N-substituted 1-aryl-2-(1H-imidazol-1-yl)-1-ethanamines with broad spectrum in vitro antimycobacterial and antifungal activities

Medicinal Chemistry Research

Volumn 7, Issue 2, 1997, Pages 87-97

  Fioravanti, Rossella ^a   Biava, Mariangela ^a   Porretta, Giulio Cesare ^a   Artico, Marino ^a   Lampis, Giorgio ^b   Deidda, Delia ^b   Pompei, Raffaello ^b  

^a SAPIENZA UNIVERSITY OF ROME   (Italy)

^b UNIVERSITY OF CAGLIARI   (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 0002945939     PISSN: 10542523     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (24)

1. Davidson, P.T.; Le, H.Q. Drugs 1992, 43, 651-673.
2. Grosset, J.H. Bull. Int. Union Tuberc. Lung Dis. 1990, 65, 86-91.
3. Marriot, M.S.; Richardson, K. Recent Trends in the Discovery, Development and Evaluation of Antifungal Agents, R.A. Fromtling, Ed., J.R. Prous Science Publishers, S.A. Barcelona, Spain, 1987.
4. Fromtling, R.A. Drugs of To-Day 1984, 20, 325-349.
5. Godefroi, E.F.; Heeres, J.; van Cutsen, J.; Janssen, P.A.J. J. Med. Chem. 1969, 12, 784-791.
6. Plempel, M.; Regel, E.; Büchel, K.H. Arzneim.-Forsch. 1983, 33, 517-524.
7. Saag, M.S.; Dismukes, W.E. Antimicrob. Agents Chemother. 1988, 52, 1-8.
8. Stütz, A. Angew. Chem. Int. 1987, 26, 320-328.
9. Petranyi, G.; Ryder, N.S.; Stütz, A. Science 1984, 224, 1239-1241.
10. Stütz, A.; Georgopoulus, A.; Granitzer, W.; Petranyi, G.; Berney, O. J. Med. Chem. 1986, 29, 112-125.
11. Fromtling, R. Drugs of To-Day 1992, 25, 501-508.
12. Arika, T.; Yokoo, M.; Hase, T.; Maeda, T.; Amemiya, K.; Yamaguchi, H. Antimicrob. Agents Chemother. 1990, 34, 2250-2253.
13. Wayne, L.G.; Sramek, H.A. Antimicrob. Agents Chemother. 1994, 38, 2054-2058.
14. Ashtekar, D.R.; Costa-Perira, R.; Nagrajan, K.; Vishvanathan, N.; Bhatt, A.D.; Rittel, W. Antimicrob. Agents Chemother. 1993, 57, 183-186.
15. Nardi, D.; Cappelletti, R.; Catto, A.; Leonardi, A.; Tajana, A.; Veronese, M. Arzneim.-Forsch. Drug Res. 1981, 31, 2123-2125.
16. Mixich, Von G., Thiele, K. Arzneim.-Forsh./Drug Res. 1979, 29, 1510-1513.
17. Porretta, G.C.; Fioravanti, R.; Biava, M.; Cirilli, R.; Simonetti, N.; Villa, A.; Bello, U.; Faccendini, P.; Tita, B. Eur. J. Med. Chem. 1993, 28, 749-769.
18. Trupp, L.D. Antibiotics in Laboratory Medicine, Williams & Wilkins, Eds, Baltimore, 1986, pp. 93-143.
19. Fioravanti, R.; Biava, M.; Porretta, G.C.; Landolfi, C.; Simonetti, N.; Villa, A.; Conte, E.; Porta-Puglia A. Eur. J. Med. Chem., 1995, 30, 123-132.
20. David, H. Bacteriology of the Mycobacterioses. DHEW Publication No. (CDC) 768316; CDC, Mycobacteriology Branch: Atlanta, 1976.
21. Hawkins, J.E.; Wallace, R.J.; Brown, B.A. Antibacteria susceptibility tests: Mycobacteria. In: Manual of Clinical Microbiology Balows W.J., Hausler K.L., Hermann K.L., Isemberg H.D. and Shadomy H.J. (Eds), ASM Press Washington, DC, 1991, pp 1138-1152.
22. National Committee for Clinical Laboratory Standards. Antimycobacterial susceptibility testing. 1990, Proposed Standard M24, Villanova, PA.
23. Cynamom, M.H.; Gimi, R.; Gyenes, F.; Sharpe, C.A.; Bergmann, K.E.; Han, H.J.; Gregor, L.B.; Rapolu, R.; Luciano, G.; Welch, J.T. J. Med. Chem. 1995, 38, 3902-3907.
24. Brown, B.A.; Swenson, J.M.; Wallace, R.J., Jr. Broth microdilution test for rapidly growing mycobacteria. In: Clinical Microbiolgy procedures Handbook, Vol. I, American Society for Microbiology, Washington, DC, 1992.