A covalent inhibitor targeting an intermediate conformation of the fusogenic subunit of the HIV-1 envelope complex

Journal of Biological Chemistry

Volumn 282, Issue 44, 2007, Pages 32406-32413

  Jacobs, Amy ^a   Quraishi, Omar ^b   Huang, Xicai ^b   Bousquet Gagnon, Nathalie ^b   Nault, Geneviève ^b   Francella, Nicholas ^a   Alvord, W Gregory ^a   Pham, Nga ^b   Soucy, Chantal ^b   Robitaille, Martin ^b   Bridon, Dominique ^b   Blumenthal, Robert ^a  

^a NATIONAL CANCER INSTITUTE   (United States)

^b INSTITUTE FOR RESEARCH IN IMMUNOLOGY AND CANCER   (Canada)

Author keywords

[No Author keywords available]

Indexed keywords

BINDING SITES; COVALENT BONDS; DISEASE CONTROL; GENE ENCODING; GLYCOPROTEINS; IMMUNOLOGY;

COVALENT REACTION; FUSOGENIC SUBUNITS; PEPTIDE INHIBITORS;

PEPTIDES;

ANTIVIRUS AGENT; GLYCOPROTEIN GP 41; PEPTIDE DERIVATIVE; VIRUS ENVELOPE PROTEIN;

ARTICLE; COVALENT BOND; PRIORITY JOURNAL; PROTEIN BINDING; PROTEIN CONFORMATION; TEMPERATURE;

ANTI-HIV AGENTS; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; HIV ENVELOPE PROTEIN GP41; HIV-1; INHIBITORY CONCENTRATION 50; MODELS, BIOLOGICAL; PEPTIDES; PROTEIN CONFORMATION; PROTEIN FOLDING; VIRUS INTERNALIZATION;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 36148954295     PISSN: 00219258     EISSN: 1083351X     Source Type: Journal    
DOI: 10.1074/jbc.M705577200     Document Type: Article

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