Synthesis of enantiomerically pure α-[4-(1-substituted)-1,2,3-triazol-4-yl]-benzylacetamides via microwave-assisted click chemistry: towards new potential antimicrobial agents

Tetrahedron Asymmetry

Volumn 18, Issue 11, 2007, Pages 1345-1350

  Castagnolo, Daniele ^a   Dessì, Filippo ^a   Radi, Marco ^a   Botta, Maurizio ^a  

^a UNIVERSITY OF SIENA   (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

ACETAMIDE DERIVATIVE; AMINE; ANTIINFECTIVE AGENT; COPPER;

ARTICLE; CHEMISTRY; MICROWAVE RADIATION; PRIORITY JOURNAL;

EID: 34447095599     PISSN: 09574166     EISSN: 1362511X     Source Type: Journal    
DOI: 10.1016/j.tetasy.2007.06.007     Document Type: Article

References (18)

1. Buchel K.H., Draber W., Regel E., and Plempel M. Arzneim.-Forsch. 22 (1972) 1260-1272
2. Heeres J., Backx L.J.J., Mostmans J.H., and Van Cutsem J. J. Med. Chem. 22 (1979) 1003-1005
3. Koltin Y. Annu. Rep. Med. Chem. 25 (1990) 141-148
4. Huy N.T., Kamei E., Kondo Y., Serada S., Kanaori K., Takano R., Tajima K., and Hara S. J. Biochem. 131 (2002) 437-444
5. Corelli F., Summa V., Brogi A., Monteagudo E., and Botta M. J. Org. Chem. 60 (1995) 2008-2015
6. Messina F., Botta M., Corelli F., Schneider M.P., and Fazio F. J. Org. Chem. 64 (1999) 3767-3769
7. Botta M., Corelli F., Gasparrini F., Messina F., and Mugnaini C. J. Org. Chem. 65 (2000) 4736-4739
8. Messina F., Botta M., Corelli F., and Paladino A. Tetrahedron: Asymmetry 11 (2000) 4895-4901
9. Tafi A., Costi R., Botta M., Di Santo R., Corelli F., Massa S., Ciacci A., Manetti F., and Artico M. J. Med. Chem. 45 (2002) 2720-2732
10. Di Santo R., Tafi A., Costi R., Botta M., Artico M., Corelli F., Forte M., Caporuscio F., Angiolella L., and Palamara A.T. J. Med. Chem. 48 (2005) 5140-5153
11. Kolb H.C., Finn M.G., and Sharpless K.B. Angew. Chem., Int. Ed. 40 (2001) 2004-2021
12. Kolb H.C., and Sharpless K.B. Drug Discovery Today 8 (2003) 1128-1137
13. Bock V.D., Hiemstra H., and van Maarseveen J.H. Eur. J. Org. Chem. (2006) 51-68
14. Huisgen R. In: Padwa A. (Ed). 1,3-Dipolar Cycloaddition Chemistry (1984), Wiley, New York
15. Castagnolo D., Renzulli M.L., Galletti E., Corelli F., and Botta M. Tetrahedron: Asymmetry 16 (2005) 2893-2896
16. Appukkuttan P., Dehaen W., Fokin V.V., and Van der Eycken E. Org. Lett. 6 (2004) 4223-4225
17. Rostovtsev V.V., Green L.G., Fokin V.V., and Sharpless K.B. Angew. Chem., Int. Ed. 41 (2002) 2596-2599
18. Pagliai F., Pirali T., Del Grosso E., Di Brisco R., Tron G.C., Sorba G., and Genazzani A.A. J. Med. Chem. 49 (2006) 467-470