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Volumn 35, Issue 1, 2008, Pages 19-27

In vitro binding of [11C]raclopride with ultrahigh specific activity in rat brain determined by homogenate assay and autoradiography

Author keywords

11C Raclopride; Autoradiography; Homogenate assay; Two affinity binding sites; Ultrahigh specific activity

Indexed keywords

RACLOPRIDE C 11;

EID: 37349016705     PISSN: 09698051     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.nucmedbio.2007.09.009     Document Type: Article
Times cited : (25)

References (36)
  • 1
    • 0022595579 scopus 로고
    • Quantitative analysis of D2 dopamine receptor binding in the living human brain by PET
    • Farde L., Hall H., Ehrin E., and Sedvall G. Quantitative analysis of D2 dopamine receptor binding in the living human brain by PET. Science 231 (1986) 258-261
    • (1986) Science , vol.231 , pp. 258-261
    • Farde, L.1    Hall, H.2    Ehrin, E.3    Sedvall, G.4
  • 2
    • 0026451481 scopus 로고
    • PET studies of dopamine receptors in relation to antipsychotic drug treatment
    • Farde L., Nordstrom A.L., Halldin C., Wiesel F.A., and Sedvall G. PET studies of dopamine receptors in relation to antipsychotic drug treatment. Clin Neuropharmacol 15 Suppl 1 Pt A (1992) 468A-469A
    • (1992) Clin Neuropharmacol , vol.15 , Issue.SUPPL. 1 PART A
    • Farde, L.1    Nordstrom, A.L.2    Halldin, C.3    Wiesel, F.A.4    Sedvall, G.5
  • 3
    • 0027520871 scopus 로고
    • Central D2-dopamine receptor occupancy in relation to antipsychotic drug effects: a double-blind PET study of schizophrenic patients
    • Nordstrom A.L., Farde L., Wiesel F.A., Forslund K., Pauli S., Halldin C., et al. Central D2-dopamine receptor occupancy in relation to antipsychotic drug effects: a double-blind PET study of schizophrenic patients. Biol Psychiatry 33 (1993) 227-235
    • (1993) Biol Psychiatry , vol.33 , pp. 227-235
    • Nordstrom, A.L.1    Farde, L.2    Wiesel, F.A.3    Forslund, K.4    Pauli, S.5    Halldin, C.6
  • 4
    • 0027176890 scopus 로고
    • PET study on striatal dopamine D2 receptor changes during the progression of early Parkinson's disease
    • Rinne J.O., Laihinen A., Rinne U.K., Nagren K., Bergman J., and Ruotsalainen U. PET study on striatal dopamine D2 receptor changes during the progression of early Parkinson's disease. Mov Disord 8 (1993) 134-138
    • (1993) Mov Disord , vol.8 , pp. 134-138
    • Rinne, J.O.1    Laihinen, A.2    Rinne, U.K.3    Nagren, K.4    Bergman, J.5    Ruotsalainen, U.6
  • 5
    • 33846206946 scopus 로고    scopus 로고
    • Effects of repetitive transcranial magnetic stimulation on [(11)C]raclopride binding and cognitive function in patients with depression
    • Kuroda Y., Motohashi N., Ito H., Ito S., Takano A., Nishikawa T., et al. Effects of repetitive transcranial magnetic stimulation on [(11)C]raclopride binding and cognitive function in patients with depression. J Affect Disord 95 1-3 (2006) 35-42
    • (2006) J Affect Disord , vol.95 , Issue.1-3 , pp. 35-42
    • Kuroda, Y.1    Motohashi, N.2    Ito, H.3    Ito, S.4    Takano, A.5    Nishikawa, T.6
  • 6
    • 33745013551 scopus 로고    scopus 로고
    • Is psychological stress in man associated with increased striatal dopamine levels? A [(11)C]raclopride PET study
    • Montgomery A.J., Mehta M.A., and Grasby P.M. Is psychological stress in man associated with increased striatal dopamine levels? A [(11)C]raclopride PET study. Synapse 60 (2006) 124-131
    • (2006) Synapse , vol.60 , pp. 124-131
    • Montgomery, A.J.1    Mehta, M.A.2    Grasby, P.M.3
  • 7
    • 0030612278 scopus 로고    scopus 로고
    • 4 dopamine receptor mRNAs in the primate cerebral cortex vs. neostriatum: effects of chronic treatment with typical and atypical antipsychotic drugs
    • 4 dopamine receptor mRNAs in the primate cerebral cortex vs. neostriatum: effects of chronic treatment with typical and atypical antipsychotic drugs. J Pharmacol Exper Ther 283 (1997) 939-946
