Functional characterization of the native NH2-terminal transactivation domain of the human androgen receptor: Binding kinetics for interactions with TFIIF and SRC-1a

Biochemistry

Volumn 47, Issue 11, 2008, Pages 3352-3359

  Lavery, Derek N ^a,b   McEwan, Iain J ^a  

^a UNIVERSITY OF ABERDEEN   (United Kingdom)

^b IMPERIAL COLLEGE LONDON   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

ANDROGEN RECEPTOR (AR); DISSOCIATION CONSTANTS; TRANSACTIVATION FUNCTION;

BINDING SITES; GENES; LIGANDS; POLYPEPTIDES;

TRANSCRIPTION FACTORS;

ADENOSINE DIPHOSPHATE RIBOSYLATION FACTOR 1; ADENOSINE RECEPTOR; ANDROGEN RECEPTOR; POLYPEPTIDE; RAP 74 PROTEIN; RAP PROTEIN; RNA POLYMERASE II; STEROID RECEPTOR COACTIVATOR 1; STEROID RECEPTOR COACTIVATOR 1A; TRANSCRIPTION FACTOR; TRANSCRIPTION FACTOR TFIIF; UNCLASSIFIED DRUG;

AMINO TERMINAL SEQUENCE; ARTICLE; DISSOCIATION CONSTANT; ENZYME BINDING; ENZYME SUBUNIT; HYDROPHOBICITY; PRIORITY JOURNAL; PROTEIN ANALYSIS; PROTEIN BINDING; PROTEIN DOMAIN; PROTEIN PROTEIN INTERACTION; PROTEIN SECONDARY STRUCTURE; PROTEIN STRUCTURE; RECEPTOR BINDING; RECEPTOR GENE; SURFACE PLASMON RESONANCE; TRANSACTIVATION; TRANSCRIPTION INITIATION;

AMINO ACID SEQUENCE; BINDING SITES; HISTONE ACETYLTRANSFERASES; HUMANS; KINETICS; MOLECULAR SEQUENCE DATA; MUTAGENESIS, SITE-DIRECTED; PEPTIDES; PROTEIN BINDING; PROTEIN INTERACTION MAPPING; PROTEIN STRUCTURE, SECONDARY; PROTEIN STRUCTURE, TERTIARY; PROTEIN SUBUNITS; RECEPTORS, ANDROGEN; SURFACE PLASMON RESONANCE; TRANS-ACTIVATORS; TRANSCRIPTION FACTORS; TRANSCRIPTION FACTORS, TFII;

EID: 40849102545     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi702220p     Document Type: Article

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