Design, synthesis of novel peptidomimetic derivatives of 4-HPR for rhabdoid tumors

Bioorganic and Medicinal Chemistry Letters

Volumn 18, Issue 14, 2008, Pages 4177-4180

  Das, Bhaskar C ^a   Smith, Melissa E ^a   Kalpana, Ganjam V ^a  

^a ALBERT EINSTEIN COLLEGE OF MEDICINE   (United States)

Author keywords

4 HPR; Cyclin D1; Retinoid; Rhabdoid tumor

Indexed keywords

4 [(3 ETHYL 2,4,4 TRIMETHYLCYCLOHEX 2 ENYLIDENE)METHYL] N (4 HYDROXY 3 IODOPHENYL)BENZAMIDE; CYCLIN D1; FENRETINIDE; FENRETINIDE DERIVATIVE; RETINOID;

ANIMAL CELL; ANTINEOPLASTIC ACTIVITY; ARTICLE; CANCER CELL CULTURE; CANCER INHIBITION; DRUG DESIGN; DRUG SYNTHESIS; IC 50; MOUSE; NONHUMAN; REACTION ANALYSIS; RHABDOID TUMOR; STRUCTURE ACTIVITY RELATION;

ALKENES; CELL CYCLE; CELL LINE, TUMOR; CELL PROLIFERATION; CHEMISTRY, PHARMACEUTICAL; CYCLIN D1; DRUG DESIGN; FENRETINIDE; HUMANS; INHIBITORY CONCENTRATION 50; MODELS, CHEMICAL; MODELS, STATISTICAL; PEPTIDES; RHABDOID TUMOR;

EID: 47149102333     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2008.05.097     Document Type: Article

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