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Volumn 17, Issue 1, 2007, Pages 33-41

Development of a vesicular system for effective ocular delivery of acetazolamide A comprehensive approach and successful venture

Author keywords

Acetazolamide; Bioadhesive; Challenge test; Corneal penetration; Cytotoxicity; Introcular pressure; Microdialysis; Niosomes; Stability; Topical preparation

Indexed keywords

ACETAZOLAMIDE; BENZALKONIUM CHLORIDE; BORIC ACID; CARBOMER; DORZOLAMIDE; DORZOX; NIOSOME; NONIONIC SURFACTANT; PERBORATE SODIUM; POLYSORBATE 80; PRESERVATIVE; UNCLASSIFIED DRUG;

EID: 33847340168     PISSN: 17732247     EISSN: None     Source Type: Journal    
DOI: 10.1016/S1773-2247(07)50005-5     Document Type: Article
Times cited : (7)

References (55)
  • 1
    • 0037032464 scopus 로고    scopus 로고
    • Acetazolamide: Future perspective in topical glaucoma therapeutics
    • Kaur I. P., Smitha R., Aggarwal D., Kapil M. - Acetazolamide: future perspective in topical glaucoma therapeutics. - Int. J. Pharm., 248, 1-14, 2002.
    • (2002) Int. J. Pharm , vol.248 , pp. 1-14
    • Kaur, I.P.1    Smitha, R.2    Aggarwal, D.3    Kapil, M.4
  • 3
    • 0016242615 scopus 로고
    • Diffusional system for controlled release to the eye
    • Shell J. W., Baker R. - Diffusional system for controlled release to the eye. - Ann. Ophthalmol., 6, 1037-1043, 1974.
    • (1974) Ann. Ophthalmol , vol.6 , pp. 1037-1043
    • Shell, J.W.1    Baker, R.2
  • 4
    • 0022325722 scopus 로고
    • Review: Corneal penetration and ocular availability of drugs
    • Burstein N. L., Anderson J. A. - Review: Corneal penetration and ocular availability of drugs. - J. Ocul. Pharmacol., 1, 309-326, 1985.
    • (1985) J. Ocul. Pharmacol , vol.1 , pp. 309-326
    • Burstein, N.L.1    Anderson, J.A.2
  • 5
    • 0021717424 scopus 로고
    • Ophthalmic drug delivery systems
    • Shell J. W. - Ophthalmic drug delivery systems. - Surv. Ophthalmol., 29, 117-128, 1984.
    • (1984) Surv. Ophthalmol , vol.29 , pp. 117-128
    • Shell, J.W.1
  • 6
    • 0007790885 scopus 로고    scopus 로고
    • Ocular therapeutics and drug delivery: An overview
    • I.K. Reddy Ed, Technomic Publishing Company, Philadelphia, USA
    • Reddy I.K., Ganeshan M.G. - Ocular therapeutics and drug delivery: an overview. - In: Ocular Therapeutics and Drug Delivery: A Multidisciplinary Approach, I.K. Reddy Ed., Technomic Publishing Company, Philadelphia, USA, 1996, pp. 3-29.
    • (1996) Ocular Therapeutics and Drug Delivery: A Multidisciplinary Approach , pp. 3-29
    • Reddy, I.K.1    Ganeshan, M.G.2
  • 7
    • 0036269833 scopus 로고    scopus 로고
    • The ocular hypertension treatment study: A randomized trial determines that topical ocular hypotensive medication delays or prevents the onset of primary open-angle glaucoma
    • Kass M.A., Heuer D.K., Higginbotham E.J., Johnson C.A., Keltner J.L., Miller J.P., Parrish R.K., Wilson M.R., Gordon M.O. - The ocular hypertension treatment study: a randomized trial determines that topical ocular hypotensive medication delays or prevents the onset of primary open-angle glaucoma. - Arch. Ophthalmol., 120, 701-713, 2002.
