메뉴 건너뛰기




Volumn 12, Issue 3, 1996, Pages 363-376

The preclinical pharmacology of dorzolamide hydrochloride, a topical carbonic anhydrase inhibitor

Author keywords

[No Author keywords available]

Indexed keywords

6 HYDROXY 2 BENZOTHIAZOLESULFONAMIDE; 6 HYDROXY 2 BENZO[B]THIOPHENESULFONAMIDE; 6 PIVALOYLOXY 2 BENZOTHIAZOLESULFONAMIDE; ACETAZOLAMIDE; BENZOTHIAZOLE DERIVATIVE; CARBONATE DEHYDRATASE INHIBITOR; DICLOFENAMIDE; DORZOLAMIDE; ETHOXZOLAMIDE; L 651465; L 668931; METHAZOLAMIDE; SEZOLAMIDE; TIMOLOL; UNCLASSIFIED DRUG;

EID: 0029809816     PISSN: 10807683     EISSN: None     Source Type: Journal    
DOI: 10.1089/jop.1996.12.363     Document Type: Review
Times cited : (111)

References (41)
  • 1
    • 84989992371 scopus 로고
    • Carbonic anhydrase in the anterior uvea of the rabbit
    • Wistrand, P.J. Carbonic anhydrase in the anterior uvea of the rabbit. Acta Physiol. Scand., 24:144-148, 1951.
    • (1951) Acta Physiol. Scand. , vol.24 , pp. 144-148
    • Wistrand, P.J.1
  • 2
    • 0020590892 scopus 로고
    • Carbonic anhydrase distribution in the human and monkey eye by light and electron microscopy
    • Lütjen-Drecoll, E., Lönnerholm, G., and Eichhorn, M. Carbonic anhydrase distribution in the human and monkey eye by light and electron microscopy. Graefe's Arch. Clin. Exp. Ophthalmol., 220:285-291, 1983.
    • (1983) Graefe's Arch. Clin. Exp. Ophthalmol. , vol.220 , pp. 285-291
    • Lütjen-Drecoll, E.1    Lönnerholm, G.2    Eichhorn, M.3
  • 4
    • 0006872987 scopus 로고
    • The development of ideas concerning the role of carbonic anhydrase in the secretion of aqueous humor: Relation to the treatment of glaucoma
    • Drance, S.M. and Neufeld, A.H., eds., Grune and Stratton, Inc., Orlando
    • Maren, T.H. The development of ideas concerning the role of carbonic anhydrase in the secretion of aqueous humor: relation to the treatment of glaucoma. In Glaucoma: Applied Pharmacology in Medical Treatment, Drance, S.M. and Neufeld, A.H., eds., Grune and Stratton, Inc., Orlando, 1984, pp. 325-355.
    • (1984) Glaucoma: Applied Pharmacology in Medical Treatment , pp. 325-355
    • Maren, T.H.1
  • 5
    • 0002898371 scopus 로고
    • Decrease in intraocular pressure in man by a carbonic anhydrase inhibitor, Diamox
    • Becker, B. Decrease in intraocular pressure in man by a carbonic anhydrase inhibitor, Diamox. Am J. Ophthalmol., 37:13-14, 1954.
    • (1954) Am J. Ophthalmol. , vol.37 , pp. 13-14
    • Becker, B.1
  • 6
    • 0343616978 scopus 로고
    • Antiglaucoma drugs. Problem with carbonic anhydrase inhibition
    • Leopold, I.H., ed., C.V. Mosby, St. Louis
    • Grant, W.M. Antiglaucoma drugs. Problem with carbonic anhydrase inhibition. In Symposium on Ocular Therapy, Leopold, I.H., ed., C.V. Mosby, St. Louis, 1973, pp. 19-38.
    • (1973) Symposium on Ocular Therapy , pp. 19-38
    • Grant, W.M.1
  • 7
    • 0017744637 scopus 로고
    • Carbonic anhydrase inhibitor side effects. Serum chemical analysis
    • Epstein, D.L. and Grant, W.M. Carbonic anhydrase inhibitor side effects. Serum chemical analysis. Arch. Ophthalmol., 95:1378-1382, 1977.
    • (1977) Arch. Ophthalmol. , vol.95 , pp. 1378-1382
    • Epstein, D.L.1    Grant, W.M.2
  • 8
    • 0343343547 scopus 로고
    • L-645,151, a topically effective ocular hypotensive carbonic anhydrase inhibitor: Part 1. Biochemistry and metabolism
