Synthesis and biological activity of naphthalene analogues of phenstatins: Naphthylphenstatins

Bioorganic and Medicinal Chemistry Letters

Volumn 17, Issue 12, 2007, Pages 3417-3420

  Álvarez, Concepción ^a   Álvarez, Raquel ^a   Corchete, Purificación ^a   Pérez Melero, Concepción ^a   Peláez, Rafael ^a   Medarde, Manuel ^a  

^a UNIVERSITY OF SALAMANCA   (Spain)

Author keywords

Antitumour; Combretastatins; Cytotoxicity; Phenstatins; Synthesis; Tubulin

Indexed keywords

CARBONYL DERIVATIVE; COMBRETASTATIN; NAPHTHALENE DERIVATIVE;

ARTICLE; CANCER CELL CULTURE; DRUG CYTOTOXICITY; DRUG DETERMINATION; DRUG POTENCY; DRUG SYNTHESIS; HUMAN; HUMAN CELL; IC 50; MICROTUBULE ASSEMBLY; QUANTUM YIELD; REACTION ANALYSIS; STRUCTURE ACTIVITY RELATION;

ANTINEOPLASTIC AGENTS; BIBENZYLS; HELA CELLS; HUMANS; INHIBITORY CONCENTRATION 50; MODELS, CHEMICAL; NAPHTHALENES; STEREOISOMERISM; STILBENES; STRUCTURE-ACTIVITY RELATIONSHIP; TUBULIN; TUBULIN MODULATORS; TUMOR CELLS, CULTURED;

EID: 34249323026     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2007.03.082     Document Type: Article

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