    • (2002) Arch. Ophthalmol , vol.120 , pp. 701-713
    • Kass, M.A.1    Heuer, D.K.2    Higginbotham, E.J.3    Johnson, C.A.4    Keltner, J.L.5    Miller, J.P.6    Parrish, R.K.7    Wilson, M.R.8    Gordon, M.O.9
  • 8
    • 0014135426 scopus 로고
    • Carbonic anhydrase: Chemistry, physiology and inhibition
    • Maren T.H. - Carbonic anhydrase: Chemistry, physiology and inhibition. - Physiol. Rev., 47, 595-597, 1967.
    • (1967) Physiol. Rev , vol.47 , pp. 595-597
    • Maren, T.H.1
  • 9
    • 0023224380 scopus 로고
    • Carbonic anhydrase: General prospectives and advances in glaucoma research
    • Maren T.H. - Carbonic anhydrase: General prospectives and advances in glaucoma research. - Drug Dev. Res., 10, 255-276, 1987.
    • (1987) Drug Dev. Res , vol.10 , pp. 255-276
    • Maren, T.H.1
  • 10
    • 0034018870 scopus 로고    scopus 로고
    • Carbonic anhydrase inhibitors and their therapeutic potential
    • Supuran C.T., Scozzafava A. - Carbonic anhydrase inhibitors and their therapeutic potential. - Exp. Opin. Ther. Patents, 10, 575-600, 2000.
    • (2000) Exp. Opin. Ther. Patents , vol.10 , pp. 575-600
    • Supuran, C.T.1    Scozzafava, A.2
  • 11
    • 33847357909 scopus 로고    scopus 로고
    • Application of carbonic anhydrase inhibitors and activators in therapy
    • Supuran C.T., Scozzafava A. - Application of carbonic anhydrase inhibitors and activators in therapy. - Expert Opin. Ther. Patents, 14, 1-104, 2002.
    • (2002) Expert Opin. Ther. Patents , vol.14 , pp. 1-104
    • Supuran, C.T.1    Scozzafava, A.2
  • 12
    • 0017744637 scopus 로고
    • Carbonic anhydrase inhibitor side effects
    • Epstein D.L., Grant W.M. - Carbonic anhydrase inhibitor side effects. - Arch Opthamol., 95, 1378-1382, 1977.
    • (1977) Arch Opthamol , vol.95 , pp. 1378-1382
    • Epstein, D.L.1    Grant, W.M.2
  • 13
    • 0011441428 scopus 로고
    • Origination of side effects of acetazolamide
    • Gamm E. - Origination of side effects of acetazolamide. - Glaucoma, 6, 60-63, 1984.
    • (1984) Glaucoma , vol.6 , pp. 60-63
    • Gamm, E.1
  • 14
    • 10044235824 scopus 로고    scopus 로고
    • Novel approaches for topical delivery of acetazolamide
    • Singla A.K., Kaurl P., Garg A., Aggarwal D. - Novel approaches for topical delivery of acetazolamide. - Pharm Tech., 26, 24-34, 2002.
    • (2002) Pharm Tech , vol.26 , pp. 24-34
    • Singla, A.K.1    Kaurl, P.2    Garg, A.3    Aggarwal, D.4
  • 15
    • 0022518254 scopus 로고
    • Substituted sulfonamide carbonic anhydrase inhibitors with topical effects on intraocular pressure
    • Duffel M.W., Ing I.S., Segarra T.M., Dixson J.A., Barfknecht C.F., Schoenwald R.D. - Substituted sulfonamide carbonic anhydrase inhibitors with topical effects on intraocular pressure. - J. Med. Chem., 29, 1488-1494, 1986.
    • (1986) J. Med. Chem , vol.29 , pp. 1488-1494
    • Duffel, M.W.1    Ing, I.S.2    Segarra, T.M.3    Dixson, J.A.4    Barfknecht, C.F.5    Schoenwald, R.D.6
  • 16
    • 2042424475 scopus 로고    scopus 로고
    • Parasrampuria J. - Acetazolamide. - In: Analytical Profile of Drug Substances, H.G. Brittains Ed., 1, Academic Press, New York, 1993, pp. 1-28.