    • (1997) J Pharmacol Exper Ther , vol.283 , pp. 939-946
    • Lidow, M.S.1    Goldman-Rakic, P.S.2
  • 8
    • 23044435473 scopus 로고    scopus 로고
    • Parametric mapping of binding in human brain of D2 receptor ligands of different affinities
    • Siessmeier T., Zhou Y., Buchholz H.G., Landvogt C., Vernaleken I., Piel M., et al. Parametric mapping of binding in human brain of D2 receptor ligands of different affinities. J Nucl Med 46 (2005) 964-972
    • (2005) J Nucl Med , vol.46 , pp. 964-972
    • Siessmeier, T.1    Zhou, Y.2    Buchholz, H.G.3    Landvogt, C.4    Vernaleken, I.5    Piel, M.6
  • 11
    • 0033502044 scopus 로고    scopus 로고
    • Quantitation of extrastriatal D2 receptors using a very high-affinity ligand (FLB 457) and the multi-injection approach
    • Delforge J., Bottlaender M., Loc'h C., Guenther I., Fuseau C., Bendriem B., et al. Quantitation of extrastriatal D2 receptors using a very high-affinity ligand (FLB 457) and the multi-injection approach. J Cereb Blood Flow Metab 19 (1999) 533-546
    • (1999) J Cereb Blood Flow Metab , vol.19 , pp. 533-546
    • Delforge, J.1    Bottlaender, M.2    Loc'h, C.3    Guenther, I.4    Fuseau, C.5    Bendriem, B.6
  • 12
    • 0003026818 scopus 로고    scopus 로고
    • Extrastriatal dopamine D2 receptor density and affinity in the human brain measured by 3D PET
    • Suhara T., Sudo Y., Okauchi T., Maeda J., Kawabe K., Suzuki K., et al. Extrastriatal dopamine D2 receptor density and affinity in the human brain measured by 3D PET. Int J Neuropsychopharmacol 2 (1999) 73-82
    • (1999) Int J Neuropsychopharmacol , vol.2 , pp. 73-82
    • Suhara, T.1    Sudo, Y.2    Okauchi, T.3    Maeda, J.4    Kawabe, K.5    Suzuki, K.6
  • 14
    • 34247123791 scopus 로고    scopus 로고
    • Conditioned dopamine release in humans: a positron emission tomography [11C]raclopride study with amphetamine
    • Boileau I., Dagher A., Leyton M., Welfeld K., Booij L., Diksic M., et al. Conditioned dopamine release in humans: a positron emission tomography [11C]raclopride study with amphetamine. J Neurosci 27 (2007) 3998-4003
    • (2007) J Neurosci , vol.27 , pp. 3998-4003
    • Boileau, I.1    Dagher, A.2    Leyton, M.3    Welfeld, K.4    Booij, L.5    Diksic, M.6
  • 18
    • 4344576928 scopus 로고    scopus 로고
    • Effect of amphetamine on [(18)F]fallypride in vivo binding to D(2) receptors in striatal and extrastriatal regions of the primate brain: single bolus and bolus plus constant infusion studies
    • Slifstein M., Narendran R., Hwang D.R., Sudo Y., Talbot P.S., Huang Y., et al. Effect of amphetamine on [(18)F]fallypride in vivo binding to D(2) receptors in striatal and extrastriatal regions of the primate brain: single bolus and bolus plus constant infusion studies. Synapse 54 (2004) 46-63
    • (2004) Synapse , vol.54 , pp. 46-63
    • Slifstein, M.1    Narendran, R.2    Hwang, D.R.3    Sudo, Y.4    Talbot, P.S.5    Huang, Y.6
  • 19
    • 33846427725 scopus 로고    scopus 로고
    • Quantification of PET studies with the very high-affinity dopamine D(2)/D(3) receptor ligand [(11)C]FLB 457: re-evaluation of the validity of using a cerebellar reference region
    • Asselin M.C., Montgomery A.J., Grasby P.M., and Hume S.P. Quantification of PET studies with the very high-affinity dopamine D(2)/D(3) receptor ligand [(11)C]FLB 457: re-evaluation of the validity of using a cerebellar reference region. J Cereb Blood Flow Metab 27 (2007) 378-392
    • (2007) J Cereb Blood Flow Metab , vol.27 , pp. 378-392
    • Asselin, M.C.1    Montgomery, A.J.2    Grasby, P.M.3    Hume, S.P.4
  • 20
    • 0021910620 scopus 로고
    • D-2 dopamine receptors in the frontal cortex of rat and human
    • Liskowsky D.R., and Potter L.T. D-2 dopamine receptors in the frontal cortex of rat and human. Life Sci 36 (1985) 1551-1559
