Preparation of novel anthranilic acids as antibacterial agents: Extensive evaluation of structural and physical properties on antibacterial activity and human serum albumin affinity

Bioorganic and Medicinal Chemistry Letters

Volumn 17, Issue 11, 2007, Pages 3113-3116

  Thorarensen, Atli ^a   Li, Jianke ^a   Wakefield, Brian D ^a   Romero, Donna L ^a   Marotti, Keith R ^a   Sweeney, Michael T ^a   Zurenko, Gary E ^a   Sarver, Ronald W ^a  

^a PFIZER INC   (United States)

Author keywords

Antibacterial; HSA; Human serum albumin; Protein binding

Indexed keywords

ALBUMIN; ANTHRANILIC ACID DERIVATIVE;

ANTIBACTERIAL ACTIVITY; ARTICLE; BINDING AFFINITY; DRUG IDENTIFICATION; DRUG STRUCTURE; HUMAN;

ANTHRANILIC ACIDS; ANTI-BACTERIAL AGENTS; BACTERIA; HUMANS; SERUM ALBUMIN; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 34247855032     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2007.03.036     Document Type: Article

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