    • Parasrampuria J. - Acetazolamide. - In: Analytical Profile of Drug Substances, H.G. Brittains Ed., 1, Academic Press, New York, 1993, pp. 1-28.
  • 17
    • 0034633968 scopus 로고    scopus 로고
    • Application of in vivo confocal microscopy to the objective evaluation of occular irritation induced by surfactants
    • Furrer P., Plazonnet B., Mayer J.M., Gurny R. - Application of in vivo confocal microscopy to the objective evaluation of occular irritation induced by surfactants. - Int. J. Pharm., 207, 89-98, 2000.
    • (2000) Int. J. Pharm , vol.207 , pp. 89-98
    • Furrer, P.1    Plazonnet, B.2    Mayer, J.M.3    Gurny, R.4
  • 18
    • 55449102594 scopus 로고    scopus 로고
    • Functional differences in nucleoside and nucleobase transporters expressed on the rabbit corneal epithelial cell line (SIRC) and isolated rabbit cornea
    • Majumdar S., Tirucheri G.S., Pal D., Mitra A.K. - Functional differences in nucleoside and nucleobase transporters expressed on the rabbit corneal epithelial cell line (SIRC) and isolated rabbit cornea. - AAPS Pharm. Sci., 5, 145-158, 2003.
    • (2003) AAPS Pharm. Sci , vol.5 , pp. 145-158
    • Majumdar, S.1    Tirucheri, G.S.2    Pal, D.3    Mitra, A.K.4
  • 19
    • 0032970822 scopus 로고    scopus 로고
    • Permeability characteristics of novel mydriatic agents using an in vitro cell culture model that utilizes SIRC rabbit corneal cells
    • Goskonda V.R., Khan M.A., Hutak C.M., Reddy I.K. - Permeability characteristics of novel mydriatic agents using an in vitro cell culture model that utilizes SIRC rabbit corneal cells. - J. Pharm. Sci., 88, 180-184, 1999.
    • (1999) J. Pharm. Sci , vol.88 , pp. 180-184
    • Goskonda, V.R.1    Khan, M.A.2    Hutak, C.M.3    Reddy, I.K.4
  • 20
    • 0034763155 scopus 로고    scopus 로고
    • Transport of acyclovir easter prodrugs through rabbit cornea and SIRC-rabbit corneal epithelial cell line
    • Tak R.V., Pal D., Gao H., Dey S., Mitra A.K. - Transport of acyclovir easter prodrugs through rabbit cornea and SIRC-rabbit corneal epithelial cell line. - J.Pharm. Sci., 190, 1505-1515, 2001.
    • (2001) J.Pharm. Sci , vol.190 , pp. 1505-1515
    • Tak, R.V.1    Pal, D.2    Gao, H.3    Dey, S.4    Mitra, A.K.5
  • 21
    • 0142138814 scopus 로고    scopus 로고
    • In vitro effects of preserved or preservative-free antiglaucoma medications on human complement system
    • Blondin C., Hamard P., Cholley B., Haeffner-Cavaillon N., Baudouin C. - In vitro effects of preserved or preservative-free antiglaucoma medications on human complement system. - Curr. Eye Res., 27, 253-259, 2003.
    • (2003) Curr. Eye Res , vol.27 , pp. 253-259
    • Blondin, C.1    Hamard, P.2    Cholley, B.3    Haeffner-Cavaillon, N.4    Baudouin, C.5
  • 22
    • 0029758421 scopus 로고    scopus 로고
    • Side effcets of antiglaucomatous drugs on the ocular surface
    • Boudouin C. - Side effcets of antiglaucomatous drugs on the ocular surface. - Curr. Opin. Ophthalmol., 7, 80-86, 1996.
    • (1996) Curr. Opin. Ophthalmol , vol.7 , pp. 80-86
    • Boudouin, C.1
  • 23
    • 0030472676 scopus 로고    scopus 로고
    • Mechanisms of failure in glaucoma filtering surgery: A consequence of antiglaucomatous drugs?
