Outside-in and inside-out signaling: The new concept that selectivity of ligand binding at the gonadotropin-releasing hormone receptor is modulated by the intracellular environment

Endocrinology

Volumn 145, Issue 8, 2004, Pages 3590-3593

  Millar, Robert P ^a,b   Pawson, Adam J ^a  

^a Med Res Cncl Hum Repro Sci U   (United Kingdom)

^b UNIVERSITY OF EDINBURGH   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

BUSERELIN; GONADORELIN AGONIST; GONADORELIN ANTAGONIST; GONADORELIN DERIVATIVE; GONADORELIN RECEPTOR; PROTEIN KINASE C; RECEPTOR SUBTYPE;

BINDING KINETICS; CONFORMATIONAL TRANSITION; DRUG BINDING SITE; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; HELA CELL; HUMAN; INTRACELLULAR SPACE; LIGAND BINDING; MEDICAL LITERATURE; MOLECULAR STABILITY; NONHUMAN; PRIORITY JOURNAL; PROTEIN DOMAIN; PROTEIN PHOSPHORYLATION; RECEPTOR AFFINITY; SHORT SURVEY; SIGNAL TRANSDUCTION; XENOPUS;

GONADOTROPIN-RELEASING HORMONE; HUMANS; PROTEIN CONFORMATION; PROTEIN KINASE C; RECEPTORS, LHRH; SIGNAL TRANSDUCTION;

EID: 3843102580     PISSN: 00137227     EISSN: None     Source Type: Journal    
DOI: 10.1210/en.2004-0461     Document Type: Short Survey

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