Molecular modeling of a PAMAM-CGS21680 dendrimer bound to an A2A adenosine receptor homodimer

Bioorganic and Medicinal Chemistry Letters

Volumn 18, Issue 15, 2008, Pages 4312-4315

  Ivanov, Andrei A ^a   Jacobson, Kenneth A ^a  

^a NATIONAL INSTITUTE OF DIABETES AND DIGESTIVE AND KIDNEY DISEASES   (United States)

Author keywords

Dimerization; Functionalized congener; G protein coupled receptor; Homology modeling; Nucleoside; Polymerbound drug; Purines

Indexed keywords

2 [4 (2 CARBOXYETHYL)PHENETHYLAMINO]ADENOSINE 5' (N ETHYLCARBOXAMIDE); ADENOSINE A2A RECEPTOR; DENDRIMER; LIGAND; POLYAMIDOAMINE;

ARTICLE; BINDING AFFINITY; COVALENT BOND; DIMERIZATION; MOLECULAR MODEL; RECEPTOR BINDING;

ADENOSINE; DENDRIMERS; HUMANS; LIGANDS; MODELS, MOLECULAR; MOLECULAR CONFORMATION; MOLECULAR STRUCTURE; PHENETHYLAMINES; POLYAMINES; RECEPTOR, ADENOSINE A2A; RECEPTORS, G-PROTEIN-COUPLED;

EID: 47749103678     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2008.06.087     Document Type: Article

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