3,4-Disubstituted-1,2,3,4,5,6,7,8-octahydroquinazoline-2-thiones: Synthesis, antimicrobial evaluation and QSAR investigations using Hansch analysis

Archiv der Pharmazie

Volumn 341, Issue 4, 2008, Pages 231-239

  Minu, Maninder ^a   Thangadurai, Ananda ^a   Wakode, Sharad R ^a   Agrawal, Shyam S ^a   Narasimhan, Balasubramanian ^b  

^a DELHI INSTITUTE OF PHARMACEUTICAL SCIENCES AND RESEARCH   (India)

^b GURU JAMBHESHWAR UNIVERSITY OF SCIENCE AND TECHNOLOGY   (India)

Author keywords

Antibacterial; Antifungal; q2; QSAR; Quinazoline 2 thione

Indexed keywords

1,2,3,4,5,6,7,8 OCTAHYDROQUINAZOLINE 2 THIONE DERIVATIVE; 4 (4 CHLOROPHENYL) 3 (4 NITROPHENYLSULFONYL) 1,2,3,4,5,6,7,8 OCTAHYDROQUINAZOLINE 2 THIONE; 4 (4 FLUOROPHENYL) 3 (4 NITROPHENYLSULFONYL) 1,2,3,4,5,6,7,8 OCTAHYDROQUINAZOLINE 2 THIONE; ANTIINFECTIVE AGENT; UNCLASSIFIED DRUG; QUINAZOLINE DERIVATIVE;

ANALYTIC METHOD; ANTIMICROBIAL ACTIVITY; ARTICLE; CANDIDA ALBICANS; DRUG SCREENING; DRUG SYNTHESIS; ESCHERICHIA COLI; HANSCH ANALYSIS; NONHUMAN; PRIORITY JOURNAL; QUANTITATIVE STRUCTURE ACTIVITY RELATION; STAPHYLOCOCCUS AUREUS; CHEMISTRY; DRUG EFFECT; INFRARED SPECTROPHOTOMETRY; MICROBIOLOGICAL EXAMINATION; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; SYNTHESIS;

ANTI-INFECTIVE AGENTS; CANDIDA ALBICANS; ESCHERICHIA COLI; MAGNETIC RESONANCE SPECTROSCOPY; MICROBIAL SENSITIVITY TESTS; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; QUINAZOLINES; SPECTROPHOTOMETRY, INFRARED; STAPHYLOCOCCUS AUREUS;

EID: 48949120102     PISSN: 03656233     EISSN: 15214184     Source Type: Journal    
DOI: 10.1002/ardp.200700153     Document Type: Article

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