A rapid synthesis of 3-sulfenyl indoles using Selectfluor™

Tetrahedron Letters

Volumn 48, Issue 39, 2007, Pages 7034-7037

  Yadav, J S ^a   Reddy, B V Subba ^a   Reddy, Y Jayasudhan ^a  

^a INDIAN INSTITUTE OF CHEMICAL TECHNOLOGY   (India)

Author keywords

3 Arylthioindoles; Indoles; Thiolation; Thiols

Indexed keywords

1 CHLOROMETHYL 4 FLUORO 1,4 DIAZONIABICYCLO[2,2,2]OCTANE BIS(TETRAFLUOROBORIC ACID); 3 SULFENYL INDOLE DERIVATIVE; 3 THIOINDOLE DERIVATIVE; INDOLE DERIVATIVE; REAGENT; THIOL; UNCLASSIFIED DRUG;

ARTICLE; DRUG STRUCTURE; DRUG SYNTHESIS; MASS SPECTROMETRY; PROTON NUCLEAR MAGNETIC RESONANCE; STOICHIOMETRY;

EID: 34548280409     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tetlet.2007.07.130     Document Type: Article

References (26)

1. Maeda Y., Koyabu M., Nishimura T., and Uemura S. J. Org. Chem. 69 (2004) 7688-7693
2. Campbell J.A., Broka C.A., Gong L., Walker K.A.M., and Wang J.-H. Tetrahedron Lett. 45 (2004) 4073-4075
3. Williams T.M., Ciccarone T.M., MacTough S.C., Rooney C.S., Balani S.K., Condra J.H., Emini E.A., Goldman M.E., Greenlee W.J., Kauffman L.R., O'Brien J.A., Sardana V.V., Schleif W.A., Theoharides A.D., and Anderson P.S. J. Med. Chem. 36 (1993) 1291-1294
4. Silvestri R., De Martino G., La Regina G., Artico M., Massa S., Vargiu L., Mura M., Loi A.G., Marceddu T., and La Colla P. J. Med. Chem. 46 (2003) 2482-2493
5. Avis I., Marti{dotless}nez A., Tauler J., Zudaire E., Mayburd A., Abu-Ghazaleh R., Ondrey F., and Mulshine J.L. Cancer Res. 65 (2005) 4181-4190
6. De Martino G., La Regina G., Coluccia A., Edler M.C., Barbera M.C., Brancale A., Wilcox E., Hamel E., Artico M., and Silvestri R. J. Med. Chem. 47 (2004) 6120-6123
7. Funk C.D. Nat. Rev. Drug Disc. 4 (2005) 664-672
8. Khandekar S.S., Gentry D.R., Van Aller G.S., Doyle M.L., Chambers P.A., Konstantinidis A.K., Brandt M., Daines R.A., and Lonsdale J.T. J. Biol. Chem. 276 (2001) 30024-30030
9. Atkinson J.G., Hamel P., and Girard Y. Synthesis (1988) 480-481
10. Scoffone E., Fontana A., and Rocchi R. Biochemistry 7 (1968) 971-979
11. Anzai K. J. Heterocycl. Chem. 16 (1979) 567-569
12. Raban M., and Chern L. J. Org. Chem. 45 (1980) 1688-1691
13. Ranken P.F., and McKinnie B.G. J. Org. Chem. 54 (1989) 2985-2988
14. Browder C.C., Mitchell M.O., Smith R.L., and El-Sulayman G. Tetrahedron Lett. 34 (1993) 6245-6246
15. Matsugi M., Murata K., Gotanda K., Nambu H., Anilkumar G., Matsumoto K., and Kita Y. J. Org. Chem. 66 (2001) 2434-2441
16. Tudge M., Tamiya M., Savarin C., and Humphrey G.R. Org. Lett. 8 (2006) 565-568
17. Schlosser K.M., Krasutsky A.P., Hamilton H.W., Reed J.E., and Sexton K. Org. Lett. 6 (2004) 819-821
18. Singh R.P., and Shreeve J.M. Acc. Chem. Res. 37 (2004) 31-44
19. Stavbera S., and Zupan M. Acta Chim. Slov. 52 (2005) 13-26
20. Nyffeler P.T., Duron S.G., Burkart M.D., Vincent S.P., and Wong C.-H. Angew. Chem., Int. Ed. 44 (2005) 192-212
21. Yadav J.S., Reddy B.V.S., and Srinivas Reddy Ch. Tetrahedron Lett. 45 (2004) 1291-1293
22. Yadav J.S., Reddy B.V.S., Sunitha V., and Reddy K.S. Adv. Synth. Catal. 345 (2003) 1203-1206
23. Syvret R.G., Butt K.M., Nguyen T.P., Bulleck V.L., and Rieth R.D. J. Org. Chem. 67 (2002) 4487-4493
24. Stavber S., Jereb M., and Zupan M. Chem. Commun. (2002) 488
25. Manandhar S., Singh R.P., Eggers G.V., and Shreeve J.M. J. Org. Chem. 67 (2002) 6415-6420
26. +): 274.0457. Found: 274.0459.