    • Schwam, H., Michelson, S.R., Sondey, J.M., and Smith, R.L. L-645,151, a topically effective ocular hypotensive carbonic anhydrase inhibitor: Part 1. Biochemistry and metabolism. Invest. Ophthalmol. Vis. Scl., 25 Suppl: 180, 1984.
    • (1984) Invest. Ophthalmol. Vis. Scl. , vol.25 , Issue.SUPPL. , pp. 180
    • Schwam, H.1    Michelson, S.R.2    Sondey, J.M.3    Smith, R.L.4
  • 10
    • 0023033313 scopus 로고
    • Ocular penetration and hypotensive activity of the topically applied carbonic anhydrase inhibitor L-645,151
    • Bar-Ilan, A., Pessah, N.I., and Maren, T.H. Ocular penetration and hypotensive activity of the topically applied carbonic anhydrase inhibitor L-645,151. J. Ocular Pharmacol., 2:109-120, 1986.
    • (1986) J. Ocular Pharmacol. , vol.2 , pp. 109-120
    • Bar-Ilan, A.1    Pessah, N.I.2    Maren, T.H.3
  • 12
    • 0023616162 scopus 로고
    • Effect of a topical carbonic anhydrase inhibitor, 6-hydroxybenzo[b]thiophene-2-sulfonamide, on intraocular pressure in normotensive subjects
    • Werner, E.B., Gerber, D.S., and Yoder, Y.L. Effect of a topical carbonic anhydrase inhibitor, 6-hydroxybenzo[b]thiophene-2-sulfonamide, on intraocular pressure in normotensive subjects. Can. J. Ophthalmol., 22:316-319, 1987.
    • (1987) Can. J. Ophthalmol. , vol.22 , pp. 316-319
    • Werner, E.B.1    Gerber, D.S.2    Yoder, Y.L.3
  • 13
    • 0009645290 scopus 로고
    • The eye: Topical carbonic anhydrase inhibitors
    • Dodgson, S.J., Tashian, R.E., Gros, G., and Carter, N.D., eds., Plenum Publishing Corp., New York
    • Lippa, E.A. The eye: topical carbonic anhydrase inhibitors. In The Carbonic Anhydrases. Dodgson, S.J., Tashian, R.E., Gros, G., and Carter, N.D., eds., Plenum Publishing Corp., New York, 1991, pp. 171-181.
    • (1991) The Carbonic Anhydrases , pp. 171-181
    • Lippa, E.A.1
  • 15
    • 0022852854 scopus 로고
    • Review: Topical ocular drug delivery: recent developments and future challenges
    • Lee, V.H.L. and Robinson, J.R. Review: topical ocular drug delivery: recent developments and future challenges. J. Ocular Pharmacol., 2:67-108, 1986.
    • (1986) J. Ocular Pharmacol. , vol.2 , pp. 67-108
    • Lee, V.H.L.1    Robinson, J.R.2
  • 19
    • 0024211865 scopus 로고
    • Local tolerance and activity of MK-927, a novel topical carbonic anhydrase inhibitor
    • Lippa, E.A., von Denffer, H.A., Hofmann, H.M., and Brunner-Ferber, F.L. Local tolerance and activity of MK-927, a novel topical carbonic anhydrase inhibitor. Arch. Ophthalmol., 106:1694-1696, 1988.
    • (1988) Arch. Ophthalmol. , vol.106 , pp. 1694-1696
    • Lippa, E.A.1    Von Denffer, H.A.2    Hofmann, H.M.3    Brunner-Ferber, F.L.4
  • 22
    • 0025256966 scopus 로고
    • The effect of MK-927, a topical carbonic anhydrase inhibitor, on IOP in glaucomatous monkeys
    • Wang, R.-F., Serie, J.B., Podos, S.M., and Sugrue, M.F. The effect of MK-927, a topical carbonic anhydrase inhibitor, on IOP in glaucomatous monkeys. Curr. Eye Res., 9:163-168, 1990.
    • (1990) Curr. Eye Res. , vol.9 , pp. 163-168
    • Wang, R.-F.1    Serie, J.B.2    Podos, S.M.3    Sugrue, M.F.4
  • 24
    • 0025046292 scopus 로고
    • A comparison of L-671,152 and MK-927, two topically effective ocular hypotensive carbonic anhydrase inhibitors, in experimental animals
    • Sugrue, M.F., Mallorga, P., Schwam, H., Baldwin, J.J., and Ponticello, G.S. A comparison of L-671,152 and MK-927, two topically effective ocular hypotensive carbonic anhydrase inhibitors, in experimental animals. Curr. Eye Res., 9:607-615, 1990.