    • Baudouin C. - Mechanisms of failure in glaucoma filtering surgery: a consequence of antiglaucomatous drugs? - Int. J. Clin. Pharmacol. Res., 16, 29-41, 1996.
    • (1996) Int. J. Clin. Pharmacol. Res , vol.16 , pp. 29-41
    • Baudouin, C.1
  • 24
    • 0344305387 scopus 로고    scopus 로고
    • Ishibashi T., Yokoin., Kinoshi S. - Comparison of the short-term effects on the human corneal surface of topical timolol maleate with and without benzalkonium chloride. - J. Glaucoma, 12, 486-490, 2003.
    • Ishibashi T., Yokoin., Kinoshi S. - Comparison of the short-term effects on the human corneal surface of topical timolol maleate with and without benzalkonium chloride. - J. Glaucoma, 12, 486-490, 2003.
  • 26
    • 0033966428 scopus 로고    scopus 로고
    • Comparison of the effects of preserved and unpreserved formulations of timolol in the ocular surface of albino rabbits
    • Pisella P.J., Fillacier K., Elena P.P., Debbasch C., Baudouin C. - Comparison of the effects of preserved and unpreserved formulations of timolol in the ocular surface of albino rabbits. - Ophthalmic Res., 32, 3-8, 2000.
    • (2000) Ophthalmic Res , vol.32 , pp. 3-8
    • Pisella, P.J.1    Fillacier, K.2    Elena, P.P.3    Debbasch, C.4    Baudouin, C.5
  • 27
    • 0035200807 scopus 로고    scopus 로고
    • Effects of common ophthalmic preservatives on ocular health
    • Nocker R. - Effects of common ophthalmic preservatives on ocular health. - Adv. Ther., 18, 205-215, 2001.
    • (2001) Adv. Ther , vol.18 , pp. 205-215
    • Nocker, R.1
  • 28
    • 85030522745 scopus 로고    scopus 로고
    • British Pharmacopoeia. - In: British Pharmacopoeia, II, The Stationary Office, London, 1999, A266-A268.
    • British Pharmacopoeia. - In: British Pharmacopoeia, II, The Stationary Office, London, 1999, A266-A268.
  • 29
    • 10044255251 scopus 로고    scopus 로고
    • Aggarwal D., Garg A.,Kaurl.P. - Development of a topical niosomal preparation of acetazolamide: preparation and evaluation. - J.Pharm. Pharmacol., 56, 1509-1517, 2004.
    • Aggarwal D., Garg A.,Kaurl.P. - Development of a topical niosomal preparation of acetazolamide: preparation and evaluation. - J.Pharm. Pharmacol., 56, 1509-1517, 2004.
  • 30
    • 85030513226 scopus 로고    scopus 로고
    • Indian Pharmacopoeia. - Controller of Publication, Delhi, 2, Appendix 9.5, 1996 A117-A124.
    • Indian Pharmacopoeia. - Controller of Publication, Delhi, 2, Appendix 9.5, 1996 A117-A124.
  • 31
    • 0026066853 scopus 로고
    • 5-(3-carboxymethoxyphenyl)-2-(4,5-dimenthylthiazoly)-3- (4-sulfophenyl) tetrazolium, inner salt (MTS) and related analogs of 3-(4,5-dimethylthiazolyl)-2,5-diphenyltetrazolium bromide (MTT) reducing to purple water-soluble formazans a cell-viability indicators
    • Barltrop J.A. - 5-(3-carboxymethoxyphenyl)-2-(4,5-dimenthylthiazoly)-3- (4-sulfophenyl) tetrazolium, inner salt (MTS) and related analogs of 3-(4,5-dimethylthiazolyl)-2,5-diphenyltetrazolium bromide (MTT) reducing to purple water-soluble formazans a cell-viability indicators. - Bioorg. & Med. Chem. Lett., 1, 611, 1991.
    • (1991) Bioorg. & Med. Chem. Lett , vol.1 , pp. 611
    • Barltrop, J.A.1
  • 32
    • 85030509121 scopus 로고    scopus 로고
    • Riss T.L., Moravec R.A. - Comparison of MTT, XTT, and a novel tetrazolium compound for MTS for in vitro proliferation and chemosensitivity assays. - Mol. Biol. Cell (Suppl.), 3, 184a, 1992.
