Conformationally restricted monoprotected diamines as scaffolds for design of biologically active compounds and peptidomimetics

Chimica Oggi

Volumn 25, Issue 3 SUPPL., 2007, Pages 12-13

  Shivanyuk, Alexander N ^a,b   Volochnyuk, Dmitry M ^b,c   Komarov, Igor V ^a,b   Nazarenko, Konstantin G ^d   Radchenko, Dmitry S ^a,b   Kostyuk, Alexander ^b,c   Tolmachev, Andrey A ^a,b  

^a TARAS SHEVCHENKO NATIONAL UNIVERSITY OF KYIV   (Ukraine)

^b ENAMINE LTD   (Ukraine)

^c INSTITUTE OF ORGANIC CHEMISTRY   (Ukraine)

^d NONE

Author keywords

[No Author keywords available]

Indexed keywords

EID: 34547179933     PISSN: 0392839X     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (19)

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2. For a review on peptidomimetics see: J. Gante Angew Chem. Int. Ed. 1994, 33, 1699-1720.
3. For a review see: S. R. S. S. Kotti, C. Timmons, G. Li Chem. Biol. Drug Des. 2005, 67, 101-114.
4. K. Tomita, Y. Tsuzuki, K. Shibamori, M. Tashima, EKajikawa, Y. Sato, S. Kashimoto, K. Chiba K. Hino J. Med. Chem. 2002, 45, 5564-5575
5. V. A. Kumar, M. D. Costa, P. S. Lonkar, M. P. S. Pallan, K. N. Ganesh Pure. & Appl. Chem.2004, 76, 1599-1603.
6. M. L. Skar, J. S. Svendsen Tetrahedron 1997, 53, 17425-17440.
7. MMX force field, PCMODEL 7, Serena Software, Dr. K. E. Gilbert, P.O. 3076, Bloomington, IN 47402.
8. www.enamine.net
9. I. V. Komarov, O. O. Grigorenko, D. S. Radchenko, O.S. Artamonov, A. N. Kostyuk, A. A. Tolmachov Chemistry Today 2006, 24, 22-23.
10. For synthesis of compound 3 see: J. K. Pokorski, M. C. Myers, D. H. Apella Tetrahedron Lett. 2005, 46, 905-917.
11. For synthesis of syn-diastereomer compound 4 see: R. Kuang, D. Blythin, N. - Y. Shih, H. - J Shue, J.Cao, D. Cu, Y. Huang, J. H. Schwerdt, P. C. Ting, S. - C. Wong, Li. Xiao WO 2005/116009.
12. For original synthesis of compound 5 see: Y. Tsuzuki, K. Chiba, M. Kazahiro, T. Kyoji, K. Suzuki, Tetrahedron: Asymmetry 2001, 12, 2989 - 2997.
13. For original synthesis of compound 8-11 see: T. Schenke, U. Petersen US 5071999.
14. For original synthesis of compound 13 see: D. P. Becker, R. K. Husa, A. E. Moormann, C. I. Villamil, D. L. Flynn Tetrahedron 1999, 55, 11787-11802.
15. For original synthesis of compounds 14 and 15 see: A. deMeijere, C. M. Williams, A. Kourdioukov, S. V. Sviridov,V. Chaplinski, M. Kordes, A. I. Savchenko, C. Stratmann, M. Noltemeyer Chem. Eur. J. 2002, 8, 3788-3801.
16. For original synthesis of compound 16 and 17 see: D. J. Blythin, X. Chen, R. J. Friary, K. D. Mccormick, J. J. Piwinski, N.-Y. Shih, H.-J. Shue. US 5968929.
17. For original synthesis of compound 20 and 21 see: a) S. Ciblat, J.-L. Canet, Y. Troin Tetrahedron Lett. 2001, 42, 4815-4817;
18. b) B. Bollbuck, A. Denholmritain, L. Revesz, A. Schlapbach, R. Walchli J. Eder, R. Hersperger, P. Janser WO 2004/089913.
19. For original synthesis of compound 22 see: U. Petersen, T. Schenke, A. Krebs, K.Grohe, M. Schriewer, I. Haller, K. G. Metzger, R Endermann, H.-J. Zeiler US 5059597.