    • (1990) Curr. Eye Res. , vol.9 , pp. 607-615
    • Sugrue, M.F.1    Mallorga, P.2    Schwam, H.3    Baldwin, J.J.4    Ponticello, G.S.5
  • 25
    • 0024539683 scopus 로고
    • Renal membrane-bound carbonic anhydrase. Purification and properties
    • Wistrand, P.J. and Knuuttila, K.-G. Renal membrane-bound carbonic anhydrase. Purification and properties. Kidney Intl., 35:851-859, 1989.
    • (1989) Kidney Intl. , vol.35 , pp. 851-859
    • Wistrand, P.J.1    Knuuttila, K.-G.2
  • 26
    • 0025798971 scopus 로고
    • Localization of carbonic anhydrase IV in a specific capillary bed of the human eye
    • Hageman, G.S., Zhu, X.L., Waheed, A., and Sly, W.S. Localization of carbonic anhydrase IV in a specific capillary bed of the human eye. Proc. Natl. Acad. Sci. USA, 88:2716-2720, 1991.
    • (1991) Proc. Natl. Acad. Sci. USA , vol.88 , pp. 2716-2720
    • Hageman, G.S.1    Zhu, X.L.2    Waheed, A.3    Sly, W.S.4
  • 28
  • 29
    • 85007752460 scopus 로고
    • The loci of carbonic anhydrase activity in the ciliary epithelium of the rabbit eye: Electrophysiological study with isolated ciliary epithelial bilayer
    • Murakami, M., Sears, M.L., Mori, N., Mead, A., Horio, B., and Yamada, E. The loci of carbonic anhydrase activity in the ciliary epithelium of the rabbit eye: electrophysiological study with isolated ciliary epithelial bilayer. Acta Histochem. Cytochem., 25:77-85, 1992.
    • (1992) Acta Histochem. Cytochem. , vol.25 , pp. 77-85
    • Murakami, M.1    Sears, M.L.2    Mori, N.3    Mead, A.4    Horio, B.5    Yamada, E.6
  • 31
    • 0027443910 scopus 로고
    • Chemical properties of carbonic anhydrase IV, the membrane-bound enzyme
    • Maren, T.H., Wynns, G.C., and Wistrand, P.J. Chemical properties of carbonic anhydrase IV, the membrane-bound enzyme. Mol. Pharmacol., 44:901-905, 1993.
    • (1993) Mol. Pharmacol. , vol.44 , pp. 901-905
    • Maren, T.H.1    Wynns, G.C.2    Wistrand, P.J.3
  • 32
    • 0025269576 scopus 로고
    • The ocular hypotensive effect of the topical carbonic anhydrase inhibitor L-671,152 in glaucomatous monkeys
    • Wang, R.-F., Serle, J.B., Podos, S.M., and Sugrue, M.F. The ocular hypotensive effect of the topical carbonic anhydrase inhibitor L-671,152 in glaucomatous monkeys. Arch. Ophthalmol., 108:511-513, 1990.
    • (1990) Arch. Ophthalmol. , vol.108 , pp. 511-513
    • Wang, R.-F.1    Serle, J.B.2    Podos, S.M.3    Sugrue, M.F.4
  • 33
    • 0025774167 scopus 로고
    • MK-507 (L-671,152), a topically active carbonic anhydrase inhibitor, reduces aqueous humor production in monkeys
    • Wang, R.-F., Serie, J.B., Podos, S.M., and Sugrue, M.F. MK-507 (L-671,152), a topically active carbonic anhydrase inhibitor, reduces aqueous humor production in monkeys. Arch. Ophthalmol., 109:1297-1299, 1991.
    • (1991) Arch. Ophthalmol. , vol.109 , pp. 1297-1299
    • Wang, R.-F.1    Serie, J.B.2    Podos, S.M.3    Sugrue, M.F.4
  • 34
    • 0019350144 scopus 로고
    • Effect of timolol on aqueous humor dynamics in the rabbit
    • Vareilles, P. and Lotti, V.J. Effect of timolol on aqueous humor dynamics in the rabbit. Ophthalmic Res., 13:72-79, 1981.
    • (1981) Ophthalmic Res. , vol.13 , pp. 72-79
    • Vareilles, P.1    Lotti, V.J.2
  • 35
    • 0000037568 scopus 로고
    • Carbonic anhydrase: Pharmacology of inhibitors and treatment of glaucoma
