Directed molecular screening for RecA ATPase inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 17, Issue 12, 2007, Pages 3249-3253

  Wigle, Tim J ^a   Singleton, Scott F ^a  

^a UNIVERSITY OF NORTH CAROLINA   (United States)

Author keywords

Antibiotic resistance; DNA repair; High throughput screening; RecA; Recombination

Indexed keywords

4 AMINO 7 TERT BUTYL 5 (4 CHLOROPHENYL)PYRAZOLO[3,4 D]PYRIMIDINE; ADENOSINE DIPHOSPHATE; ADENOSINE TRIPHOSPHATASE INHIBITOR; CINNAMALDEHYDE; CONGO RED; COUMAMYCIN; CURCUMIN; GENISTEIN; GENISTIN; METHOTREXATE; NOVOBIOCIN; NUCLEOTIDE DERIVATIVE; PROTEIN KINASE C INHIBITOR; PYRIDOXAL PHOSPHATE 6 AZOPHENYL 2',4' DISULFONIC ACID; RADICICOL; RECA PROTEIN; SCAFFOLD PROTEIN; SURAMIN; TENOFOVIR; VANILLIN;

ANTIBIOTIC RESISTANCE; ARTICLE; DRUG SCREENING; ENZYME ACTIVITY; ENZYME ASSAY; ENZYME INHIBITION; FLUORESCENCE; GENETIC VARIABILITY; HYDROLYSIS; MOLECULAR BIOLOGY; MOLECULAR EVOLUTION; NONHUMAN; RECA GENE;

ADENOSINE DIPHOSPHATE; ADENOSINE TRIPHOSPHATASES; ADENOSINE TRIPHOSPHATE; BINDING SITES; BIOLOGICAL ASSAY; DNA GYRASE; DRUG EVALUATION, PRECLINICAL; ENZYME INHIBITORS; ESCHERICHIA COLI; FLUORESCENT DYES; HYDROLYSIS; NUCLEOTIDES; PROTEIN-TYROSINE KINASES; REC A RECOMBINASES; SENSITIVITY AND SPECIFICITY; SURAMIN; TIME FACTORS;

BACTERIA (MICROORGANISMS);

EID: 34249289724     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2007.04.013     Document Type: Article

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