    • Riss T.L., Moravec R.A. - Comparison of MTT, XTT, and a novel tetrazolium compound for MTS for in vitro proliferation and chemosensitivity assays. - Mol. Biol. Cell (Suppl.), 3, 184a, 1992.
  • 33
    • 85030516979 scopus 로고    scopus 로고
    • The Merck Index. - In: Merck and Co., Windholz M., NY, 1983, 8492.
    • The Merck Index. - In: Merck and Co., Windholz M., NY, 1983, 8492.
  • 34
    • 85030508543 scopus 로고    scopus 로고
    • Indian Pharmacopoeia. - Controller of Publication, Delhi, 1, 1996, 21.
    • Indian Pharmacopoeia. - Controller of Publication, Delhi, 1, 1996, 21.
  • 35
    • 31544437230 scopus 로고
    • Preparation of large unilamellar liposomes with high entrapment yield by rotary dialysis or agarose plug diffusion
    • G. Gregoridis Ed, CRC Press, Boca Raton
    • Gould-Fogerite S., Mannino R.J. - Preparation of large unilamellar liposomes with high entrapment yield by rotary dialysis or agarose plug diffusion. - In: Liposome Technology: Liposome Preparation and Related Techniques, G. Gregoridis Ed., CRC Press, Boca Raton, 1992, pp. 68-79.
    • (1992) Liposome Technology: Liposome Preparation and Related Techniques , pp. 68-79
    • Gould-Fogerite, S.1    Mannino, R.J.2
  • 36
    • 0028213925 scopus 로고
    • Improved ocular penetration of gentamicin by mucoadhesive polymer polycarbophil in the pigmented rabbit
    • Lehr C.M., Lee Y.H., Lee V.H. - Improved ocular penetration of gentamicin by mucoadhesive polymer polycarbophil in the pigmented rabbit. - Invest Ophthalmol. Vis. Sci., 35, 2809-2814, 1994.
    • (1994) Invest Ophthalmol. Vis. Sci , vol.35 , pp. 2809-2814
    • Lehr, C.M.1    Lee, Y.H.2    Lee, V.H.3
  • 37
    • 10044245291 scopus 로고    scopus 로고
    • Ophthalmic preparations
    • A.R. Gennaro Ed, Lipincott Williams and Wilkins, USA
    • Hecht G. - Ophthalmic preparations. - In: Remington: The Science and Practice of Pharmacy, A.R. Gennaro Ed., Lipincott Williams and Wilkins, USA, 2001, pp. 821-833.
    • (2001) Remington: The Science and Practice of Pharmacy , pp. 821-833
    • Hecht, G.1
  • 38
    • 85030510551 scopus 로고    scopus 로고
    • Riegelman S., Sorby D.L. - EENT preparations. - In: Husa's Pharmaceutics, E.W. Martin and J.E. Hoover Eds., Mack Publishing Company, Easton, PA, 1966, pp. 311-356.
    • Riegelman S., Sorby D.L. - EENT preparations. - In: Husa's Pharmaceutics, E.W. Martin and J.E. Hoover Eds., Mack Publishing Company, Easton, PA, 1966, pp. 311-356.
  • 39
    • 15844397498 scopus 로고
    • Moses Ed, Mosby, St. Louis, USA
    • Moses (Ed.). - Alder's Physiology of the Eye. - Mosby, St. Louis, USA, 1981.
    • (1981) Alder's Physiology of the Eye
  • 40
    • 0029809816 scopus 로고    scopus 로고
    • The preclinical pharmacology of dorzolamide hydrochloride, a topical carbonic anhydrase inhibitor
    • Surgue M.F. - The preclinical pharmacology of dorzolamide hydrochloride, a topical carbonic anhydrase inhibitor. - J. Ocul. Pharmacol. Ther, 12, 363-376, 1996.