    • Sears, M.L., ed., Springer-Verlag, Berlin
    • Friedland, B.R. and Maren, T.H. Carbonic anhydrase: pharmacology of inhibitors and treatment of glaucoma. In Pharmacology of the Eye, Sears, M.L., ed., Springer-Verlag, Berlin, 1984, pp. 279-309.
    • (1984) Pharmacology of the Eye , pp. 279-309
    • Friedland, B.R.1    Maren, T.H.2
  • 36
    • 0026333066 scopus 로고
    • The effect of cyclooxygenase inhibition on the ocular hypotensive action of topical carbonic anhydrase inhibitors in rabbits
    • Sugrue, M.F. and O'Neill-Davis, L. The effect of cyclooxygenase inhibition on the ocular hypotensive action of topical carbonic anhydrase inhibitors in rabbits. J. Ocular Pharmacol., 7:201-211, 1991.
    • (1991) J. Ocular Pharmacol. , vol.7 , pp. 201-211
    • Sugrue, M.F.1    O'Neill-Davis, L.2
  • 37
    • 0015309358 scopus 로고
    • The oxygen supply to the retina, II. Effects of high intraocular pressure and of increased arterial carbon dioxide tension on uveal and retinal blood flow in cats. A study with radioactively labelled microspheres including flow determinations in brain and some other tissues
    • Alm, A. and Bill, A. The oxygen supply to the retina, II. Effects of high intraocular pressure and of increased arterial carbon dioxide tension on uveal and retinal blood flow in cats. A study with radioactively labelled microspheres including flow determinations in brain and some other tissues. Acta Physiol. Scand., 84:306-319, 1972.
    • (1972) Acta Physiol. Scand. , vol.84 , pp. 306-319
    • Alm, A.1    Bill, A.2
  • 38
    • 0015534943 scopus 로고
    • Ocular and optic nerve blood flow at normal and increased intraocular pressures in monkeys (Macaca irus): A study with radioactively labelled microspheres including flow determinations in brain and some other tissues
    • Alm, A. and Bill, A. Ocular and optic nerve blood flow at normal and increased intraocular pressures in monkeys (Macaca irus): a study with radioactively labelled microspheres including flow determinations in brain and some other tissues. Exp Eye Res., 15:15-29, 1973.
    • (1973) Exp Eye Res. , vol.15 , pp. 15-29
    • Alm, A.1    Bill, A.2
  • 39
    • 0011188865 scopus 로고
    • The effect of topical ocular hypotensive carbonic anhydrase inhibitors on regional ocular blood flow in albino rabbits
    • Sugrue, M.F. and Ludden, C. The effect of topical ocular hypotensive carbonic anhydrase inhibitors on regional ocular blood flow in albino rabbits. Invest. Ophthalmol. Vis. Sci., 32 Suppl:1186, 1991.
    • (1991) Invest. Ophthalmol. Vis. Sci. , vol.32 , Issue.SUPPL. , pp. 1186
    • Sugrue, M.F.1    Ludden, C.2
  • 40
    • 10144226988 scopus 로고
    • Preclinical findings in ocular irritation studies with dorzolamide hydrochloride
    • Gordon, L.R., Bailly, Y., Durand-Cavagna, G., and Peter, C.P. Preclinical findings in ocular irritation studies with dorzolamide hydrochloride. Exp. Eye Res., 59 Suppl 1:S29, 1994.
    • (1994) Exp. Eye Res. , vol.59 , Issue.1 SUPPL.
    • Gordon, L.R.1    Bailly, Y.2    Durand-Cavagna, G.3    Peter, C.P.4
  • 41
    • 0028928792 scopus 로고
    • The development of topical carbonic anhydrase inhibitors
    • Maren, T.H. The development of topical carbonic anhydrase inhibitors J. Glaucoma, 4:49-62, 1995.
    • (1995) J. Glaucoma , vol.4 , pp. 49-62
    • Maren, T.H.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.