Acid-catalyzed synthesis of oxathiolone fused chalcones. Comparison of their activity toward various microorganisms and human cancer cells line

European Journal of Medicinal Chemistry

Volumn 42, Issue 5, 2007, Pages 729-733

  Konieczny, Marek T ^a   Konieczny, Wojciech ^a   Sabisz, Michał ^b   Skladanowski, Andrzej ^b   Wakieć, Roland ^b   Augustynowicz Kopeć, Ewa ^c   Zwolska, Zofia ^c  

^a MEDICAL UNIVERSITY OF GDANSK   (Poland)

^b GDANSK UNIVERSITY OF TECHNOLOGY   (Poland)

^c NATIONAL TUBERCULOSIS AND LUNG DISEASES RESEARCH INSTITUTE   (Poland)

Author keywords

Antibacterial; Antifungal; Chalcones; Cytotoxic; Oxathiolone; Tuberculostatic

Indexed keywords

5 METHOXY 4 (3 PHENYLACRYOLYLBENZO[D][1,3] OXATHIOL 2 ONE; 5 METHOXY 4 [3 (2' CHLOROPHENYL)ACRYOLYL]BENZO [D][1,3]OXATHIOL 2 ONE; 5 METHOXY 4 [3 (3',4' DIMETHOXYPHENYL)ACRYOLYL] BENZO[D][1,3]OXATHIOL 2 ONE; 5 METHOXY 4 [3 (4' BROMOPHENYL)ACRYOLYL]BENZO[D] [1,3]OXATHIOL 2 ONE; 5 METHOXY 4 [3 (4' DIMETHYLAMINOPHENYL)ACRYOLYL]BENZO[D][1,3]OXATHIOL 2 ONE; 5 METHOXY 4 [3 (4' METHOXYPHENYL)ACRYOLYL]BENZO [D][1,3]OXATHIOL 2 ONE; 5 METHOXY 4 [3 (4' NITROPHENYL)ACRYOLYL]BENZO [D][1,3]OXATHIOL 2 ONE; 5 METHOXY 4 [3 {4' CHLOROPHENYL)ACRYOLYL]BENZO [D][1,3]OXATHIOL 2 ONE; BENZALDEHYDE; CHALCONE DERIVATIVE; UNCLASSIFIED DRUG;

ANTIFUNGAL ACTIVITY; ARTICLE; CANCER CELL CULTURE; CONTROLLED STUDY; CYTOTOXICITY; DRUG ACTIVITY; DRUG EFFECT; DRUG SYNTHESIS; HUMAN; HUMAN CELL; MICROCOCCUS LUTEUS; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; POLYMERIZATION; STAPHYLOCOCCUS AUREUS;

ACIDS; ANTI-BACTERIAL AGENTS; ANTINEOPLASTIC AGENTS; CATALYSIS; CHALCONES; DRUG SCREENING ASSAYS, ANTITUMOR; HELA CELLS; HUMANS; MICROBIAL SENSITIVITY TESTS; THIONES;

EID: 34248189167     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2006.12.014     Document Type: Article

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