    • (1996) J. Ocul. Pharmacol. Ther , vol.12 , pp. 363-376
    • Surgue, M.F.1
  • 42
    • 0017724862 scopus 로고
    • Short-term dose response characteristics of acetazolamide in man
    • FriedLand B.R., Mallonee J., Anderson D.R. - Short-term dose response characteristics of acetazolamide in man. - Arch. Ophthalmol., 95, 1809-1812, 1977.
    • (1977) Arch. Ophthalmol , vol.95 , pp. 1809-1812
    • FriedLand, B.R.1    Mallonee, J.2    Anderson, D.R.3
  • 44
    • 33645811993 scopus 로고
    • The pharmacokinetics of acetazolamide in relation to its use in the treatment of glaucoma and to its effects as an inhibitor of carbonic anhydrases
    • G. Rospe Ed, Pergamon, New York
    • Lehmann B., Linner E., Wristrand P.J. - The pharmacokinetics of acetazolamide in relation to its use in the treatment of glaucoma and to its effects as an inhibitor of carbonic anhydrases. - In: Schering Workshop in Pharmacokinetics, Advances in the Biosciences, G. Rospe Ed., Pergamon, New York, 1969, pp. 197-217.
    • (1969) Schering Workshop in Pharmacokinetics, Advances in the Biosciences , pp. 197-217
    • Lehmann, B.1    Linner, E.2    Wristrand, P.J.3
  • 47
    • 0035834185 scopus 로고    scopus 로고
    • Preparation and in vitro evaluation of liposomal/niosomal delivery systems for antipsoriatic drug dithranol
    • Agarwal R., Katare O.P., Vyas S.P. - Preparation and in vitro evaluation of liposomal/niosomal delivery systems for antipsoriatic drug dithranol. - Int. J. Pharm., 228, 43-52, 2001.
    • (2001) Int. J. Pharm , vol.228 , pp. 43-52
    • Agarwal, R.1    Katare, O.P.2    Vyas, S.P.3
  • 48
    • 0032902816 scopus 로고    scopus 로고
    • Encapsulation and stability of clofazamine liposomes
    • Patel V.B., Misra A.N. - Encapsulation and stability of clofazamine liposomes. - J. Microencapsul., 16, 357-367, 1999.
    • (1999) J. Microencapsul , vol.16 , pp. 357-367
    • Patel, V.B.1    Misra, A.N.2
  • 49
    • 0038025858 scopus 로고    scopus 로고
    • Hyaluronan is a key component in cryoprotection and formulation of targeted unilamellar liposomes. - Biochimica et Biophysica Acta (BBA)
    • Peer D., Florentin A., Margalit R. - Hyaluronan is a key component in cryoprotection and formulation of targeted unilamellar liposomes. - Biochimica et Biophysica Acta (BBA) Biomembranes, 1612, 76-82, 2003.
    • (2003) Biomembranes , vol.1612 , pp. 76-82
    • Peer, D.1    Florentin, A.2    Margalit, R.3
  • 52
    • 0036001084 scopus 로고    scopus 로고
    • Penetration enhancers and ocular bioadhesives: Two new avenues for ophthalmic drug delivery
    • Kaur I.P., Smitha R. - Penetration enhancers and ocular bioadhesives: two new avenues for ophthalmic drug delivery. - Drug Dev. Ind. Pharm., 28, 353-369, 2002.
    • (2002) Drug Dev. Ind. Pharm , vol.28 , pp. 353-369
    • Kaur, I.P.1    Smitha, R.2
  • 54
    • 0033966428 scopus 로고    scopus 로고
    • Comparison of the effects of preserved and unpreserved formulations of timolol in the ocular surface of albino rabbits
    • Pisella P.J., Fillacier K., Elena P.P., Debbasch C., Baudouin C. - Comparison of the effects of preserved and unpreserved formulations of timolol in the ocular surface of albino rabbits. - Ophthalmic Res., 32, 3-8, 2000.
    • (2000) Ophthalmic Res , vol.32 , pp. 3-8
    • Pisella, P.J.1    Fillacier, K.2    Elena, P.P.3    Debbasch, C.4    Baudouin, C.5


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