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Volumn 10, Issue 6, 2007, Pages 777-785

PET measurement of serotonin transporter occupancy: A comparison of escitalopram and citalopram

Author keywords

5 HTT; 11C MADAM; Escitalopram; Human; PET

Indexed keywords

CITALOPRAM; ESCITALOPRAM; SEROTONIN TRANSPORTER;

EID: 35248895978     PISSN: 14611457     EISSN: 14695111     Source Type: Journal    
DOI: 10.1017/S1461145706007486     Document Type: Article
Times cited : (51)

References (36)
  • 1
    • 0038408827 scopus 로고    scopus 로고
    • Positron emission tomographic analysis of dose-dependent NAD-299 binding to 5-hydroxytryptamine-1A receptors in the human brain
    • Andree B, Hedman A, Thorberg SO, Nilsson D, Halldin C, Farde L (2003). Positron emission tomographic analysis of dose-dependent NAD-299 binding to 5-hydroxytryptamine-1A receptors in the human brain. Psychopharmacology (Berlin) 167, 37-45.
    • (2003) Psychopharmacology (Berlin) , vol.167 , pp. 37-45
    • Andree, B.1    Hedman, A.2    Thorberg, S.O.3    Nilsson, D.4    Halldin, C.5    Farde, L.6
  • 5
    • 0036236470 scopus 로고    scopus 로고
    • Fixed-dose trial of the single isomer SSRI escitalopram in depressed outpatients
    • Burke WJ, Gergel I, Bose A (2002). Fixed-dose trial of the single isomer SSRI escitalopram in depressed outpatients. Journal of Clinical Psychiatry 63, 331-336.
    • (2002) Journal of Clinical Psychiatry , vol.63 , pp. 331-336
    • Burke, W.J.1    Gergel, I.2    Bose, A.3
  • 6
    • 13244262698 scopus 로고    scopus 로고
    • The S-enantiomer of R,S-citalopram, increases inhibitor binding to the human serotonin transporter by an allosteric mechanism. Comparison with other serotonin transporter inhibitors
    • Chen F, Larsen MB, Sanchez C, Wiborg O (2005). The S-enantiomer of R,S-citalopram, increases inhibitor binding to the human serotonin transporter by an allosteric mechanism. Comparison with other serotonin transporter inhibitors. European Neuropsychopharmacology 15, 193-198.
    • (2005) European Neuropsychopharmacology , vol.15 , pp. 193-198
    • Chen, F.1    Larsen, M.B.2    Sanchez, C.3    Wiborg, O.4
  • 8
    • 27144516427 scopus 로고    scopus 로고
    • A randomized, double-blind, 24-week study of escitalopram (10 mg/day) versus citalopram (20 mg/day) in primary care patients with major depressive disorder
    • Colonna L, Andersen HF, Reines EH (2005). A randomized, double-blind, 24-week study of escitalopram (10 mg/day) versus citalopram (20 mg/day) in primary care patients with major depressive disorder. Current Medical Research and Opinion 21, 1659-68.
    • (2005) Current Medical Research and Opinion , vol.21 , pp. 1659-1668
    • Colonna, L.1    Andersen, H.F.2    Reines, E.H.3
  • 9
    • 0029937457 scopus 로고    scopus 로고
    • The advantage of using positron emission tomography in drug research
    • Farde L (1996). The advantage of using positron emission tomography in drug research. Trends in Neurosciences 19, 211-214.
    • (1996) Trends in Neurosciences , vol.19 , pp. 211-214
    • Farde, L.1
  • 10
    • 0023853769 scopus 로고
    • Central D2-dopamine receptor occupancy in schizophrenic patients treated with antipsychotic drugs
    • Farde L, Wiesel FA, Halldin C, Sedvall G (1988). Central D2-dopamine receptor occupancy in schizophrenic patients treated with antipsychotic drugs. Archives of General Psychiatry 45, 71-76.
    • (1988) Archives of General Psychiatry , vol.45 , pp. 71-76