    • (1985) Life Sci , vol.36 , pp. 1551-1559
    • Liskowsky, D.R.1    Potter, L.T.2
  • 27
    • 0033830739 scopus 로고    scopus 로고
    • 2 gas target: effect of irradiation dose, irradiation history, oxygen content and beam energy
    • 2 gas target: effect of irradiation dose, irradiation history, oxygen content and beam energy. Radiochim Acta 88 (2000) 211-215
    • (2000) Radiochim Acta , vol.88 , pp. 211-215
    • Suzuki, K.1    Yamazaki, T.2    Sasaki, M.3    Kubodera, A.4
  • 28
    • 0038397143 scopus 로고    scopus 로고
    • 11C]Ro15-4513 and its application in an extremely low concentration region to an ARG study
    • 11C]Ro15-4513 and its application in an extremely low concentration region to an ARG study. Nucl Med Biol 30 (2003) 335-343
    • (2003) Nucl Med Biol , vol.30 , pp. 335-343
    • Noguchi, J.1    Suzuki, K.2
  • 31
    • 0037687964 scopus 로고    scopus 로고
    • Evaluation of the binding characteristics of [5-(11)C-methoxy]donepezil in the rat brain for in vivo visualization of acetylcholinesterase
    • Funaki Y., Kato M., Iwata R., Sakurai E., Tashiro M., Ido T., et al. Evaluation of the binding characteristics of [5-(11)C-methoxy]donepezil in the rat brain for in vivo visualization of acetylcholinesterase. J Pharmacol Sci 91 (2003) 105-112
    • (2003) J Pharmacol Sci , vol.91 , pp. 105-112
    • Funaki, Y.1    Kato, M.2    Iwata, R.3    Sakurai, E.4    Tashiro, M.5    Ido, T.6
  • 32
    • 37349120834 scopus 로고    scopus 로고
    • Development and validation of an ultra-fast LC method for the quality control of PET radiopharmaceuticals
    • Nakao R., Ito T., Hayashi K., and Suzuki K. Development and validation of an ultra-fast LC method for the quality control of PET radiopharmaceuticals. J Labelled Compd Radiopharm 50 (2007) S508
    • (2007) J Labelled Compd Radiopharm , vol.50
    • Nakao, R.1    Ito, T.2    Hayashi, K.3    Suzuki, K.4
  • 33
    • 0021844076 scopus 로고
    • Specific in vitro binding of 3H-raclopride. A potent substituted benzamide drug with high affinity for dopamine D-2 receptors in the rat brain
    • Kohler C., Hall H., Ogren S.O., and Gawell L. Specific in vitro binding of 3H-raclopride. A potent substituted benzamide drug with high affinity for dopamine D-2 receptors in the rat brain. Biochem Pharmacol 34 (1985) 2251-2259
    • (1985) Biochem Pharmacol , vol.34 , pp. 2251-2259
    • Kohler, C.1    Hall, H.2    Ogren, S.O.3    Gawell, L.4
  • 34
    • 0023755705 scopus 로고
    • Quantitative autoradiography of major neurotransmitter receptors in the monkey striate and extrastriate cortex
    • Rakic P., Goldman-Rakic P.S., and Gallager D. Quantitative autoradiography of major neurotransmitter receptors in the monkey striate and extrastriate cortex. J Neurosci 8 (1988) 3670-3690
    • (1988) J Neurosci , vol.8 , pp. 3670-3690
    • Rakic, P.1    Goldman-Rakic, P.S.2    Gallager, D.3
  • 35
    • 0027433305 scopus 로고
    • Comparison of two PET radioligand for imaging extrastriatal dopamine receptors in the human brain
    • Wang G.J., Volkow N.D., Fowler J.S., Wolf A.P., MacGregor R.R., Shea C.E., et al. Comparison of two PET radioligand for imaging extrastriatal dopamine receptors in the human brain. Synapse 15 (1993) 246-249
    • (1993) Synapse , vol.15 , pp. 246-249
    • Wang, G.J.1    Volkow, N.D.2    Fowler, J.S.3    Wolf, A.P.4    MacGregor, R.R.5    Shea, C.E.6
  • 36
    • 2942622711 scopus 로고    scopus 로고
    • Differentiation of extrastriatal dopamine D2 receptor density and affinity in the human brain using PET
    • Olsson H., Halldin C., and Farde L. Differentiation of extrastriatal dopamine D2 receptor density and affinity in the human brain using PET. Neuroimage 22 (2004) 794-803
    • (2004) Neuroimage , vol.22 , pp. 794-803
    • Olsson, H.1    Halldin, C.2    Farde, L.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.