Fluorescent agonists for the torpedo nicotinic acetylcholine receptor

ChemBioChem

Volumn 9, Issue 7, 2008, Pages 1146-1153

  Krieger, Florian ^a   Mourot, Alexandre ^b   Araoz, Romulo ^c   Kotzyba Hibert, Florence ^a   Molgó, Jordi ^c   Bamberg, Ernst ^b   Goeldner, Maurice ^a  

^a UNIVERSITÉ DE STRASBOURG   (France)

^b MAX PLANCK INSTITUTE OF BIOPHYSICS   (Germany)

^c LABORATOIRE DE NEUROBIOLOGIE CELLULAIRE ET MOLÉCULAIRE   (France)

Author keywords

Fluorescent probes; Kinetics; Neurotransmitters; Receptors; Structure activity relationships

Indexed keywords

7 (DIETHYLAMINO)COUMARIN 3 CARBONYLGLYCYLCHOLINE; ACETYLCHOLINE DERIVATIVE; FLUORESCENT AGONIST; FLUORESCENT DYE; N (7 NITROBENZ 2 OXA 1,3 DIAZOL YL)ACETYLCHOLINE DERIVATIVE; NICOTINIC RECEPTOR; TORPEDO NICOTINIC ACETYLCHOLINE RECEPTOR; UNCLASSIFIED DRUG; ACETYLCHOLINE; COUMARIN DERIVATIVE; FISH PROTEIN; NICOTINIC AGENT;

ANIMAL CELL; ARTICLE; BINDING SITE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DISSOCIATION CONSTANT; DRUG RECEPTOR BINDING; DRUG SCREENING; DRUG SYNTHESIS; NONHUMAN; OOCYTE; PHARMACOLOGICAL PARAMETERS; PRIORITY JOURNAL; SPECTRAL SENSITIVITY; STRUCTURE ACTIVITY RELATION; TORPEDO CALIFORNICA; TORPEDO MARMORATA; XENOPUS; ANIMAL; CHEMISTRY; DRUG EFFECT; DRUG POTENTIATION; ENZYME SPECIFICITY; FLUORESCENCE; KINETICS; METABOLISM; RADIOASSAY; SYNTHESIS; TORPEDO;

TORPEDO CALIFORNICA; TORPEDO MARMORATA;

ACETYLCHOLINE; ANIMALS; COUMARINS; FISH PROTEINS; FLUORESCENCE; FLUORESCENT DYES; KINETICS; NICOTINIC AGONISTS; OOCYTES; RADIOLIGAND ASSAY; RECEPTORS, NICOTINIC; SUBSTRATE SPECIFICITY; TORPEDO;

EID: 46649103918     PISSN: 14394227     EISSN: 14397633     Source Type: Journal    
DOI: 10.1002/cbic.200700757     Document Type: Article

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