    • Farde, L.1    Wiesel, F.A.2    Halldin, C.3    Sedvall, G.4
  • 11
    • 0037732753 scopus 로고    scopus 로고
    • An evaluation of the potential for pharmacokinetic interaction between escitalopram and the cytochrome P450 3A4 inhibitor ritonavir
    • Gutierrez MM, Rosenberg J, Abramowitz W (2003). An evaluation of the potential for pharmacokinetic interaction between escitalopram and the cytochrome P450 3A4 inhibitor ritonavir. Clinical Therapeutics 25, 1200-1210.
    • (2003) Clinical Therapeutics , vol.25 , pp. 1200-1210
    • Gutierrez, M.M.1    Rosenberg, J.2    Abramowitz, W.3
  • 12
    • 26644455497 scopus 로고    scopus 로고
    • 11)C]MADAM, a new serotonin transporter radioligand characterized in the monkey brain by PET. Synapse 58, 173-183.
    • 11)C]MADAM, a new serotonin transporter radioligand characterized in the monkey brain by PET. Synapse 58, 173-183.
  • 15
    • 0030468875 scopus 로고    scopus 로고
    • Simplified reference tissue model for PET receptor studies
    • Lammertsma AA, Hume SP (1996). Simplified reference tissue model for PET receptor studies. Neuroimage 4, 153-158.
    • (1996) Neuroimage , vol.4 , pp. 153-158
    • Lammertsma, A.A.1    Hume, S.P.2
  • 16
    • 0038441914 scopus 로고    scopus 로고
    • Escitalopram (10-20 mg/day) is effective and well tolerated in a placebo-controlled study in depression in primary care
    • Lepola UM, Loft H, Reines EH (2003). Escitalopram (10-20 mg/day) is effective and well tolerated in a placebo-controlled study in depression in primary care. International Clinical Psychopharmacology 18, 211-217.
    • (2003) International Clinical Psychopharmacology , vol.18 , pp. 211-217
    • Lepola, U.M.1    Loft, H.2    Reines, E.H.3
  • 17
    • 33745869766 scopus 로고    scopus 로고
    • 11C]MADAM: A test-retest reproducibility study
    • 11C]MADAM: a test-retest reproducibility study. Synapse 60, 256-263.
    • (2006) Synapse , vol.60 , pp. 256-263
    • Lundberg, J.1    Halldin, C.2    Farde, L.3
  • 21
    • 0021364348 scopus 로고
    • A quantitative model for the in vivo assessment of drug binding sites with positron emission tomography
    • Mintun MA, Raichle ME, Kilbourn MR, Wooten GF, Welch MJ (1984). A quantitative model for the in vivo assessment of drug binding sites with positron emission tomography. Annals of Neurology 15, 217-227.
    • (1984) Annals of Neurology , vol.15 , pp. 217-227
    • Mintun, M.A.1    Raichle, M.E.2    Kilbourn, M.R.3    Wooten, G.F.4    Welch, M.J.5
  • 22
    • 0034997617 scopus 로고    scopus 로고
    • Escitalopram (S-enantiomer of citalopram) : Clinical efficacy and onset of action predicted from a rat model
    • Montgomery SA, Loft H, Sanchez C, Reines EH, Papp M (2001). Escitalopram (S-enantiomer of citalopram) : clinical efficacy and onset of action predicted from a rat model. Pharmacology & Toxicology 88, 282-286.
    • (2001) Pharmacology & Toxicology , vol.88 , pp. 282-286
    • Montgomery, S.A.1    Loft, H.2    Sanchez, C.3    Reines, E.H.4    Papp, M.5
  • 23
    • 17644423099 scopus 로고    scopus 로고
    • Prospective, multicentre, randomized, double-blind study of the efficacy of escitalopram versus citalopram in outpatient treatment of major depressive disorder
    • Moore N, Verdoux H, Fantino B (2005). Prospective, multicentre, randomized, double-blind study of the efficacy of escitalopram versus citalopram in outpatient treatment of major depressive disorder. International Clinical Psychopharmacology 20, 131-137.
