A novel ketolide class: Synthesis and antibacterial activity of a lead compound

Bioorganic and Medicinal Chemistry Letters

Volumn 17, Issue 18, 2007, Pages 5265-5269

  Andreotti, Daniele ^a   Bientinesi, Ilaria ^a   Biondi, Stefano ^b   Donati, Daniele ^a   Erbetti, Isabelle ^a   Lociuro, Sergio ^c   Marchioro, Carla ^a   Pozzan, Alfonso ^a   Ratti, Emiliangelo ^a   Terreni, Silvia ^a  

^a GSK   (Italy)

^b NicOx Research Institute   (Italy)

^c Arpida Ltd   (Switzerland)

Author keywords

Antibacterial; GW680788X; Ketolides; Macrolides

Indexed keywords

CETHROMYCIN; CLARITHROMYCIN; ERYTHROMYCIN; GW 680788X; KETOLIDE; TELITHROMYCIN; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ARTICLE; BACTERIAL STRAIN; CONTROLLED STUDY; CYCLIZATION; DECARBOXYLATION; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; METHYLATION; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; OXIDATION; SPECTROSCOPY; STEREOCHEMISTRY;

ANTI-BACTERIAL AGENTS; KETOLIDES; MICROBIAL SENSITIVITY TESTS; MODELS, MOLECULAR;

EID: 34547868479     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2007.02.019     Document Type: Article

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