629.
26. Izumikawa H. Lidocaine transportation through a cellophane membrane by wide range AC frequencies. J Stom Sci 2005;72:183-189.(in Japanese)
27. Jadoul A, Mesens J, Caers W,et al. Transdermal permeation of alniditan by iontophoresis: In vitro optimization and human pharmacokinetic data. Pharm Res 1996;13:1348-1353.
28. Sun Y, Siddiquie O, Liu JC,et al. Transdermal modulated delivery of polypeptides: Effect of DC pulse waveform on enhancement. In Proceedings of the 13th International Symposium on Controlled Release of Bioactive Materials, Norfolk, Verginia. 1986;175-176.
29. Liu JC, Sun Y, Siddiqui O,et al. Blood glucose control in diabetic rats by transdermal iontophoretic delivery of insulin. Int J Pharm 1988;44:197-204
30. Okabe K, Yamaguchi H, Kawai Y. New iontophoretic transdermal administration of the beta-blocker metoprolol. J Control Release 1986;4:79-85.
31. Ishikawa O, Kato Y, Onishi H,et al. Enhancement of transdermal absorption by switching iontophoresis. Int J Pharm 2002;249:81-88.
32. Sebastiani P Nicoli S, Santi P. Effect of lactic acid and iontophoresis on drug permeation across rabbit ear skin. Int J Pharm 2005;292:119-126.
33. Shibaji T, Yasuhara Y, Oda N,et al. A mechanism of the high frequency AC iontophoresis. J Control Release 2001;73:37-47.
34. Singh P, Maibach HI. Iontophoresis in drug delivery: Basic principles and applications. Crit Rev Ther Drug carrier syst 1994;11:161-213.
35. Pikal MJ. The role of electroosmotic flow in transdermal iontophoresis. Adv Drug Deliv Rev 2001;46:281-305.
36. Santi P, Catellani PL, Massimo G,et al. lontophoretic transport of verapamil and melatonin. I. Cellophane membrane as a barrier. Int J Pharm 1993;92:23-28.
37. Mollee TR, Anissimov YG, Roberts MS. Periodic electric field enhanced transport through membranes. J Membr Sci 2006;278:290-300.