    • (2005) International Clinical Psychopharmacology , vol.20 , pp. 131-137
    • Moore, N.1    Verdoux, H.2    Fantino, B.3
  • 24
    • 0038168734 scopus 로고    scopus 로고
    • The R-enantiomer of citalopram counteracts escitalopram-induced increase in extracellular 5-HT in the frontal cortex of freely moving rats
    • Mork A, Kreilgaard M, Sanchez C (2003). The R-enantiomer of citalopram counteracts escitalopram-induced increase in extracellular 5-HT in the frontal cortex of freely moving rats. Neuropharmacology 45, 167-173.
    • (2003) Neuropharmacology , vol.45 , pp. 167-173
    • Mork, A.1    Kreilgaard, M.2    Sanchez, C.3
  • 25
    • 0035450364 scopus 로고    scopus 로고
    • Second-generation SSRIs: Human monoamine transporter binding profile of escitalopram and R-fluoxetine
    • Owens MJ, Knight DL, Nemeroff CB (2001). Second-generation SSRIs: human monoamine transporter binding profile of escitalopram and R-fluoxetine. Biological Psychiatry 50, 345-350.
    • (2001) Biological Psychiatry , vol.50 , pp. 345-350
    • Owens, M.J.1    Knight, D.L.2    Nemeroff, C.B.3
  • 26
    • 0029035234 scopus 로고
    • Analysis of enantiomers of citalopram and its demethylated metabolites in plasma of depressive patients using chiral reverse-phase liquid chromatography
    • Rochat B, Amey M, Baumann P (1995). Analysis of enantiomers of citalopram and its demethylated metabolites in plasma of depressive patients using chiral reverse-phase liquid chromatography. Therapeutic Drug Monitoring 17, 273-279.
    • (1995) Therapeutic Drug Monitoring , vol.17 , pp. 273-279
    • Rochat, B.1    Amey, M.2    Baumann, P.3
  • 28
    • 0037454123 scopus 로고    scopus 로고
    • R-citalopram attenuates anxiolytic effects of escitalopram in a rat ultrasonic vocalisation model
    • Sanchez C (2003). R-citalopram attenuates anxiolytic effects of escitalopram in a rat ultrasonic vocalisation model. European Journal of Pharmacology 464, 155-158.
    • (2003) European Journal of Pharmacology , vol.464 , pp. 155-158
    • Sanchez, C.1
  • 30
    • 0142074886 scopus 로고    scopus 로고
    • R-citalopram counteracts the effect of escitalopram in a rat conditioned fear stress model of anxiety
    • Sanchez C, Gruca P, Bien E, Papp M (2003a). R-citalopram counteracts the effect of escitalopram in a rat conditioned fear stress model of anxiety. Pharmacology, Biochemistry, and Behavior 75, 903-907.
    • (2003) Pharmacology, Biochemistry, and Behavior , vol.75 , pp. 903-907
    • Sanchez, C.1    Gruca, P.2    Bien, E.3    Papp, M.4
  • 31
    • 0141534297 scopus 로고    scopus 로고
    • R-citalopram counteracts the antidepressant-like effect of escitalopram in a rat chronic mild stress model
    • Sanchez C, Gruca P, Papp M (2003b). R-citalopram counteracts the antidepressant-like effect of escitalopram in a rat chronic mild stress model. Behavioural Pharmacology 14, 465-470.
    • (2003) Behavioural Pharmacology , vol.14 , pp. 465-470
    • Sanchez, C.1    Gruca, P.2    Papp, M.3
  • 32
    • 0030682236 scopus 로고    scopus 로고
    • Steady-state pharmacokinetics of the enantiomers of citalopram and its metabolites in humans
    • Sidhu J, Priskorn M, Poulsen M, Segonzac A, Grollier G, Larsen F (1997). Steady-state pharmacokinetics of the enantiomers of citalopram and its metabolites in humans. Chirality 9, 686-692.
    • (1997) Chirality , vol.9 , pp. 686-692
    • Sidhu, J.1    Priskorn, M.2    Poulsen, M.3    Segonzac, A.4    Grollier, G.5    Larsen, F.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.