Synthesis and bioevaluation of N-(arylalkyl)-homospermidine conjugates

Bioorganic and Medicinal Chemistry Letters

Volumn 17, Issue 16, 2007, Pages 4471-4475

  Xie, Songqiang ^a   Cheng, Pengfei ^a   Liu, Guangchao ^a   Ma, Yuangfang ^a   Zhao, Jin ^a   Chehtane, Mounir ^b   Khaled, Annette R ^b   Phanstiel IV, Otto ^b   Wang, Chaojie ^a  

^a HENAN UNIVERSITY   (China)

^b UNIVERSITY OF CENTRAL FLORIDA   (United States)

Author keywords

Apoptosis; Homospermidine; Polyamine conjugate; Synthesis

Indexed keywords

4 BIPHENYLMETHYL HOMOSPERMIDINE; 9 ANTHRACENEMETHYL HOMOSPERMIDINE; EFLORNITHINE; HOMOSPERMIDINE; INTERLEUKIN 3; POLYAMINE DERIVATIVE; SPERMIDINE DERIVATIVE; UNCLASSIFIED DRUG;

APOPTOSIS; ARTICLE; CARBON NUCLEAR MAGNETIC RESONANCE; CELL CYCLE; CYTOTOXICITY; DRUG SYNTHESIS; HELA CELL; HUMAN; LEUKEMIA L 1210; MELANOMA B16; NONHUMAN; PROTON NUCLEAR MAGNETIC RESONANCE;

ANIMALS; ANTINEOPLASTIC AGENTS; APOPTOSIS; CELL LINE, TUMOR; DOSE-RESPONSE RELATIONSHIP, DRUG; HUMANS; INTERLEUKIN-3; MICE; MOLECULAR STRUCTURE; SPERMIDINE; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 34447331679     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2007.06.009     Document Type: Article

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